FI821160A7 - Menetelmä 3-(4- aminoetoksibentsoyyli)bentso/b/tiofeenien valmistamiseksi. - Google Patents

Menetelmä 3-(4- aminoetoksibentsoyyli)bentso/b/tiofeenien valmistamiseksi. Download PDF

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Publication number
FI821160A7
FI821160A7 FI821160A FI821160A FI821160A7 FI 821160 A7 FI821160 A7 FI 821160A7 FI 821160 A FI821160 A FI 821160A FI 821160 A FI821160 A FI 821160A FI 821160 A7 FI821160 A7 FI 821160A7
Authority
FI
Finland
Prior art keywords
aminoethoxybenzoyl
thiophenes
benzo
preparation
Prior art date
Application number
FI821160A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI821160L (fi
FI821160A0 (fi
Inventor
Mary Elizabeth Goettel
Charles David Jones
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/246,334 external-priority patent/US4358593A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of FI821160A0 publication Critical patent/FI821160A0/fi
Publication of FI821160L publication Critical patent/FI821160L/fi
Publication of FI821160A7 publication Critical patent/FI821160A7/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Extrusion Moulding Of Plastics Or The Like (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI821160A 1981-04-03 1982-04-02 Menetelmä 3-(4- aminoetoksibentsoyyli)bentso/b/tiofeenien valmistamiseksi. FI821160A7 (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24633581A 1981-04-03 1981-04-03
US06/246,334 US4358593A (en) 1981-04-03 1981-04-03 Process for preparing 3-(4-aminoethoxybenzoyl)benzo[b]thiophenes
US33104581A 1981-12-16 1981-12-16

Publications (3)

Publication Number Publication Date
FI821160A0 FI821160A0 (fi) 1982-04-02
FI821160L FI821160L (fi) 1982-10-04
FI821160A7 true FI821160A7 (fi) 1982-10-04

Family

ID=27399920

Family Applications (1)

Application Number Title Priority Date Filing Date
FI821160A FI821160A7 (fi) 1981-04-03 1982-04-02 Menetelmä 3-(4- aminoetoksibentsoyyli)bentso/b/tiofeenien valmistamiseksi.

Country Status (17)

Country Link
EP (1) EP0062504B1 (enExample)
KR (1) KR850001882B1 (enExample)
CS (1) CS227348B2 (enExample)
DD (1) DD201793A5 (enExample)
DE (1) DE3268227D1 (enExample)
DK (1) DK151282A (enExample)
EG (1) EG15610A (enExample)
ES (1) ES511124A0 (enExample)
FI (1) FI821160A7 (enExample)
GB (1) GB2097392B (enExample)
GR (1) GR76468B (enExample)
HU (1) HU191353B (enExample)
IE (1) IE53187B1 (enExample)
IL (1) IL65378A (enExample)
PL (1) PL130867B1 (enExample)
PT (1) PT74692B (enExample)
SU (1) SU1155157A3 (enExample)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4117512A1 (de) * 1991-05-25 1992-11-26 Schering Ag 2-phenylbenzo(b)furane und -thiophene, verfahren zu deren herstellung und diese enthaltende pharmazeutische praeparate
CA2145614A1 (en) * 1994-03-31 1995-10-01 Jeffrey A. Dodge Intermediates and processes for preparing benzothiophene compounds
US5523416A (en) * 1994-07-22 1996-06-04 Eli Lilly And Company Process for preparing 3-(4-aminoethoxy-benzoyl) benzo (B)-thiophenes
US5629425A (en) * 1994-09-19 1997-05-13 Eli Lilly And Company Haloalkyl hemisolvates of 6-hydroxy-2-(4-hydroxyphenyl)-3-[4-piperidinoethoxy)-benzoyl]benzo[b]thiophene
CO4410190A1 (es) 1994-09-19 1997-01-09 Lilly Co Eli 3-[4-(2-AMINOETOXI)-BENZOIL]-2-ARIL-6-HIDROXIBENZO [b] TIOFENO CRISTALINO
US5589482A (en) * 1994-12-14 1996-12-31 Pfizer Inc. Benzo-thiophene estrogen agonists to treat prostatic hyperplasia
US6391892B1 (en) * 1995-03-10 2002-05-21 Eli Lilly And Company Naphthyl pharmaceutical compounds
US5728724A (en) * 1995-08-17 1998-03-17 Eli Lilly And Company Benzothiophene compounds
AU5258696A (en) * 1996-03-19 1997-10-10 Eli Lilly And Company Synthesis of 3-{4-(2-aminoethoxy)-benzoyl}-2-aryl-6-hydroxy-benzo{b}thiop henes
IN183239B (enExample) * 1996-09-25 1999-10-09 Lilly Co Eli
US5916916A (en) * 1996-10-10 1999-06-29 Eli Lilly And Company 1-aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods
ZA9710262B (en) * 1996-11-19 1999-05-13 Lilly Co Eli Process for the synthesis of benzothiophenes
CN1254280A (zh) * 1997-04-30 2000-05-24 伊莱利利公司 用于制备取代的苯并[b]噻吩的区域选择性烷基化方法
HUP0003187A3 (en) * 1997-04-30 2002-04-29 Lilly Co Eli Substituted benzothiophenes and process for preparing them
CA2236254A1 (en) * 1997-04-30 1998-10-30 David Warren Hoard Process for preparing benzo¬b|thiophenes
CN1252717A (zh) * 1997-04-30 2000-05-10 伊莱利利公司 制备苯并[b]噻吩的中间体和方法
CA2231013A1 (en) * 1997-04-30 1998-10-30 Eli Lilly And Company Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceuticals
AU7261498A (en) * 1997-04-30 1998-11-24 Eli Lilly And Company Intermediates and processes for preparing benzo{b}thiophenes
EP1832582A1 (en) 2002-09-30 2007-09-12 A/S GEA Farmaceutisk Fabrik Novel raloxifene malonic acid addition salts and/or solvates thereof, and pharmaceutical compositions comprising these
EP2322519A1 (en) * 2009-10-23 2011-05-18 Hexal AG A process for preparing benzo[b]thiophene derivatives
WO2011099942A1 (en) 2010-02-09 2011-08-18 Silverstone Pharma New addition salts of raloxifene, process for the preparation thereof and use thereof in therapy

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3947470A (en) * 1974-06-20 1976-03-30 Smithkline Corporation Substituted benzofurans and benzothiophenes
US4001426A (en) * 1974-10-17 1977-01-04 Smithkline Corporation Substituted benzofurans and benzothiophenes
FR2279395A1 (fr) * 1975-06-02 1976-02-20 Labaz Nouveaux derives de benzthiophene, leurs precedes de preparation ainsi que les compositions pharmaceutiques les contenant
US4133814A (en) 1975-10-28 1979-01-09 Eli Lilly And Company 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents

Also Published As

Publication number Publication date
FI821160L (fi) 1982-10-04
GR76468B (enExample) 1984-08-10
EP0062504B1 (en) 1986-01-02
ES8307240A1 (es) 1983-06-16
KR850001882B1 (ko) 1985-12-28
FI821160A0 (fi) 1982-04-02
EP0062504A1 (en) 1982-10-13
KR830010100A (ko) 1983-12-26
IL65378A0 (en) 1982-05-31
IE820786L (en) 1982-10-03
IE53187B1 (en) 1988-08-17
HU191353B (en) 1987-02-27
SU1155157A3 (ru) 1985-05-07
PT74692B (en) 1985-01-08
DD201793A5 (de) 1983-08-10
DE3268227D1 (en) 1986-02-13
IL65378A (en) 1986-02-28
PL235752A1 (enExample) 1982-11-22
DK151282A (da) 1982-10-04
GB2097392B (en) 1985-04-24
PL130867B1 (en) 1984-09-29
PT74692A (en) 1982-05-01
EG15610A (en) 1986-06-30
GB2097392A (en) 1982-11-03
CS227348B2 (en) 1984-04-16
ES511124A0 (es) 1983-06-16

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Date Code Title Description
FD Application lapsed

Owner name: ELI LILLY AND COMPANY