FR2288526A1 - Nouveaux derives de l'acide penicillanique utiles notamment pour le traitement des infections bacteriennes et leur procede de preparation - Google Patents

Nouveaux derives de l'acide penicillanique utiles notamment pour le traitement des infections bacteriennes et leur procede de preparation

Info

Publication number
FR2288526A1
FR2288526A1 FR7532049A FR7532049A FR2288526A1 FR 2288526 A1 FR2288526 A1 FR 2288526A1 FR 7532049 A FR7532049 A FR 7532049A FR 7532049 A FR7532049 A FR 7532049A FR 2288526 A1 FR2288526 A1 FR 2288526A1
Authority
FR
France
Prior art keywords
treatment
preparation process
bacterial infections
penicillanic acid
new derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
FR7532049A
Other languages
English (en)
Inventor
Cornelis Adrianus Bruynes
Johannes Karel Van Der Drift
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gist Brocades NV
Original Assignee
Gist Brocades NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gist Brocades NV filed Critical Gist Brocades NV
Publication of FR2288526A1 publication Critical patent/FR2288526A1/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
    • C07F9/36—Amides thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/06—Phosphorus compounds without P—C bonds
    • C07F9/22—Amides of acids of phosphorus
    • C07F9/24—Esteramides
    • C07F9/2454—Esteramides the amide moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/2479—Compounds containing the structure P(=X)n-N-acyl, P(=X)n-N-heteroatom, P(=X)n-N-CN (X = O, S, Se; n = 0, 1)
    • C07F9/2487—Compounds containing the structure P(=X)n-N-acyl, P(=X)n-N-heteroatom, P(=X)n-N-CN (X = O, S, Se; n = 0, 1) containing the structure P(=X)n-N-C(=X) (X = O, S, Se; n = 0, 1)
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/44—Amides thereof
    • C07F9/4461—Amides thereof the amide moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4484—Compounds containing the structure C-P(=X)(N-acyl)-X, C-P(=X)(N-heteroatom)-X or C-P(=X)(N-CN)-X (X = O, S, Se)
    • C07F9/4492—Compounds containing the structure P(=X)(N-C(=X)-) (X = O, S, Se)
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • C07F9/65611—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings containing the ring system (X = CH2, O, S, NH) optionally with an additional double bond and/or substituents, e.g. penicillins and analogs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR7532049A 1974-10-21 1975-10-20 Nouveaux derives de l'acide penicillanique utiles notamment pour le traitement des infections bacteriennes et leur procede de preparation Withdrawn FR2288526A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB45480/74A GB1523278A (en) 1974-10-21 1974-10-21 Penicillanic acid derivatives

Publications (1)

Publication Number Publication Date
FR2288526A1 true FR2288526A1 (fr) 1976-05-21

Family

ID=10437377

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7532049A Withdrawn FR2288526A1 (fr) 1974-10-21 1975-10-20 Nouveaux derives de l'acide penicillanique utiles notamment pour le traitement des infections bacteriennes et leur procede de preparation

Country Status (19)

Country Link
US (1) US4067986A (fr)
JP (2) JPS5165793A (fr)
AT (1) AT349631B (fr)
BE (1) BE834679A (fr)
CS (1) CS203096B2 (fr)
DE (1) DE2546910C3 (fr)
DK (1) DK471375A (fr)
ES (2) ES441922A1 (fr)
FI (1) FI59803C (fr)
FR (1) FR2288526A1 (fr)
GB (1) GB1523278A (fr)
HU (1) HU170700B (fr)
IE (1) IE42612B1 (fr)
IT (1) IT1047205B (fr)
LU (1) LU73606A1 (fr)
NL (1) NL164039C (fr)
NO (1) NO753519L (fr)
PL (2) PL108190B1 (fr)
SE (2) SE7511732L (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5283587A (en) * 1976-01-01 1977-07-12 Gist Brocades Nv Heterocyclic compound of novel substance
US4177189A (en) * 1977-06-01 1979-12-04 Gist-Brocades N.V. Process for the preparation of hydroxyphosphinylureidobenzylpenicillins

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1184665A (en) * 1966-12-28 1970-03-18 Astra Ab Penicillins
GB1241844A (en) * 1968-08-23 1971-08-04 Beecham Group Ltd Penicillins
US3939149A (en) * 1970-05-25 1976-02-17 Bayer Aktiengesellschaft Ureidoacetamido-penicillins
GB1430074A (en) * 1972-07-13 1976-03-31 Beecham Group Ltd Penicillins
GB1464551A (en) * 1973-02-08 1977-02-16 Gist Brocades Nv Alpha-substituted amino-phenylacetamido penicillanic acid and cephalosporanic acid derivatives methods for their preparation and their use
US3935189A (en) * 1973-05-04 1976-01-27 Beecham Group Limited Penicillins

Also Published As

Publication number Publication date
PL108190B1 (pl) 1980-03-31
ES441922A1 (es) 1977-03-16
NO753519L (fr) 1976-04-22
SE7809050L (sv) 1978-08-28
JPS5387393A (en) 1978-08-01
PL103373B1 (pl) 1979-06-30
US4067986A (en) 1978-01-10
DE2546910A1 (de) 1976-04-22
GB1523278A (en) 1978-08-31
BE834679A (fr) 1976-04-20
ES444212A1 (es) 1977-05-01
CS203096B2 (en) 1981-02-27
FI59803B (fi) 1981-06-30
NL164039B (nl) 1980-06-16
DE2546910B2 (de) 1978-02-23
ATA794975A (de) 1978-09-15
LU73606A1 (fr) 1977-05-24
JPS5165793A (fr) 1976-06-07
IE42612B1 (en) 1980-09-10
AT349631B (de) 1979-04-10
FI59803C (fi) 1981-10-12
SE7511732L (sv) 1976-04-22
FI752924A (fr) 1976-04-22
DK471375A (da) 1976-04-22
IE42612L (en) 1976-04-21
DE2546910C3 (de) 1978-09-28
NL164039C (nl) 1980-11-17
NL7512264A (nl) 1976-04-23
IT1047205B (it) 1980-09-10
HU170700B (fr) 1977-08-28

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Legal Events

Date Code Title Description
RE Withdrawal of published application