FI882360A0 - Menetelmä terapeuttisesti käyttökelpoisten -(fluorimetyleeni)-5-hydroksitryptofaanijohdannaisten valmistamiseksi - Google Patents
Menetelmä terapeuttisesti käyttökelpoisten -(fluorimetyleeni)-5-hydroksitryptofaanijohdannaisten valmistamiseksiInfo
- Publication number
- FI882360A0 FI882360A0 FI882360A FI882360A FI882360A0 FI 882360 A0 FI882360 A0 FI 882360A0 FI 882360 A FI882360 A FI 882360A FI 882360 A FI882360 A FI 882360A FI 882360 A0 FI882360 A0 FI 882360A0
- Authority
- FI
- Finland
- Prior art keywords
- fluoromethylene
- hydroxytryptophan
- derivatives
- preparation
- therapeutically useful
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D209/20—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals substituted additionally by nitrogen atoms, e.g. tryptophane
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Indole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US5321287 | 1987-05-21 | ||
| US07/053,212 US4822812A (en) | 1987-05-21 | 1987-05-21 | β-(Fluoromethylene)-5-hydroxytryptophan and derivatives and their use as prodrugs for MAO inhibition |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| FI882360A0 true FI882360A0 (fi) | 1988-05-19 |
| FI882360A FI882360A (fi) | 1988-11-22 |
| FI90531B FI90531B (fi) | 1993-11-15 |
| FI90531C FI90531C (fi) | 1994-02-25 |
Family
ID=21982670
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI882360A FI90531C (fi) | 1987-05-21 | 1988-05-19 | Menetelmä terapeuttisesti käyttökelpoisten -(fluorimetyleeni)-5-hydroksitryptofaanijohdannaisten valmistamiseksi |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US4822812A (fi) |
| EP (1) | EP0291998A3 (fi) |
| JP (1) | JP2520285B2 (fi) |
| KR (1) | KR960016521B1 (fi) |
| CN (1) | CN1031222A (fi) |
| AR (1) | AR246952A1 (fi) |
| AU (1) | AU605865B2 (fi) |
| CA (1) | CA1310973C (fi) |
| DK (1) | DK169330B1 (fi) |
| FI (1) | FI90531C (fi) |
| HU (2) | HU199790B (fi) |
| IL (1) | IL86387A0 (fi) |
| NO (1) | NO172576C (fi) |
| NZ (1) | NZ224661A (fi) |
| PH (1) | PH25384A (fi) |
| PT (1) | PT87538B (fi) |
| ZA (1) | ZA883442B (fi) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5488188A (en) * | 1994-09-29 | 1996-01-30 | Merrell Dow Pharmaceuticals Inc. | Process for the preparation of (E)-1-amino-2-(fluoromethylene)-4-(p-fluorophenyl)butane, novel processes for preparing an intermediate thereof, and novel intermediates thereof |
| ITRM20020255A1 (it) * | 2002-05-09 | 2003-11-10 | Polifarma Spa | Tautomero enolico dell'acido 3-indolilpiruvico, suoi sali e usi terapeutici. |
| US6972014B2 (en) * | 2003-01-04 | 2005-12-06 | Endocare, Inc. | Open system heat exchange catheters and methods of use |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2513597B2 (de) * | 1975-03-27 | 1977-06-02 | L-5-hydroxytryptophan-l-glutamatmonohydrat, verfahren zu seiner herstellung und arzneimittel | |
| US4183858A (en) * | 1977-07-01 | 1980-01-15 | Merrell Toraude Et Compagnie | α-Vinyl tryptophanes |
| FR2499076A1 (fr) * | 1981-02-02 | 1982-08-06 | Panmedica Laboratoires | Nouveaux derives de l'acide ((indol-3 yl)-3 amino-2 propionyloxy)-2 acetique, procedes pour leur preparation et medicaments les contenant |
| US4421767A (en) * | 1981-06-01 | 1983-12-20 | Merrell Toraude Et Compagnie | Compounds and methods for treating depression |
| US4454158A (en) * | 1981-06-01 | 1984-06-12 | Merrell Toraude Et Compagnie | Allyl amine MAO inhibitors |
| ZA855101B (en) * | 1984-07-13 | 1986-05-28 | Merrell Dow Pharma | Fluoroallylaine derivatives |
-
1987
- 1987-05-21 US US07/053,212 patent/US4822812A/en not_active Expired - Lifetime
-
1988
- 1988-05-15 IL IL86387A patent/IL86387A0/xx not_active IP Right Cessation
- 1988-05-16 CA CA000566913A patent/CA1310973C/en not_active Expired - Lifetime
- 1988-05-16 AR AR88310862A patent/AR246952A1/es active
- 1988-05-16 ZA ZA883442A patent/ZA883442B/xx unknown
- 1988-05-17 AU AU16347/88A patent/AU605865B2/en not_active Ceased
- 1988-05-17 NZ NZ224661A patent/NZ224661A/xx unknown
- 1988-05-18 PH PH36944A patent/PH25384A/en unknown
- 1988-05-19 PT PT87538A patent/PT87538B/pt not_active IP Right Cessation
- 1988-05-19 FI FI882360A patent/FI90531C/fi not_active IP Right Cessation
- 1988-05-19 KR KR1019880005872A patent/KR960016521B1/ko not_active IP Right Cessation
- 1988-05-20 HU HU882617A patent/HU199790B/hu not_active IP Right Cessation
- 1988-05-20 JP JP63122187A patent/JP2520285B2/ja not_active Expired - Lifetime
- 1988-05-20 CN CN88103199A patent/CN1031222A/zh active Pending
- 1988-05-20 EP EP88108125A patent/EP0291998A3/en not_active Withdrawn
- 1988-05-20 DK DK278388A patent/DK169330B1/da not_active IP Right Cessation
- 1988-05-20 NO NO882240A patent/NO172576C/no not_active IP Right Cessation
- 1988-05-20 HU HU89172A patent/HUT50117A/hu unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR880013891A (ko) | 1988-12-22 |
| AU605865B2 (en) | 1991-01-24 |
| IL86387A0 (en) | 1988-11-15 |
| EP0291998A2 (en) | 1988-11-23 |
| AU1634788A (en) | 1988-11-24 |
| NZ224661A (en) | 1990-08-28 |
| NO882240L (no) | 1988-11-22 |
| HUT50117A (en) | 1989-12-28 |
| FI90531C (fi) | 1994-02-25 |
| JP2520285B2 (ja) | 1996-07-31 |
| AR246952A1 (es) | 1994-10-31 |
| NO882240D0 (no) | 1988-05-20 |
| NO172576B (no) | 1993-05-03 |
| PH25384A (en) | 1991-06-03 |
| US4822812A (en) | 1989-04-18 |
| EP0291998A3 (en) | 1989-01-25 |
| FI882360A (fi) | 1988-11-22 |
| DK278388D0 (da) | 1988-05-20 |
| IL86387A (fi) | 1992-12-01 |
| KR960016521B1 (ko) | 1996-12-14 |
| PT87538B (pt) | 1992-09-30 |
| NO172576C (no) | 1993-08-11 |
| JPS63303965A (ja) | 1988-12-12 |
| HUT47905A (en) | 1989-04-28 |
| CA1310973C (en) | 1992-12-01 |
| DK169330B1 (da) | 1994-10-10 |
| FI90531B (fi) | 1993-11-15 |
| HU199790B (en) | 1990-03-28 |
| ZA883442B (en) | 1988-11-16 |
| PT87538A (pt) | 1989-05-31 |
| CN1031222A (zh) | 1989-02-22 |
| DK278388A (da) | 1988-11-22 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| FI883064A (fi) | Menetelmä terapeuttisesti käyttökelpoisten heterosyklisten yhdisteiden valmistamiseksi | |
| FI92934B (fi) | Analogiamenetelmä terapeuttisesti käyttökelpoisten 1-deoksinojirimysiinijohdannaisten valmistamiseksi | |
| FI880941A0 (fi) | Menetelmä terapeuttisesti käyttökelpoisten piperatsinyyli-heterosyklisten yhdisteiden valmistamiseksi | |
| FI90346C (fi) | Menetelmä terapeuttisesti käyttökelpoisten nor-statiini- ja nor-syklostatiinipolypeptidien valmistamiseksi | |
| FI890282A (fi) | Menetelmä terapeuttisesti käyttökelpoisten 23,24-didehydro-25-hydroksikalsiferolijohdannaisten valmistamiseksi | |
| FI882638A0 (fi) | Menetelmä terapeuttisesti käyttökelpoisten booriaminohappojohdannaisten valmistamiseksi | |
| FI880757A0 (fi) | Menetelmä valmistaa terapeuttisesti vaikuttavia tyydytettyjä heterosyklisiä karboksamidijohdoksia | |
| FI95704B (fi) | Menetelmä uusien terapeuttisesti käyttökelpoisten pyridiinijohdannaisten valmistamiseksi | |
| FI90769C (fi) | Menetelmä terapeuttisesti käyttökelpoisten triatsoliyhdisteiden valmistamiseksi | |
| FI892881A0 (fi) | Menetelmä terapeuttisesti käyttökelpoisten aminohappojohdannaisten va lmistamiseksi | |
| FI882007A (fi) | Menetelmä steroidi-5- -reduktaasin inhibiittorien valmistamiseksi | |
| FI874459A0 (fi) | Menetelmä uusien terapeuttisesti käyttökelpoisten piperidiinijohdannaisten valmistamiseksi | |
| FI850654A0 (fi) | Menetelmä terapeuttisesti käyttökelpoisten pleuromutilinijohdannaisten valmistamiseksi | |
| FI892182A (fi) | Menetelmä terapeuttisesti käyttökelpoisten kromaanijohdannaisten valmistamiseksi | |
| FI94752C (fi) | Menetelmä terapeuttisesti käyttökelpoisten propenonioksiimieettereiden valmistamiseksi | |
| FI880869A (fi) | Menetelmä terapeuttisesti aktiivisten tetratsolijohdannaisten valmistamiseksi | |
| FI93215C (fi) | Menetelmä terapeuttisesti käyttökelpoisten aminoalkoksifenyylijohdannaisten valmistamiseksi | |
| FI880467A (fi) | Menetelmä terapeuttisesti käyttökelpoisten substituoitujen 3,4-dihydro-2H-bentsopyraanien valmistamiseksi | |
| FI884910A (fi) | Menetelmä terapeuttisesti käyttökelpoisten bentsopyraanijohdannaisten valmistamiseksi | |
| FI873350A (fi) | Menetelmä terapeuttisesti käyttökelpoisten 1,4-dihydropyridiinijohdannaisten valmistamiseksi | |
| FI872769A (fi) | Menetelmä alfa-mono-olefiinien polymeroimiseksi | |
| FI893003A0 (fi) | Menetelmä uusien terapeuttisesti käyttökelpoisten neplanosiinijohdannaisten valmistamiseksi | |
| FI892948A (fi) | Menetelmä terapeuttisesti käyttökelpoisten kromaanijohdannaisten valmistamiseksi | |
| FI891144A0 (fi) | Menetelmä uusien terapeuttisesti käyttökelpoisten suolayhdisteiden valmistamiseksi | |
| FI92188C (fi) | Menetelmä terapeuttisesti käyttökelpoisten fenoksialkyylipyrokatekolijohdannaisten valmistamiseksi |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| BB | Publication of examined application | ||
| MM | Patent lapsed |
Owner name: MERRELL DOW PHARMACEUTICALS INC. |