BRPI0814548A2 - Forma cristalina de 4-[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]amino]-2 pirimidinil]amino]benzonitrila - Google Patents
Forma cristalina de 4-[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]amino]-2 pirimidinil]amino]benzonitrilaInfo
- Publication number
- BRPI0814548A2 BRPI0814548A2 BRPI0814548-2A2A BRPI0814548A BRPI0814548A2 BR PI0814548 A2 BRPI0814548 A2 BR PI0814548A2 BR PI0814548 A BRPI0814548 A BR PI0814548A BR PI0814548 A2 BRPI0814548 A2 BR PI0814548A2
- Authority
- BR
- Brazil
- Prior art keywords
- amino
- dimethylphylen
- benzonitril
- cyanoethenyl
- pyrimidinyl
- Prior art date
Links
- -1 2-CYANOETHENYL Chemical class 0.000 title 1
- JFDZBHWFFUWGJE-UHFFFAOYSA-N benzonitrile Chemical compound N#CC1=CC=CC=C1 JFDZBHWFFUWGJE-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Virology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- AIDS & HIV (AREA)
- Tropical Medicine & Parasitology (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP07112392 | 2007-07-12 | ||
PCT/EP2008/059054 WO2009007441A2 (en) | 2007-07-12 | 2008-07-11 | Crystalline form of (e) 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2 pyrimidinyl]amino]benzonitrile |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0814548A2 true BRPI0814548A2 (pt) | 2015-01-06 |
Family
ID=38706528
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0814548-2A2A BRPI0814548A2 (pt) | 2007-07-12 | 2008-07-11 | Forma cristalina de 4-[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]amino]-2 pirimidinil]amino]benzonitrila |
Country Status (15)
Country | Link |
---|---|
US (1) | US8426434B2 (pt) |
EP (1) | EP2175857B1 (pt) |
JP (1) | JP5701057B2 (pt) |
CN (1) | CN101743006B (pt) |
AU (1) | AU2008274185B2 (pt) |
BR (1) | BRPI0814548A2 (pt) |
CA (1) | CA2693044C (pt) |
DK (1) | DK2175857T3 (pt) |
ES (1) | ES2437331T3 (pt) |
HK (1) | HK1144669A1 (pt) |
HR (1) | HRP20131128T1 (pt) |
IL (1) | IL202363A (pt) |
RU (1) | RU2498979C2 (pt) |
SI (1) | SI2175857T1 (pt) |
WO (1) | WO2009007441A2 (pt) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MY169670A (en) | 2003-09-03 | 2019-05-08 | Tibotec Pharm Ltd | Combinations of a pyrimidine containing nnrti with rt inhibitors |
TWI494133B (zh) | 2007-03-14 | 2015-08-01 | Tibotec Pharm Ltd | 重組用粉末 |
ES2530941T3 (es) * | 2009-09-22 | 2015-03-09 | Janssen Sciences Ireland Uc | Tratamiento y prevención de infección por el VIH |
US20120295898A1 (en) * | 2010-01-27 | 2012-11-22 | Mark Richard Underwood | Antiviral Therapy |
TWI577377B (zh) * | 2010-09-16 | 2017-04-11 | Viiv醫療保健公司 | 醫藥組合物 |
WO2012125993A1 (en) | 2011-03-17 | 2012-09-20 | Teva Pharmaceutical Industries Ltd. | Solid state forms of rilpivirine base, and rilipivirine salts |
CN108210469A (zh) | 2011-04-15 | 2018-06-29 | 詹森药业有限公司 | 冻干药物纳米混悬剂 |
EP2604593A1 (en) * | 2011-12-14 | 2013-06-19 | Sandoz AG | Polymorph of Rilpivirine hydrochloride and its use as antiviral |
EP2628732A1 (en) * | 2012-02-20 | 2013-08-21 | Sandoz AG | Novel crystalline form of rilpivirine hydrochloride |
WO2013087794A1 (en) * | 2011-12-14 | 2013-06-20 | Sandoz Ag | Polymorph of rilpivirine hydrochloride and its use as antiviral |
EA201590862A1 (ru) * | 2012-12-14 | 2016-05-31 | ГЛАКСОСМИТКЛАЙН ЭлЭлСи | Фармацевтические композиции |
CZ2015579A3 (cs) | 2015-08-27 | 2017-03-08 | Zentiva, K.S. | Krystalická forma A Rilpivirin Adipátu a způsob její přípravy |
FI3597646T3 (fi) | 2016-08-19 | 2023-09-07 | Gilead Sciences Inc | Hi-virusinfektion profylaktiseen tai terapeuttiseen hoitoon käyttökelpoisia terapeuttisia yhdisteitä |
CN115397422A (zh) | 2019-11-29 | 2022-11-25 | 西皮欧生命科学有限公司 | 包含利匹韦林的组合物和其用于治疗肿瘤或癌症的用途 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5145684A (en) | 1991-01-25 | 1992-09-08 | Sterling Drug Inc. | Surface modified drug nanoparticles |
JO3429B1 (ar) * | 2001-08-13 | 2019-10-20 | Janssen Pharmaceutica Nv | مشتقات برميدينات مثبطة فيروس الايدز |
CA2493794C (en) | 2002-08-09 | 2010-05-25 | Janssen Pharmaceutica N.V. | Processes for the preparation of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl]amino]benzonitrile |
NZ540321A (en) | 2002-11-15 | 2007-09-28 | Tibotec Pharm Ltd | Substituted indolepyridinium as anti-infective compounds |
AU2005279158C1 (en) | 2004-09-02 | 2010-12-16 | Janssen Pharmaceutica N.V. | Hydrochloride of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl] amino]benzonitrile |
BRPI0609299A2 (pt) * | 2005-04-13 | 2010-03-23 | Pfizer Prod Inc | formulaÇÕes de depàsito injetÁveis e mÉtodos para proporcionar liberaÇço sustentada de composiÇÕes de nanopartÍculas |
-
2008
- 2008-07-11 EP EP08786055.7A patent/EP2175857B1/en active Active
- 2008-07-11 WO PCT/EP2008/059054 patent/WO2009007441A2/en active Application Filing
- 2008-07-11 DK DK08786055.7T patent/DK2175857T3/da active
- 2008-07-11 SI SI200831105T patent/SI2175857T1/sl unknown
- 2008-07-11 AU AU2008274185A patent/AU2008274185B2/en active Active
- 2008-07-11 JP JP2010515519A patent/JP5701057B2/ja active Active
- 2008-07-11 ES ES08786055.7T patent/ES2437331T3/es active Active
- 2008-07-11 US US12/668,079 patent/US8426434B2/en active Active
- 2008-07-11 CA CA2693044A patent/CA2693044C/en active Active
- 2008-07-11 RU RU2010104848/04A patent/RU2498979C2/ru active
- 2008-07-11 BR BRPI0814548-2A2A patent/BRPI0814548A2/pt not_active Application Discontinuation
- 2008-07-11 CN CN2008800243222A patent/CN101743006B/zh active Active
-
2009
- 2009-11-26 IL IL202363A patent/IL202363A/en active IP Right Grant
-
2010
- 2010-12-08 HK HK10111404.5A patent/HK1144669A1/xx unknown
-
2013
- 2013-11-26 HR HRP20131128AT patent/HRP20131128T1/hr unknown
Also Published As
Publication number | Publication date |
---|---|
HRP20131128T1 (hr) | 2013-12-20 |
HK1144669A1 (pt) | 2011-03-04 |
IL202363A (en) | 2016-04-21 |
DK2175857T3 (da) | 2013-12-02 |
WO2009007441A3 (en) | 2009-04-30 |
JP2010533148A (ja) | 2010-10-21 |
SI2175857T1 (sl) | 2014-01-31 |
WO2009007441A2 (en) | 2009-01-15 |
CN101743006B (zh) | 2013-09-11 |
CA2693044A1 (en) | 2009-01-15 |
US20100189796A1 (en) | 2010-07-29 |
AU2008274185B2 (en) | 2014-07-03 |
JP5701057B2 (ja) | 2015-04-15 |
IL202363A0 (en) | 2010-06-30 |
CN101743006A (zh) | 2010-06-16 |
AU2008274185A1 (en) | 2009-01-15 |
CA2693044C (en) | 2017-03-14 |
ES2437331T3 (es) | 2014-01-10 |
EP2175857B1 (en) | 2013-09-11 |
RU2498979C2 (ru) | 2013-11-20 |
EP2175857A2 (en) | 2010-04-21 |
US8426434B2 (en) | 2013-04-23 |
RU2010104848A (ru) | 2011-08-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B25D | Requested change of name of applicant approved |
Owner name: JANSSEN R AND D IRELAND (IE) |
|
B25A | Requested transfer of rights approved |
Owner name: JANSSEN SCIENCES IRELAND UC (IE) |
|
B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] |
Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI |
|
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B09B | Patent application refused [chapter 9.2 patent gazette] | ||
B12B | Appeal against refusal [chapter 12.2 patent gazette] |