IT1063074B - Ammidi di acidi(z-pirimidiniltio)al canoici quali agent antilipemici - Google Patents

Ammidi di acidi(z-pirimidiniltio)al canoici quali agent antilipemici

Info

Publication number
IT1063074B
IT1063074B IT21317/76A IT2131776A IT1063074B IT 1063074 B IT1063074 B IT 1063074B IT 21317/76 A IT21317/76 A IT 21317/76A IT 2131776 A IT2131776 A IT 2131776A IT 1063074 B IT1063074 B IT 1063074B
Authority
IT
Italy
Prior art keywords
pyrimidinylti
canoics
acid amides
lipemic agents
lipemic
Prior art date
Application number
IT21317/76A
Other languages
English (en)
Inventor
Scolastico Carlo
Tronconi Giovanni
Original Assignee
Lpb Ist Farm
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lpb Ist Farm filed Critical Lpb Ist Farm
Priority to IT21317/76A priority Critical patent/IT1063074B/it
Priority to PH19485A priority patent/PH14865A/en
Priority to CA273,420A priority patent/CA1081230A/en
Priority to BE2055735A priority patent/BE852401A/xx
Priority to CH317377A priority patent/CH631169A5/it
Priority to DE2711149A priority patent/DE2711149C3/de
Priority to SE7702922A priority patent/SE434743B/xx
Priority to FR7707617A priority patent/FR2344545A1/fr
Priority to GB10995/77A priority patent/GB1532195A/en
Priority to DK114377A priority patent/DK143558C/da
Priority to MX775544U priority patent/MX4818E/es
Priority to JP2811277A priority patent/JPS52113983A/ja
Priority to ES456902A priority patent/ES456902A1/es
Priority to NL7702821.A priority patent/NL166933C/xx
Priority to US05/947,094 priority patent/US4188484A/en
Application granted granted Critical
Publication of IT1063074B publication Critical patent/IT1063074B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32One oxygen, sulfur or nitrogen atom
    • C07D239/38One sulfur atom
IT21317/76A 1976-03-17 1976-03-17 Ammidi di acidi(z-pirimidiniltio)al canoici quali agent antilipemici IT1063074B (it)

Priority Applications (15)

Application Number Priority Date Filing Date Title
IT21317/76A IT1063074B (it) 1976-03-17 1976-03-17 Ammidi di acidi(z-pirimidiniltio)al canoici quali agent antilipemici
PH19485A PH14865A (en) 1976-03-17 1977-02-23 (2-pyrimidinyl-thio)alkanoic acid amides and their preparation
CA273,420A CA1081230A (en) 1976-03-17 1977-03-08 (2-pyrimidinyl-thio) alkanoic acid amides and their preparation
CH317377A CH631169A5 (en) 1976-03-17 1977-03-14 Method for preparing amides of (2-pyrimidinylthio)-alkanoic acids, having an antilipemic activity
BE2055735A BE852401A (fr) 1976-03-17 1977-03-14 Amides d'acides (2-pyrimidinylthio)-alcanoiques ayant une activite antilipemique
SE7702922A SE434743B (sv) 1976-03-17 1977-03-15 Forfarande for framstellning av (2-pyrimidinyl-tio)-alkansyraamider
DE2711149A DE2711149C3 (de) 1976-03-17 1977-03-15 N-Substituierte[4-Chlor-6-(23-xylidino)-2· pyrimidinyl- thio] essigsäureamide sowie Verfahren zu deren Herstellung
FR7707617A FR2344545A1 (fr) 1976-03-17 1977-03-15 Amides d'acides (2-pyrimidinylthio)-alcanoiques ayant une activite antilipemique, procedes pour leur preparation et compositions pharmaceutiques les contenant
GB10995/77A GB1532195A (en) 1976-03-17 1977-03-15 (2-pyrimidinyl-thio)-alkanoic acid amides and their preparation
DK114377A DK143558C (da) 1976-03-17 1977-03-16 Analogifremgangsmaade til fremstilling af n-substituerede (4-chlor-6-(2,3-xylidino)-2-pyrimidinyl-thio)acetamider
MX775544U MX4818E (es) 1976-03-17 1977-03-16 Procedimiento para la preparacion de amidas de acidos(2-pirimidiniltio)alcanoicos
JP2811277A JPS52113983A (en) 1976-03-17 1977-03-16 *22pyrimidinyllthioalkanoneamide*its production and antiilipemic agent containing same
ES456902A ES456902A1 (es) 1976-03-17 1977-03-16 Procedimiento para la preparacion de amidas de acidos (2-pi-rimidiniltio) alcanoicos.
NL7702821.A NL166933C (nl) 1976-03-17 1977-03-16 Werkwijze ter bereiding van een farmaceutisch preparaat met anti-lipemische werking, alsmede de aldus vervaar- digde farmaceutische voorwerpen en werkwijze ter berei- ding van (2-pyrimidinylthio)-alkaanzuuramide- -verbindingen.
US05/947,094 US4188484A (en) 1976-03-17 1978-09-29 (2-Pyrimidinyl-thio)-alkanoic acid amides and their preparation

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT21317/76A IT1063074B (it) 1976-03-17 1976-03-17 Ammidi di acidi(z-pirimidiniltio)al canoici quali agent antilipemici

Publications (1)

Publication Number Publication Date
IT1063074B true IT1063074B (it) 1985-02-11

Family

ID=11180012

Family Applications (1)

Application Number Title Priority Date Filing Date
IT21317/76A IT1063074B (it) 1976-03-17 1976-03-17 Ammidi di acidi(z-pirimidiniltio)al canoici quali agent antilipemici

Country Status (14)

Country Link
JP (1) JPS52113983A (it)
BE (1) BE852401A (it)
CA (1) CA1081230A (it)
CH (1) CH631169A5 (it)
DE (1) DE2711149C3 (it)
DK (1) DK143558C (it)
ES (1) ES456902A1 (it)
FR (1) FR2344545A1 (it)
GB (1) GB1532195A (it)
IT (1) IT1063074B (it)
MX (1) MX4818E (it)
NL (1) NL166933C (it)
PH (1) PH14865A (it)
SE (1) SE434743B (it)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5810525Y2 (ja) * 1978-08-04 1983-02-25 三菱電機株式会社 小型電気掃除機
IT1211096B (it) * 1981-08-20 1989-09-29 Lpb Ist Farm Pirimidine e s.triazinici adattivita' ipolipidemizzante.
JPS59199673A (ja) * 1983-04-25 1984-11-12 Sumitomo Chem Co Ltd 含窒素複素環化合物、その製造法およびそれを有効成分とする有害生物防除剤
FR2636064B1 (fr) * 1988-09-08 1990-12-07 Fabre Sa Pierre Thioformamidines, leur preparation et leur application en tant que medicaments
EP1399426A2 (en) * 2001-06-12 2004-03-24 Active Pass Pharmaceuticals, Inc. Compounds, compositions and methods for modulating beta-amyloid production

Also Published As

Publication number Publication date
FR2344545B1 (it) 1980-03-21
GB1532195A (en) 1978-11-15
DE2711149C3 (de) 1980-12-11
DK143558C (da) 1982-03-22
MX4818E (es) 1982-10-20
NL7702821A (nl) 1977-09-20
JPS52113983A (en) 1977-09-24
CA1081230A (en) 1980-07-08
SE434743B (sv) 1984-08-13
DK143558B (da) 1981-09-07
BE852401A (fr) 1977-07-01
ES456902A1 (es) 1978-01-16
DK114377A (da) 1977-09-18
DE2711149A1 (de) 1977-09-29
SE7702922L (sv) 1977-09-18
FR2344545A1 (fr) 1977-10-14
PH14865A (en) 1982-01-08
CH631169A5 (en) 1982-07-30
DE2711149B2 (it) 1980-04-24
NL166933C (nl) 1981-10-15
JPS554746B2 (it) 1980-01-31
NL166933B (nl) 1981-05-15

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