FR2344545A1 - Amides d'acides (2-pyrimidinylthio)-alcanoiques ayant une activite antilipemique, procedes pour leur preparation et compositions pharmaceutiques les contenant - Google Patents

Amides d'acides (2-pyrimidinylthio)-alcanoiques ayant une activite antilipemique, procedes pour leur preparation et compositions pharmaceutiques les contenant

Info

Publication number
FR2344545A1
FR2344545A1 FR7707617A FR7707617A FR2344545A1 FR 2344545 A1 FR2344545 A1 FR 2344545A1 FR 7707617 A FR7707617 A FR 7707617A FR 7707617 A FR7707617 A FR 7707617A FR 2344545 A1 FR2344545 A1 FR 2344545A1
Authority
FR
France
Prior art keywords
pyrimidinylthio
preparation
methods
pharmaceutical compositions
compositions containing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7707617A
Other languages
English (en)
Other versions
FR2344545B1 (fr
Inventor
Carlo Scolastico
Giovanni Tronconi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Lpb Istituto Farmaceutico SpA
Original Assignee
Lpb Istituto Farmaceutico SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lpb Istituto Farmaceutico SpA filed Critical Lpb Istituto Farmaceutico SpA
Publication of FR2344545A1 publication Critical patent/FR2344545A1/fr
Application granted granted Critical
Publication of FR2344545B1 publication Critical patent/FR2344545B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32One oxygen, sulfur or nitrogen atom
    • C07D239/38One sulfur atom
FR7707617A 1976-03-17 1977-03-15 Amides d'acides (2-pyrimidinylthio)-alcanoiques ayant une activite antilipemique, procedes pour leur preparation et compositions pharmaceutiques les contenant Granted FR2344545A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT21317/76A IT1063074B (it) 1976-03-17 1976-03-17 Ammidi di acidi(z-pirimidiniltio)al canoici quali agent antilipemici

Publications (2)

Publication Number Publication Date
FR2344545A1 true FR2344545A1 (fr) 1977-10-14
FR2344545B1 FR2344545B1 (fr) 1980-03-21

Family

ID=11180012

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7707617A Granted FR2344545A1 (fr) 1976-03-17 1977-03-15 Amides d'acides (2-pyrimidinylthio)-alcanoiques ayant une activite antilipemique, procedes pour leur preparation et compositions pharmaceutiques les contenant

Country Status (14)

Country Link
JP (1) JPS52113983A (fr)
BE (1) BE852401A (fr)
CA (1) CA1081230A (fr)
CH (1) CH631169A5 (fr)
DE (1) DE2711149C3 (fr)
DK (1) DK143558C (fr)
ES (1) ES456902A1 (fr)
FR (1) FR2344545A1 (fr)
GB (1) GB1532195A (fr)
IT (1) IT1063074B (fr)
MX (1) MX4818E (fr)
NL (1) NL166933C (fr)
PH (1) PH14865A (fr)
SE (1) SE434743B (fr)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0073328A1 (fr) * 1981-08-20 1983-03-09 LPB Istituto Farmaceutico s.p.a. Dérivés de pyrimidine et de s-triazine avec une activité antilipidémique
FR2636064A1 (fr) * 1988-09-08 1990-03-09 Fabre Sa Pierre Thioformamidines, leur preparation et leur application en tant que medicaments
WO2002100836A2 (fr) * 2001-06-12 2002-12-19 Active Pass Pharmaceuticals, Inc. Composes, compositions et methodes de modulation de la production de beta-amyloide

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5810525Y2 (ja) * 1978-08-04 1983-02-25 三菱電機株式会社 小型電気掃除機
JPS59199673A (ja) * 1983-04-25 1984-11-12 Sumitomo Chem Co Ltd 含窒素複素環化合物、その製造法およびそれを有効成分とする有害生物防除剤

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0073328A1 (fr) * 1981-08-20 1983-03-09 LPB Istituto Farmaceutico s.p.a. Dérivés de pyrimidine et de s-triazine avec une activité antilipidémique
FR2636064A1 (fr) * 1988-09-08 1990-03-09 Fabre Sa Pierre Thioformamidines, leur preparation et leur application en tant que medicaments
EP0358571A1 (fr) * 1988-09-08 1990-03-14 Pierre Fabre Medicament Thioformamidines, leur préparation et leur application en tant que médicaments
WO2002100836A2 (fr) * 2001-06-12 2002-12-19 Active Pass Pharmaceuticals, Inc. Composes, compositions et methodes de modulation de la production de beta-amyloide
WO2002100836A3 (fr) * 2001-06-12 2003-05-15 Active Pass Pharmaceuticals In Composes, compositions et methodes de modulation de la production de beta-amyloide

Also Published As

Publication number Publication date
FR2344545B1 (fr) 1980-03-21
GB1532195A (en) 1978-11-15
DE2711149C3 (de) 1980-12-11
DK143558C (da) 1982-03-22
MX4818E (es) 1982-10-20
IT1063074B (it) 1985-02-11
NL7702821A (nl) 1977-09-20
JPS52113983A (en) 1977-09-24
CA1081230A (fr) 1980-07-08
SE434743B (sv) 1984-08-13
DK143558B (da) 1981-09-07
BE852401A (fr) 1977-07-01
ES456902A1 (es) 1978-01-16
DK114377A (da) 1977-09-18
DE2711149A1 (de) 1977-09-29
SE7702922L (sv) 1977-09-18
PH14865A (en) 1982-01-08
CH631169A5 (en) 1982-07-30
DE2711149B2 (fr) 1980-04-24
NL166933C (nl) 1981-10-15
JPS554746B2 (fr) 1980-01-31
NL166933B (nl) 1981-05-15

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