FR15C0073I1 - - Google Patents

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Publication number
FR15C0073I1
FR15C0073I1 FR15C0073C FR15C0073I1 FR 15C0073 I1 FR15C0073 I1 FR 15C0073I1 FR 15C0073 C FR15C0073 C FR 15C0073C FR 15C0073 I1 FR15C0073 I1 FR 15C0073I1
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FR
France
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French (fr)
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34280181&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FR15C0073(I1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Publication of FR15C0073I1 publication Critical patent/FR15C0073I1/fr
Application filed filed Critical
Application granted granted Critical
Publication of FR15C0073I2 publication Critical patent/FR15C0073I2/fr
Active legal-status Critical Current

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/675Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
FR15C0073C 2003-09-03 2015-10-21 Combinaison d'un inhibiteur non-nucleosidique de la transcriptase inverse (nnrti) contenant une pyrimidine avec un inhibiteur nucleosidique de la transcriptase inverse (nrti) Active FR15C0073I2 (fr)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US49977103P 2003-09-03 2003-09-03
EP03103275 2003-09-03
EP03103319 2003-09-08
EP03103335 2003-09-10
EP03103668 2003-10-02
US50848603P 2003-10-03 2003-10-03
EP04787096.9A EP1663240B2 (en) 2003-09-03 2004-09-03 Combinations of a pyrimidine containing nnrti with rt inhibitors
PCT/EP2004/052028 WO2005021001A1 (en) 2003-09-03 2004-09-03 Combinations of a pyrimidine containing nnrti with rt inhibitors

Publications (2)

Publication Number Publication Date
FR15C0073I1 true FR15C0073I1 (uk) 2015-04-12
FR15C0073I2 FR15C0073I2 (fr) 2016-02-12

Family

ID=34280181

Family Applications (3)

Application Number Title Priority Date Filing Date
FR15C0073C Active FR15C0073I2 (fr) 2003-09-03 2015-10-21 Combinaison d'un inhibiteur non-nucleosidique de la transcriptase inverse (nnrti) contenant une pyrimidine avec un inhibiteur nucleosidique de la transcriptase inverse (nrti)
FR15C0072C Active FR15C0072I2 (fr) 2003-09-03 2015-10-21 Combinaison d'un inhibiteur non-nucleosidique de la transcriptase inverse (nnrti) contenant une pyrimidine avec un inhibiteur nucleosidique de la transcriptase inverse (nrti)
FR15C0071C Active FR15C0071I2 (fr) 2003-09-03 2015-10-21 Combinaison d'un inhibiteur non-nucleosidique de la transcriptase inverse (nnrti) contenant une pyrimidine avec un inhibiteur nucleosidique de la transcriptase inverse (nrti)

Family Applications After (2)

Application Number Title Priority Date Filing Date
FR15C0072C Active FR15C0072I2 (fr) 2003-09-03 2015-10-21 Combinaison d'un inhibiteur non-nucleosidique de la transcriptase inverse (nnrti) contenant une pyrimidine avec un inhibiteur nucleosidique de la transcriptase inverse (nrti)
FR15C0071C Active FR15C0071I2 (fr) 2003-09-03 2015-10-21 Combinaison d'un inhibiteur non-nucleosidique de la transcriptase inverse (nnrti) contenant une pyrimidine avec un inhibiteur nucleosidique de la transcriptase inverse (nrti)

Country Status (25)

Country Link
US (9) US20080200435A1 (uk)
EP (1) EP1663240B2 (uk)
JP (3) JP5507791B2 (uk)
KR (1) KR20060090658A (uk)
CN (1) CN101060844B (uk)
AP (1) AP2109A (uk)
AU (5) AU2004268390B2 (uk)
BE (1) BE2015C053I2 (uk)
CA (1) CA2537095C (uk)
CY (5) CY2015040I1 (uk)
FI (1) FI1663240T4 (uk)
FR (3) FR15C0073I2 (uk)
HK (1) HK1092698A1 (uk)
HR (1) HRP20150798T4 (uk)
HU (5) HUS1500053I1 (uk)
IL (2) IL173438A (uk)
LT (2) LTPA2016045I1 (uk)
LU (3) LU92853I2 (uk)
MX (1) MXPA06002437A (uk)
MY (1) MY169670A (uk)
NL (2) NL300781I2 (uk)
NO (6) NO334877B1 (uk)
NZ (1) NZ545306A (uk)
PL (1) PL1663240T5 (uk)
WO (1) WO2005021001A1 (uk)

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Also Published As

Publication number Publication date
US20170100398A1 (en) 2017-04-13
CY2015040I2 (el) 2016-08-31
PL1663240T3 (pl) 2015-10-30
IL173438A0 (en) 2006-06-11
PL1663240T5 (pl) 2024-02-26
US20100029591A1 (en) 2010-02-04
US20220008417A1 (en) 2022-01-13
AU2014203484B2 (en) 2016-09-29
JP2015044839A (ja) 2015-03-12
LU92854I2 (fr) 2015-12-21
IL173438A (en) 2012-03-29
BE2015C053I2 (uk) 2023-12-14
US20140349971A1 (en) 2014-11-27
KR20060090658A (ko) 2006-08-14
HUS1500054I1 (hu) 2016-03-29
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AP2006003551A0 (en) 2006-04-30
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US20200171027A1 (en) 2020-06-04
FR15C0072I1 (uk) 2015-04-12
US8841310B2 (en) 2014-09-23
NL300781I1 (uk) 2016-04-19
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AU2014203484A1 (en) 2014-07-17
FI1663240T4 (fi) 2023-04-25
US20150283135A1 (en) 2015-10-08
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AU2011201123B2 (en) 2013-10-10
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MY169670A (en) 2019-05-08
NO2016025I1 (uk) 2016-12-20
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US20190216807A1 (en) 2019-07-18
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HK1092698A1 (en) 2007-02-16
CY2016048I1 (el) 2017-07-12
LU92855I2 (fr) 2015-12-21
US20180228800A1 (en) 2018-08-16
FR15C0072I2 (fr) 2019-05-17
AP2109A (en) 2010-02-26
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NO2014030I2 (no) 2014-12-18
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AU2011201123A1 (en) 2011-04-07
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US20080200435A1 (en) 2008-08-21
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FR15C0071I1 (uk) 2015-04-12
CY2016048I2 (el) 2017-07-12
JP5507791B2 (ja) 2014-05-28
FR15C0073I2 (fr) 2016-02-12
CY2016049I1 (el) 2017-07-12
AU2016210733B2 (en) 2018-11-08
EP1663240A1 (en) 2006-06-07
CN101060844A (zh) 2007-10-24
HUS1600059I1 (hu) 2017-02-28
NO2014030I1 (no) 2015-01-05
NO2014031I2 (no) 2014-12-18
CY2015038I2 (el) 2016-08-31
NL300768I2 (nl) 2023-08-09
IL213104A (en) 2016-02-29
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JP5820045B2 (ja) 2015-11-24
CY2015039I2 (el) 2016-08-31
CY2015040I1 (el) 2016-08-31
WO2005021001A1 (en) 2005-03-10
HRP20150798T1 (hr) 2015-09-11
NO20061374L (no) 2006-03-27
AU2004268390B2 (en) 2011-03-31
HRP20150798T4 (hr) 2023-06-09
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EP1663240B2 (en) 2023-03-01
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LTPA2016044I1 (lt) 2017-01-10

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