FI892908A0 - Menetelmä uusien terapeuttisesti käyttökelpoisten imidatso/1,5-a/kinoksaliinijohdannaisten valmistamiseksi - Google Patents

Menetelmä uusien terapeuttisesti käyttökelpoisten imidatso/1,5-a/kinoksaliinijohdannaisten valmistamiseksi

Info

Publication number
FI892908A0
FI892908A0 FI892908A FI892908A FI892908A0 FI 892908 A0 FI892908 A0 FI 892908A0 FI 892908 A FI892908 A FI 892908A FI 892908 A FI892908 A FI 892908A FI 892908 A0 FI892908 A0 FI 892908A0
Authority
FI
Finland
Prior art keywords
preparation
therapeutically useful
quinoxaline derivatives
novel therapeutically
imidazo
Prior art date
Application number
FI892908A
Other languages
English (en)
Swedish (sv)
Other versions
FI92204C (fi
FI92204B (fi
FI892908A (fi
Inventor
Holger Claus Hansen
Frank Waetjen
Original Assignee
Ferrosan As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ferrosan As filed Critical Ferrosan As
Publication of FI892908A0 publication Critical patent/FI892908A0/fi
Publication of FI892908A publication Critical patent/FI892908A/fi
Application granted granted Critical
Publication of FI92204B publication Critical patent/FI92204B/fi
Publication of FI92204C publication Critical patent/FI92204C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicinal Preparation (AREA)
FI892908A 1988-06-14 1989-06-14 Menetelmä uusien terapeuttisesti käyttökelpoisten imidatso/1,5-a/kinoksaliinijohdannaisten valmistamiseksi FI92204C (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK322088A DK161148C (da) 1988-06-14 1988-06-14 Imidazoquinoxalinforbindelser, fremgangsmaade til fremstilling deraf samt farmaceutiske praeprater indeholdende forbindelserne

Publications (4)

Publication Number Publication Date
FI892908A0 true FI892908A0 (fi) 1989-06-14
FI892908A FI892908A (fi) 1989-12-15
FI92204B FI92204B (fi) 1994-06-30
FI92204C FI92204C (fi) 1994-10-10

Family

ID=8120424

Family Applications (1)

Application Number Title Priority Date Filing Date
FI892908A FI92204C (fi) 1988-06-14 1989-06-14 Menetelmä uusien terapeuttisesti käyttökelpoisten imidatso/1,5-a/kinoksaliinijohdannaisten valmistamiseksi

Country Status (18)

Country Link
US (1) US5034530A (fi)
EP (1) EP0347094B1 (fi)
JP (1) JPH0236184A (fi)
KR (1) KR910000665A (fi)
AT (1) ATE111100T1 (fi)
AU (1) AU618366B2 (fi)
CA (1) CA1327798C (fi)
DE (1) DE68918003T2 (fi)
DK (1) DK161148C (fi)
ES (1) ES2060769T3 (fi)
FI (1) FI92204C (fi)
IE (1) IE69963B1 (fi)
IL (1) IL90543A0 (fi)
NO (1) NO170806C (fi)
NZ (1) NZ229499A (fi)
PH (1) PH26337A (fi)
PT (1) PT90865B (fi)
ZA (1) ZA894430B (fi)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK160876C (da) * 1987-12-08 1991-10-14 Novo Nordisk As Imidazoquinoxalinforbindelser, fremgangsmaade til deres fremstilling, anvendelse af forbindelserne og farmaceutiske praeparater, hvori forbindelserne indgaar
US5371080A (en) * 1990-06-22 1994-12-06 Novo Nordisk A/S Imidazoquinazoline compounds and their use
US5276028A (en) * 1990-06-22 1994-01-04 Nordisk A/S Imidazoquinoxaline compounds
DK151890D0 (da) * 1990-06-22 1990-06-22 Ferrosan As Heterocykliske forbindelser deres fremstilling og brug
US5153196A (en) * 1991-06-05 1992-10-06 Eli Lilly And Company Excitatory amino acid receptor antagonists and methods for the use thereof
AU657986B2 (en) * 1991-06-14 1995-03-30 Pharmacia & Upjohn Company Imidazo(1,5-a)quinoxalines
US6235740B1 (en) 1997-08-25 2001-05-22 Bristol-Myers Squibb Co. Imidazoquinoxaline protein tyrosine kinase inhibitors
US6635626B1 (en) * 1997-08-25 2003-10-21 Bristol-Myers Squibb Co. Imidazoquinoxaline protein tyrosine kinase inhibitors
CA2322311C (en) * 1998-03-04 2009-10-13 Bristol-Myers Squibb Company Heterocyclo-substituted imidazopyrazine protein tyrosine kinase inhibitors
US20040180898A1 (en) * 2003-03-03 2004-09-16 Bang-Chi Chen Processes for preparing imidazoquinoxalinones, heterocyclic-substituted imidazopyrazinones, imidazoquinoxalines and heterocyclic-substituted imidazopyrazines
JP2011505366A (ja) 2007-11-30 2011-02-24 ワイス・エルエルシー ホスホエステラーゼ10の阻害剤としてのアリールおよびヘテロアリール縮合イミダゾ[1,5−a]ピラジン
AU2008329072A1 (en) * 2007-11-30 2009-06-04 Elbion Gmbh Aryl and heteroaryl fused imidazo (1,5-A) pyrazines as inhibitors of phosphodiesterase 10
TW201111383A (en) * 2009-05-29 2011-04-01 Wyeth Llc Substituted imidazo[1,5-a]quinoxalines as inhibitors of phosphodiesterase 10

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4440929A (en) * 1981-07-16 1984-04-03 Usv Pharmaceutical Corporation Imidazoquinoxaline compounds
DK476885D0 (da) * 1985-10-17 1985-10-17 Ferrosan As Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf
DE3668116D1 (de) * 1985-10-19 1990-02-15 Beecham Group Plc Zusammensetzung zur behandlung von infektionen.
DK155524C (da) * 1987-03-18 1989-09-11 Ferrosan As Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse

Also Published As

Publication number Publication date
JPH0236184A (ja) 1990-02-06
DK161148B (da) 1991-06-03
KR910000665A (ko) 1991-01-30
DE68918003D1 (de) 1994-10-13
NO170806B (no) 1992-08-31
PH26337A (en) 1992-04-29
DE68918003T2 (de) 1995-01-05
FI92204C (fi) 1994-10-10
IL90543A0 (en) 1990-01-18
DK322088A (da) 1990-03-27
IE69963B1 (en) 1996-10-16
AU618366B2 (en) 1991-12-19
FI92204B (fi) 1994-06-30
DK322088D0 (da) 1988-06-14
PT90865B (pt) 1994-11-30
ATE111100T1 (de) 1994-09-15
ES2060769T3 (es) 1994-12-01
DK161148C (da) 1991-11-18
US5034530A (en) 1991-07-23
FI892908A (fi) 1989-12-15
IE891892L (en) 1989-12-14
EP0347094B1 (en) 1994-09-07
NO170806C (no) 1992-12-09
NO892456D0 (no) 1989-06-13
AU3624489A (en) 1989-12-21
EP0347094A1 (en) 1989-12-20
NO892456L (no) 1989-12-15
PT90865A (pt) 1989-12-29
NZ229499A (en) 1991-04-26
CA1327798C (en) 1994-03-15
ZA894430B (en) 1990-02-28

Similar Documents

Publication Publication Date Title
FI92204C (fi) Menetelmä uusien terapeuttisesti käyttökelpoisten imidatso/1,5-a/kinoksaliinijohdannaisten valmistamiseksi
FI925309A0 (fi) Menetelmä uusien terapeuttisesti käyttökelpoisten 4,5-dihydro-4-okso-5-isopropyyli-imidatso/1,5-a/pyrido/2,3-e/pyratsiinijohdannaisten valmistamiseksi
PH25034A (en) Process for the preparation of imidazoquinazoline compounds and intermediate for use in said process
FI922267A0 (fi) Menetelmä uusien terapeuttisesti käyttökelpoisten 3-isoksatsolyyli-4-okso-imidatso/1,5-a/kinoksaliinijohdannaisten valmistamiseksi
NZ226461A (en) S-oxo-imidazo-(1,5-a)-thienopyrimidine derivatives; pharmaceutical compositions and processes for preparation
FI922269A (fi) Menetelmä uusien terapeuttisesti käyttökelpoisten 4-okso-imidatso/1,5-a/kinoksaliinijohdannaisten valmistamiseksi

Legal Events

Date Code Title Description
BB Publication of examined application
MM Patent lapsed
MM Patent lapsed

Owner name: NOVO NORDISK A/S