FI833931A - Foerbaettringar vid foerfaranden foer framstaellning av 3-aryl-5-pyrazol-derivat - Google Patents
Foerbaettringar vid foerfaranden foer framstaellning av 3-aryl-5-pyrazol-derivat Download PDFInfo
- Publication number
- FI833931A FI833931A FI833931A FI833931A FI833931A FI 833931 A FI833931 A FI 833931A FI 833931 A FI833931 A FI 833931A FI 833931 A FI833931 A FI 833931A FI 833931 A FI833931 A FI 833931A
- Authority
- FI
- Finland
- Prior art keywords
- derivat
- pyrazol
- aryl
- foer framstaellning
- foerfaranden foer
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/437,994 US4495195A (en) | 1982-11-01 | 1982-11-01 | Xanthine oxidase inhibiting 3(5)-phenyl-substituted-5(3)-pyrazole-carboxylic acid derivatives, compositions, and methods of use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FI833931A0 FI833931A0 (fi) | 1983-10-27 |
| FI833931A true FI833931A (fi) | 1984-05-02 |
Family
ID=23738785
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI833931A FI833931A (fi) | 1982-11-01 | 1983-10-27 | Foerbaettringar vid foerfaranden foer framstaellning av 3-aryl-5-pyrazol-derivat |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US4495195A (fi) |
| EP (1) | EP0112623A2 (fi) |
| JP (1) | JPS5995272A (fi) |
| KR (1) | KR840006629A (fi) |
| AU (1) | AU2068583A (fi) |
| DD (1) | DD210265A5 (fi) |
| DK (1) | DK492783D0 (fi) |
| ES (1) | ES8601900A1 (fi) |
| FI (1) | FI833931A (fi) |
| GB (1) | GB2130205A (fi) |
| GR (1) | GR79640B (fi) |
| IL (1) | IL70075A0 (fi) |
| PT (1) | PT77583B (fi) |
Families Citing this family (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ208555A (en) * | 1983-06-23 | 1987-06-30 | American Cyanamid Co | (3-amino-1h-pyrazol-4-yl)-arylmethanone derivatives |
| IE59813B1 (en) * | 1986-05-09 | 1994-04-06 | Warner Lambert Co | Styryl pyrazoles, isoxazoles and analogs thereof having activity as 5-lipoxy-genase inhibitors and pharmaceutical compositions containing them |
| JPS6425763A (en) | 1987-04-24 | 1989-01-27 | Mitsubishi Chem Ind | Pyrazoles and insecticide and acaricide containing said pyrazoles as active ingredient |
| US4861777A (en) * | 1987-09-11 | 1989-08-29 | Mitsubishi Kasei Corporation | Pyrazole derivative and insecticidal and miticidal composition containing the derivative as active ingredient |
| JP2751309B2 (ja) * | 1988-02-16 | 1998-05-18 | 三菱化学株式会社 | ピラゾール類およびこれを有効成分とする殺虫、殺ダニ、殺菌剤 |
| JP2784925B2 (ja) * | 1988-09-07 | 1998-08-13 | 日本農薬株式会社 | ３又は５−フェニルピラゾール類又はその塩及び除草剤 |
| CA2036192A1 (en) | 1990-02-13 | 1991-08-14 | Nicholas Meanwell | Heterocyclic carboxylic acids and esters |
| US4956379A (en) * | 1990-02-13 | 1990-09-11 | Bristol-Myers Squibb Company | Pyrazole carboxylic acids and esters and inhibition of blood platelet aggregation therewith |
| FR2665898B1 (fr) * | 1990-08-20 | 1994-03-11 | Sanofi | Derives d'amido-3 pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant. |
| US5294630A (en) * | 1992-07-07 | 1994-03-15 | Eli Lilly And Company | Treatment of inflammatory bowel disease |
| US5436258A (en) * | 1992-09-09 | 1995-07-25 | Eli Lilly And Company | Prevention of bone resorption |
| GB9312853D0 (en) * | 1993-06-22 | 1993-08-04 | Euro Celtique Sa | Chemical compounds |
| US5591776A (en) * | 1994-06-24 | 1997-01-07 | Euro-Celtique, S.A. | Pheynl or benzyl-substituted rolipram-based compounds for and method of inhibiting phosphodiesterase IV |
| HRP950330A2 (en) * | 1994-07-05 | 1997-10-31 | Ciba Geigy Ag | New herbicides |
| EP0814809B1 (en) * | 1994-12-13 | 2003-08-13 | Euroceltique S.A. | Aryl thioxanthines |
| DE69531555T2 (de) * | 1994-12-13 | 2004-06-17 | Euroceltique S.A. | Dreifachsubstituierte thioxanthine |
| US6025361A (en) * | 1994-12-13 | 2000-02-15 | Euro-Celtique, S.A. | Trisubstituted thioxanthines |
| US6166041A (en) * | 1995-10-11 | 2000-12-26 | Euro-Celtique, S.A. | 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma |
| US6075016A (en) * | 1996-04-10 | 2000-06-13 | Euro-Celtique S.A. | 6,5-fused aromatic ring systems having enhanced phosphodiesterase IV inhibitory activity |
| ID21775A (id) * | 1996-10-25 | 1999-07-22 | Yoshitomi Pharmaceutical | Senyawa-senyawa 1-fenilpirazol dan penggunaan farmasinya |
| US5723608A (en) * | 1996-12-31 | 1998-03-03 | Neurogen Corporation | 3-aryl substituted pyrazolo 4,3-d!pyrimidine derivatives; corticotropin-releasing factor receptor (CRF1) specific ligands |
| AU1520699A (en) | 1997-11-07 | 1999-05-31 | Johns Hopkins University, The | Methods for treatment of disorders of cardiac contractility |
| EP1783124A4 (en) * | 2004-08-27 | 2009-07-08 | Astellas Pharma Inc | 2-PHENYLTHIOPHENDERIVAT |
| CA2578168A1 (en) * | 2004-08-27 | 2006-03-02 | Astellas Pharma Inc. | 2-phenylpyridine derivative |
| AU2006300422A1 (en) | 2005-10-07 | 2007-04-19 | Astellas Pharma Inc. | Triarylcarboxylic acid derivative |
| WO2007097403A1 (ja) | 2006-02-24 | 2007-08-30 | Astellas Pharma Inc. | 消化管潰瘍治療又は予防薬 |
| CN102333765B (zh) | 2009-02-27 | 2015-01-14 | 帝人制药株式会社 | 基于使用过渡金属催化剂的偶联法的苯基取代杂环衍生物的制造方法 |
| PL2610248T3 (pl) | 2010-08-27 | 2016-12-30 | Sposób wytwarzania podstawionych fenylem pochodnych heterocyklicznych metodą sprzęgania z użyciem związku palladu | |
| ES2666918T3 (es) | 2013-03-29 | 2018-05-08 | Teijin Pharma Limited | Derivado de pirazol |
| EP2944635B1 (en) * | 2014-05-15 | 2018-11-28 | Council of Scientific & Industrial Research | Pyrazole linked benzimidazole conjugates and a process for preparation thereof |
| CN106632245B (zh) * | 2016-09-30 | 2019-11-15 | 华南理工大学 | 氮取代基苯基吡唑类黄嘌呤氧化还原酶抑制剂及制备与应用 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1261124B (de) * | 1961-09-22 | 1968-02-15 | Hoechst Ag | Verfahren zur Herstellung von Pyrazolen |
| IT1053661B (it) * | 1966-09-27 | 1981-10-10 | Farmacosmici S P A | Ammidi dell acido 3 5 metil 5 3 pirazol carbossilico |
| FR2104931B1 (fi) * | 1970-09-08 | 1975-01-10 | Ferlux | |
| DE2508934A1 (de) * | 1974-03-04 | 1975-09-11 | Byk Gulden Lomberg Chem Fab | Neue substituierte 5-amino-4- formyl-carbamoyl-pyrazole, verfahren zu ihrer herstellung und sie enthaltende arzneimittel |
| DE2410653A1 (de) * | 1974-03-06 | 1975-10-30 | Byk Gulden Lomberg Chem Fab | Neue heterocyclisch substituierte 5amino-4-formylcarbamoyl-pyrazole, verfahren zu ihrer herstellung und sie enthaltende arzneimittel |
| US3903106A (en) * | 1974-04-12 | 1975-09-02 | Lilly Co Eli | Pyrazole-3-carboxylic acids |
| US3895027A (en) * | 1974-04-12 | 1975-07-15 | Lilly Co Eli | Process for preparing pyrazole-3-carboxylic acids |
| US3899508A (en) * | 1974-04-12 | 1975-08-12 | Lilly Co Eli | 5-(2-Aminophenyl)pyrazole-3-carboxylic acids and esters thereof |
| FR2353292A1 (fr) * | 1975-08-05 | 1977-12-30 | Sogeras | Nouveaux derives du benzoyl-3 pyrazole |
| FR2320093A1 (fr) * | 1975-08-05 | 1977-03-04 | Sogeras | Nouveaux acides diphenyl-pyrazole-5-acetiques |
| US4214090A (en) * | 1976-01-14 | 1980-07-22 | Commonwealth Scientific And Industrial Research Organization | Fungicidal carboxamidopyrazoles |
| US4134987A (en) * | 1976-01-14 | 1979-01-16 | Huppatz John L | Compounds and compositions |
| US4245106A (en) * | 1979-07-05 | 1981-01-13 | Monsanto Company | Process for the preparation of 1-alkyl-3-aryl-4-pyrazolecarboxylates |
| US4346097A (en) * | 1980-09-30 | 1982-08-24 | Warner-Lambert Company | Method for treating convulsions with pyrazole-4-carboxamide derivatives |
-
1982
- 1982-11-01 US US06/437,994 patent/US4495195A/en not_active Expired - Fee Related
-
1983
- 1983-10-26 GR GR72796A patent/GR79640B/el unknown
- 1983-10-27 EP EP83306530A patent/EP0112623A2/en not_active Withdrawn
- 1983-10-27 DK DK4927/83A patent/DK492783D0/da not_active Application Discontinuation
- 1983-10-27 IL IL70075A patent/IL70075A0/xx unknown
- 1983-10-27 GB GB08328755A patent/GB2130205A/en not_active Withdrawn
- 1983-10-27 FI FI833931A patent/FI833931A/fi not_active Application Discontinuation
- 1983-10-28 KR KR1019830005109A patent/KR840006629A/ko not_active IP Right Cessation
- 1983-10-28 PT PT77583A patent/PT77583B/pt unknown
- 1983-10-28 ES ES526869A patent/ES8601900A1/es not_active Expired
- 1983-10-28 AU AU20685/83A patent/AU2068583A/en not_active Abandoned
- 1983-10-28 JP JP58203575A patent/JPS5995272A/ja active Pending
- 1983-10-28 DD DD83256094A patent/DD210265A5/de unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DD210265A5 (de) | 1984-06-06 |
| ES526869A0 (es) | 1985-05-01 |
| US4495195A (en) | 1985-01-22 |
| ES8601900A1 (es) | 1985-05-01 |
| GR79640B (fi) | 1984-10-31 |
| KR840006629A (ko) | 1984-12-01 |
| PT77583B (en) | 1986-05-27 |
| GB2130205A (en) | 1984-05-31 |
| DK492783D0 (da) | 1983-10-27 |
| PT77583A (en) | 1983-11-01 |
| EP0112623A2 (en) | 1984-07-04 |
| GB8328755D0 (en) | 1983-11-30 |
| AU2068583A (en) | 1984-05-10 |
| IL70075A0 (en) | 1984-01-31 |
| FI833931A0 (fi) | 1983-10-27 |
| JPS5995272A (ja) | 1984-06-01 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| FI833855A (fi) | Anordning vid engaongsbloeja | |
| FI833931A (fi) | Foerbaettringar vid foerfaranden foer framstaellning av 3-aryl-5-pyrazol-derivat | |
| FI830964A0 (fi) | Slityta foer ytterdaeck anvaendbara vid terraengkoerning | |
| FI831449A0 (fi) | Saett vid framstaellning av sulfatmassa | |
| FI65375B (fi) | Saett vid aoterkompressionsindustning av en loesning | |
| FI821186L (fi) | Sugskaop vid en flaekt | |
| FI830460A0 (fi) | Anordning vid elektrod | |
| FI831004A0 (fi) | Drivanordning foer tvinnhuvudena vid en sz-tvinnmaskin | |
| FI824534A0 (fi) | Anordning vid en absorptionskylapparat | |
| FI831348L (fi) | Anordning vid sjoefoerlagda roervaermevaexlare | |
| FI831351A0 (fi) | Anordning vid flishuggmaskiner | |
| FI833812A0 (fi) | Anordning vid innerpanel foer eliminering av en kallstraolande vaegg-, tak- eller golvyta | |
| FI830209A0 (fi) | Foerbaettringar vid cigarettfilter | |
| FI822958A0 (fi) | Anordning vid luftkuddefarkoster | |
| FI824342A0 (fi) | Filmbehandlingssystem vid tomografiavbildningsapparat | |
| FI822570A0 (fi) | Anvaendning av pneumatik vid kuvertmaskin | |
| FI820186L (fi) | Anordning foer koppling av en arbetsmaskin vid en dragmaskins lyft- eller dragarm | |
| FI824484A0 (fi) | Foerfarande foer laddning av laosanordning vid vapen | |
| FI822193L (fi) | Foerfarande vid delignifiering av cellulosamassa | |
| FI821532A0 (fi) | Anslutningsanordning foer anvaendning vid hantering av saogat virke | |
| FI821251L (fi) | Foerfarande vid delignifiering av cellulosamassa | |
| FI820036L (fi) | Optimering av befuktningen vid plantrycksfoerfaranden | |
| FI820213L (fi) | Arbetsredskap foer anvaendning vid fastspikning av spontgolv | |
| FI65670B (fi) | Faeststativ foer kikare vid hagelstudsare | |
| FI822904A0 (fi) | Anordning vid en kopplingsarmatur foer belysningsstolpar |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Application withdrawn |
Owner name: ELI LILLY AND COMPANY |