FR2240009A1 - 3-(5-Nitro-2-imidazolyl)pyrazoles - antibacterials antifungals and antiprotozoals useful in veterinary medicine - Google Patents

3-(5-Nitro-2-imidazolyl)pyrazoles - antibacterials antifungals and antiprotozoals useful in veterinary medicine

Info

Publication number
FR2240009A1
FR2240009A1 FR7427017A FR7427017A FR2240009A1 FR 2240009 A1 FR2240009 A1 FR 2240009A1 FR 7427017 A FR7427017 A FR 7427017A FR 7427017 A FR7427017 A FR 7427017A FR 2240009 A1 FR2240009 A1 FR 2240009A1
Authority
FR
France
Prior art keywords
alkyl
antiprotozoals
antifungals
antibacterials
useful
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7427017A
Other languages
French (fr)
Other versions
FR2240009B1 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of FR2240009A1 publication Critical patent/FR2240009A1/en
Application granted granted Critical
Publication of FR2240009B1 publication Critical patent/FR2240009B1/fr
Granted legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/116Heterocyclic compounds

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Polymers & Plastics (AREA)
  • Animal Husbandry (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Food Science & Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Cpds. of formula (I): where R = 1-3C alkyl, 1-3C haloalkyl or 1-3C hydroxyalkyl; R1 = -NR3R4 or -N=CR5-X; R2 = H, -CN, -COOH or -CONHR6; R3, R4 = same or different H, 1-3C alkyl, 1-4C alkanoyl or -SO2N(CH3)2; R5 = H or 1-3C alkyl; X = -OR7, phenyl, -CH=CH-CH3, -CH=CH-C6H5, -CCl3, 2-furyl, 3-pyridyl, 3,4-methylenedioxyphenyl, -NH-NH-1-4C alkyl or -NR8R9; R6 = H or 1-4C alkanoyl; R7 = 1-8C alkyl, 2-5C alkenyl or 1-3C haloalkyl; R8, R9 = same or different 1-3C alkyl. Specif. claimed are (I) where R2 = CN and (a) R=CH3 and R1 = -NH2, -N=CH-OCH3 and -N=CH-OC4H9 and (B) R = C2H5 and R1 = -NH2. (I) are useful as antibacterials, antifungals and antiprotozoals active against Escherichia coli, Pasteurella multocida, Salmonella Typhimurium, Treponema hyodysentereae and coccidiosis etc.
FR7427017A 1973-08-02 1974-08-02 3-(5-Nitro-2-imidazolyl)pyrazoles - antibacterials antifungals and antiprotozoals useful in veterinary medicine Granted FR2240009A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US38513673A 1973-08-02 1973-08-02

Publications (2)

Publication Number Publication Date
FR2240009A1 true FR2240009A1 (en) 1975-03-07
FR2240009B1 FR2240009B1 (en) 1978-07-28

Family

ID=23520163

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7427017A Granted FR2240009A1 (en) 1973-08-02 1974-08-02 3-(5-Nitro-2-imidazolyl)pyrazoles - antibacterials antifungals and antiprotozoals useful in veterinary medicine

Country Status (18)

Country Link
JP (1) JPS5047978A (en)
AR (3) AR203854A1 (en)
AT (1) AT337691B (en)
BE (1) BE818417A (en)
BR (1) BR7406317D0 (en)
DD (1) DD112759A5 (en)
DE (1) DE2431775A1 (en)
DK (1) DK410874A (en)
ES (1) ES428914A0 (en)
FR (1) FR2240009A1 (en)
IL (1) IL45073A (en)
IT (1) IT1049204B (en)
NL (1) NL7410033A (en)
PL (5) PL96804B1 (en)
RO (1) RO63973A (en)
SE (1) SE7409957L (en)
SU (2) SU565630A3 (en)
ZA (1) ZA743887B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014189947A1 (en) * 2013-05-20 2014-11-27 University Of Washington Through Its Center For Commercialization 5-aminopyrazole-4-carboxamide inhibitors of cdpk1 from t. gondii and c. parvum

Also Published As

Publication number Publication date
NL7410033A (en) 1975-02-04
DD112759A5 (en) 1975-05-05
ES428914A0 (en) 1977-02-01
AT337691B (en) 1977-07-11
IL45073A (en) 1977-07-31
ZA743887B (en) 1975-06-25
FR2240009B1 (en) 1978-07-28
BE818417A (en) 1975-02-03
DE2431775A1 (en) 1975-02-20
DK410874A (en) 1975-04-01
BR7406317D0 (en) 1975-05-20
AR205814A1 (en) 1976-06-07
PL96804B1 (en) 1978-01-31
RO63973A (en) 1978-09-15
AU7052874A (en) 1976-01-08
PL94238B1 (en) 1977-07-30
ATA627474A (en) 1976-11-15
SE7409957L (en) 1975-02-03
IL45073A0 (en) 1974-09-10
SU565630A3 (en) 1977-07-15
JPS5047978A (en) 1975-04-28
IT1049204B (en) 1981-01-20
PL92429B1 (en) 1977-04-30
AR203854A1 (en) 1975-10-31
AR204130A1 (en) 1975-11-20
SU582758A3 (en) 1977-11-30
PL91696B1 (en) 1977-03-31
PL96805B1 (en) 1978-01-31

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Legal Events

Date Code Title Description
ST Notification of lapse