FI925443A0 - 3-amino-2-arylkinuklidiner, foerfarande foer deras framstaellning och dessa innehaollande farmaceutiska kompositioner - Google Patents

3-amino-2-arylkinuklidiner, foerfarande foer deras framstaellning och dessa innehaollande farmaceutiska kompositioner

Info

Publication number
FI925443A0
FI925443A0 FI925443A FI925443A FI925443A0 FI 925443 A0 FI925443 A0 FI 925443A0 FI 925443 A FI925443 A FI 925443A FI 925443 A FI925443 A FI 925443A FI 925443 A0 FI925443 A0 FI 925443A0
Authority
FI
Finland
Prior art keywords
pct
alkyl
compounds
date dec
furyl
Prior art date
Application number
FI925443A
Other languages
English (en)
Other versions
FI925443A (fi
FI113654B (fi
Inventor
John A Lowe Iii
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI925443A publication Critical patent/FI925443A/fi
Publication of FI925443A0 publication Critical patent/FI925443A0/fi
Application granted granted Critical
Publication of FI113654B publication Critical patent/FI113654B/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI925443A 1990-06-01 1992-11-30 Menetelmä terapeuttisesti käyttökelpoisten atsabisyklo[2.2.2]oktaani-3-amiinien valmistamiseksi FI113654B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US53252590A 1990-06-01 1990-06-01
US53252590 1990-06-01
PCT/US1991/002853 WO1991018899A1 (en) 1990-06-01 1991-04-25 3-amino-2-aryl quinuclidines, process for their preparation and pharmaceutical compositions containing them
US9102853 1991-04-25

Publications (3)

Publication Number Publication Date
FI925443A FI925443A (fi) 1992-11-30
FI925443A0 true FI925443A0 (fi) 1992-11-30
FI113654B FI113654B (fi) 2004-05-31

Family

ID=24122165

Family Applications (1)

Application Number Title Priority Date Filing Date
FI925443A FI113654B (fi) 1990-06-01 1992-11-30 Menetelmä terapeuttisesti käyttökelpoisten atsabisyklo[2.2.2]oktaani-3-amiinien valmistamiseksi

Country Status (18)

Country Link
US (1) US5451586A (fi)
EP (1) EP0532527B1 (fi)
JP (1) JPH072740B2 (fi)
KR (1) KR930700499A (fi)
AT (1) ATE113947T1 (fi)
AU (1) AU648317B2 (fi)
CA (1) CA2084193C (fi)
DE (1) DE69105131T2 (fi)
DK (1) DK0532527T3 (fi)
ES (1) ES2063507T3 (fi)
FI (1) FI113654B (fi)
HU (1) HUT62891A (fi)
IE (1) IE911856A1 (fi)
IL (1) IL98259A0 (fi)
NO (1) NO924612D0 (fi)
PT (1) PT97771A (fi)
WO (1) WO1991018899A1 (fi)
ZA (1) ZA914134B (fi)

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AU2681392A (en) * 1991-11-12 1993-06-15 Pfizer Inc. Acyclic ethylenediamine derivatives as substance p receptor antagonists
FR2688219B1 (fr) 1992-03-03 1994-07-08 Sanofi Elf Sels d'ammonium quaternaires de composes aromatiques amines, leur preparation et compositions pharmaceutiques les contenant.
CA2134964C (en) * 1992-05-18 1997-12-30 Manoj C. Desai Bridged aza-bicyclic derivatives as substance p antagonists
US6048859A (en) 1992-06-29 2000-04-11 Merck & Co., Inc. Morpholine and thiomorpholine tachykinin receptor antagonists
US5637699A (en) * 1992-06-29 1997-06-10 Merck & Co., Inc. Process for preparing morpholine tachykinin receptor antagonists
US5719147A (en) * 1992-06-29 1998-02-17 Merck & Co., Inc. Morpholine and thiomorpholine tachykinin receptor antagonists
GB2268931A (en) * 1992-07-22 1994-01-26 Merck Sharp & Dohme Azabicyclic tachykinin-receptor antagonists
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EP0655996B1 (en) * 1992-08-19 2001-11-07 Pfizer Inc. Substituted benzylamino nitrogen containing non-aromatic heterocycles
US5387595A (en) * 1992-08-26 1995-02-07 Merck & Co., Inc. Alicyclic compounds as tachykinin receptor antagonists
US5837711A (en) * 1992-10-28 1998-11-17 Pfizer Inc. Substituted quinuclidines as substance P antagonists
AU676489B2 (en) * 1992-11-12 1997-03-13 Pfizer Inc. Quinuclidine derivative as substance P antagonist
US5344830A (en) * 1992-12-10 1994-09-06 Merck & Co., Inc. N,N-diacylpiperazine tachykinin antagonists
US5830854A (en) * 1992-12-14 1998-11-03 Merck Sharp & Dohme, Limited Method of treating cystic fibrosis using a tachykinin receptor antagonist
US5340826A (en) * 1993-02-04 1994-08-23 Pfizer Inc. Pharmaceutical agents for treatment of urinary incontinence
US5393762A (en) * 1993-06-04 1995-02-28 Pfizer Inc. Pharmaceutical agents for treatment of emesis
EP0655246A1 (en) * 1993-11-30 1995-05-31 Pfizer Inc. Substance P antagonists for the treatment of disorders caused by helicobacter pylori or other spiral urease-positive gram-negative bacteria
IT1271462B (it) * 1993-12-03 1997-05-28 Menarini Farma Ind Antagonisti delle tachichinine,procedimento per la loro preparazione e loro impiego in formulazioni farmaceutiche.
IL112778A0 (en) * 1994-03-04 1995-05-26 Merck & Co Inc Substituted heterocycles, their preparation and pharmaceutical compositions containing them
FR2719474B1 (fr) * 1994-05-05 1996-05-31 Oreal Utilisation d'un antagoniste de substance P dans une composition cosmétique et composition obtenue.
US6203803B1 (en) 1994-12-14 2001-03-20 Societe L'oreal S.A. Use of a substance P antagonist in a cosmetic composition, and the composition thus obtained
FR2719476B1 (fr) * 1994-05-05 1997-05-23 Oreal Utilisation d'un antagoniste de substance P dans une composition cosmétique et composition obtenue.
TW397825B (en) * 1994-10-14 2000-07-11 Novartis Ag Aroyl-piperidine derivatives
FR2725900B1 (fr) * 1994-10-21 1997-07-18 Sanofi Sa Utilisation d'antagonistes des recepteurs nk1 pour la preparation de medicaments a action cardioregulatrice
IL116249A (en) * 1994-12-12 2003-07-06 Pfizer Nk-1 receptor antagonists for the treatment of neuronal damage and stroke
FR2728165A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
FR2728169A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des prurits et des dysesthesies oculaires ou palpebrales
FR2728166A1 (fr) 1994-12-19 1996-06-21 Oreal Composition topique contenant un antagoniste de substance p
FR2729954B1 (fr) 1995-01-30 1997-08-01 Sanofi Sa Composes heterocycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant
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Also Published As

Publication number Publication date
US5451586A (en) 1995-09-19
DE69105131D1 (de) 1994-12-15
JPH05506243A (ja) 1993-09-16
NO924612L (no) 1992-11-30
FI925443A (fi) 1992-11-30
ATE113947T1 (de) 1994-11-15
HU9203777D0 (en) 1993-03-29
CA2084193A1 (en) 1991-12-02
CA2084193C (en) 1998-04-07
AU648317B2 (en) 1994-04-21
ES2063507T3 (es) 1995-01-01
KR930700499A (ko) 1993-03-15
PT97771A (pt) 1992-03-31
IL98259A0 (en) 1992-06-21
AU7860291A (en) 1991-12-31
HUT62891A (en) 1993-06-28
ZA914134B (en) 1993-01-27
JPH072740B2 (ja) 1995-01-18
FI113654B (fi) 2004-05-31
IE911856A1 (en) 1991-12-04
EP0532527B1 (en) 1994-11-09
DK0532527T3 (da) 1995-01-02
DE69105131T2 (de) 1995-03-23
NO924612D0 (no) 1992-11-30
WO1991018899A1 (en) 1991-12-12
EP0532527A1 (en) 1993-03-24

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