FR2324633A1 - Pyrazoles substitues et leur preparation - Google Patents

Pyrazoles substitues et leur preparation

Info

Publication number
FR2324633A1
FR2324633A1 FR7534913A FR7534913A FR2324633A1 FR 2324633 A1 FR2324633 A1 FR 2324633A1 FR 7534913 A FR7534913 A FR 7534913A FR 7534913 A FR7534913 A FR 7534913A FR 2324633 A1 FR2324633 A1 FR 2324633A1
Authority
FR
France
Prior art keywords
pyrazoles
substitute
preparation
substitute pyrazoles
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
FR7534913A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia and Upjohn Co
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of FR2324633A1 publication Critical patent/FR2324633A1/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16Halogen atoms or nitro radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FR7534913A 1974-11-15 1975-11-14 Pyrazoles substitues et leur preparation Withdrawn FR2324633A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US52423174A 1974-11-15 1974-11-15

Publications (1)

Publication Number Publication Date
FR2324633A1 true FR2324633A1 (fr) 1977-04-15

Family

ID=24088332

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7534913A Withdrawn FR2324633A1 (fr) 1974-11-15 1975-11-14 Pyrazoles substitues et leur preparation

Country Status (14)

Country Link
US (1) US4072498A (fr)
JP (1) JPS5182269A (fr)
BE (1) BE835604A (fr)
BR (1) BR7507364A (fr)
CH (1) CH629364A5 (fr)
DE (1) DE2550566A1 (fr)
FR (1) FR2324633A1 (fr)
GB (1) GB1483162A (fr)
IT (1) IT1052194B (fr)
NZ (1) NZ178996A (fr)
PH (1) PH12819A (fr)
PL (1) PL101829B1 (fr)
SU (2) SU613722A3 (fr)
ZA (1) ZA756627B (fr)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2901593A1 (de) * 1979-01-17 1980-08-07 Basf Ag N-azolylessigsaeureanilide
DE3041702A1 (de) * 1980-11-05 1982-06-09 Basf Ag, 6700 Ludwigshafen Verfahren zur bekaempfung unerwuenschten pflanzenwuchses mit 2-aryloxy-2-azolylalkancarbonsaeureamiden, diese enthaltende herbizide und verfahren zu ihrer herstellung
US4515623A (en) * 1981-10-09 1985-05-07 Basf Aktiengesellschaft Control of unwanted plant growth with 2-aryloxy-2-azolylalkanecarboxamides
US4874871A (en) * 1987-03-25 1989-10-17 Syntex (U.S.A.) Inc. Process for preparing (+)-2,3-Dihydro-1H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds
US4870095A (en) * 1988-06-13 1989-09-26 Sterling Drug, Inc. 1H-pyrazole-1-alkanamides, antiarrhythmic compositions and use
JP2784925B2 (ja) * 1988-09-07 1998-08-13 日本農薬株式会社 3又は5−フェニルピラゾール類又はその塩及び除草剤
US4898880A (en) * 1989-03-22 1990-02-06 Sterling Drug Inc. N-(heterocycle)alkyl)-1H-pyrazole-1-alkanamides as antiarrhythmic agents, compositions and use
US4988725A (en) * 1989-03-22 1991-01-29 Sterling Drug Inc. 1H-pyrazole-1-(branched)alkanamides as antiarrhythmic agents, compositions and use
US4925857A (en) * 1989-03-22 1990-05-15 Sterling Drug Inc. Pyridinyl-1H-pyrazole-1-alkanamides as antiarrhythmic agents
US4916150A (en) * 1989-03-22 1990-04-10 Sterling Drug Inc. 1H-pyrazole-1-alkanamines antiarrhythmic compositions and use
US4888352A (en) * 1989-03-22 1989-12-19 Sterling Drug Inc. 3,4, or 5-aryl-1H-pyrazole-1-alkanamides as antiarrhythmic agents, compositions and use
US4994482A (en) * 1989-07-31 1991-02-19 Bristol-Myers Squibb Company Arylpyrazol derivatives as anti-platelet agents, compositions and use
JPH0393774A (ja) * 1989-09-07 1991-04-18 Nippon Nohyaku Co Ltd 3又は5―フェニルピラゾール類又はその塩及び除草剤
US5366987A (en) * 1991-08-22 1994-11-22 Warner-Lambert Company Isoxazolyl-substituted alkyl amide ACAT inhibitors
US5532416A (en) * 1994-07-20 1996-07-02 Monsanto Company Benzoyl derivatives and synthesis thereof
FR2682379B1 (fr) 1991-10-09 1994-02-11 Rhone Poulenc Agrochimie Nouveaux phenylpyrazoles fongicides.
FR2690440B1 (fr) * 1992-04-27 1995-05-19 Rhone Poulenc Agrochimie Arylpyrazoles fongicides.
IL112014A (en) * 1993-12-24 1999-10-28 Rhone Poulenc Agrochimie 1,3-Oxazin-4-one derivatives and herbicides containing the same
US5880290A (en) * 1994-01-31 1999-03-09 Monsanto Company Preparation of substituted 3-aryl-5-haloalkyl-pyrazoles having herbicidal activity
US5869688A (en) * 1994-07-20 1999-02-09 Monsanto Company Preparation of substituted 3-aryl-5-haloalkyl-pyrazoles having herbicidal activity
US5698708A (en) * 1996-06-20 1997-12-16 Monsanto Company Preparation of substituted 3-aryl-5-haloalkyl-pyrazoles having herbicidal activity
DE19744026A1 (de) * 1997-10-06 1999-04-08 Hoechst Marion Roussel De Gmbh Pyrazol-Derivate, ihre Herstellung und ihre Verwendung in Arzneimitteln
RU2001129155A (ru) 1999-03-26 2003-08-10 Еро-Сельтик С.А. (Lu) Соединения с арильными заместителями (варианты), фармацевтическая композиция и способ лечения расстройства, чувствительного к блокаде натриевых каналов у млекопитающего, способ лечения, профилактики различных заболеваний или уменьшения интенсивности гибели или потери нейронов (варианты), способ облегчения или предупреждения эпилептических припадков у животного (варианты), соединение - радиоактивный лиганд для участка связывания в натриевом канале
HU229371B1 (en) * 2000-03-24 2013-11-28 Euro Celtique Sa Aryl substituted pyrazoles, triazoles and tetrazoles, and the use thereof
KR100613212B1 (ko) * 2001-12-20 2006-08-21 가부시키가이샤 에스디에스 바이오테크 신규의 치환된 피라졸 유도체, 그의 제조 방법 및 그것을함유하는 제초제 조성물
CN103265537B (zh) * 2013-05-14 2015-05-27 浙江医药高等专科学校 抗肿瘤化合物、其制备方法和用途
GB201616439D0 (en) * 2016-09-28 2016-11-09 Mironid Limited Compounds and uses
WO2019081485A1 (fr) 2017-10-26 2019-05-02 Bayer Cropscience Aktiengesellschaft Pyrazoles substitués, leurs sels et leur utilisation comme agents herbicides
WO2019081477A1 (fr) 2017-10-26 2019-05-02 Bayer Cropscience Aktiengesellschaft Pyrazoles substitués, leurs sels et leur utilisation comme agents herbicides
GB201805527D0 (en) 2018-04-04 2018-05-16 Mironid Ltd Compounds and their use as pde4 activators
CN110963957B (zh) * 2018-09-28 2021-10-22 深圳恩多凯医药科技有限公司 N-芳香酰胺类化合物及其制备方法和用途

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH485736A (de) * 1967-04-26 1970-02-15 Agripat Sa Verfahren zur Herstellung halogensubstituierter Imidazol-Derivate
BE795881A (fr) * 1972-02-23 1973-08-23 Upjohn Co Tribromopyrazoles et leur preparation

Also Published As

Publication number Publication date
IT1052194B (it) 1981-06-20
CH629364A5 (de) 1982-04-30
BE835604A (fr) 1976-05-14
BR7507364A (pt) 1976-08-10
JPS5182269A (fr) 1976-07-19
PL101829B1 (pl) 1979-02-28
GB1483162A (en) 1977-08-17
AU8595775A (en) 1977-04-28
PH12819A (en) 1979-08-31
SU581838A3 (ru) 1977-11-25
SU613722A3 (ru) 1978-06-30
NZ178996A (en) 1978-06-02
US4072498A (en) 1978-02-07
ZA756627B (en) 1977-05-25
DE2550566A1 (de) 1976-05-20

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Legal Events

Date Code Title Description
ST Notification of lapse