FI69082C - Foerfarande foer framstaellning av paromomycinderivat - Google Patents

Foerfarande foer framstaellning av paromomycinderivat Download PDF

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Publication number
FI69082C
FI69082C FI801769A FI801769A FI69082C FI 69082 C FI69082 C FI 69082C FI 801769 A FI801769 A FI 801769A FI 801769 A FI801769 A FI 801769A FI 69082 C FI69082 C FI 69082C
Authority
FI
Finland
Prior art keywords
benzoyl
deoxy
penta
paromomycin
acyl
Prior art date
Application number
FI801769A
Other languages
English (en)
Finnish (fi)
Other versions
FI801769A (fi
FI69082B (fi
Inventor
Carlo Battistini
Giuseppe Cassinelli
Giovanni Franceschi
Rosanna Mazzoleni
Federico Arcamone
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of FI801769A publication Critical patent/FI801769A/fi
Publication of FI69082B publication Critical patent/FI69082B/fi
Application granted granted Critical
Publication of FI69082C publication Critical patent/FI69082C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/228—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to adjacent ring-carbon atoms of the cyclohexane rings
    • C07H15/232—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to adjacent ring-carbon atoms of the cyclohexane rings with at least three saccharide radicals in the molecule, e.g. lividomycin, neomycin, paromomycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
FI801769A 1979-06-07 1980-06-02 Foerfarande foer framstaellning av paromomycinderivat FI69082C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7919778 1979-06-07
GB7919778 1979-06-07

Publications (3)

Publication Number Publication Date
FI801769A FI801769A (fi) 1980-12-08
FI69082B FI69082B (fi) 1985-08-30
FI69082C true FI69082C (fi) 1985-12-10

Family

ID=10505676

Family Applications (1)

Application Number Title Priority Date Filing Date
FI801769A FI69082C (fi) 1979-06-07 1980-06-02 Foerfarande foer framstaellning av paromomycinderivat

Country Status (17)

Country Link
US (1) US4337248A (xx)
EP (1) EP0021150B1 (xx)
JP (1) JPS55164697A (xx)
AT (1) ATE3429T1 (xx)
AU (1) AU534470B2 (xx)
BE (1) BE883686A (xx)
CA (1) CA1137982A (xx)
CS (1) CS226412B2 (xx)
DE (1) DE3063288D1 (xx)
DK (1) DK246180A (xx)
FI (1) FI69082C (xx)
FR (1) FR2458556A1 (xx)
IE (1) IE50057B1 (xx)
IL (1) IL60217A (xx)
IT (1) IT1201934B (xx)
SU (1) SU1103796A3 (xx)
ZA (1) ZA803031B (xx)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5470836A (en) * 1988-04-29 1995-11-28 Farmitalia Carlo Erba S.R.L. Paromomycin or its derivatives or salts thereof in combination with sodium stirogluconate for parenteral treatment of human parasitic diseases
WO2004062674A2 (en) * 2003-01-07 2004-07-29 Paratek Pharmaceuticals, Inc. Substituted polyamines as inhibitors of bacterial efflux pumps
EP1957507B1 (en) 2005-12-02 2018-10-24 Ionis Pharmaceuticals, Inc. Antibacterial 4,5-substituted aminoglycoside analogs having multiple substituents
CA2684957A1 (en) 2007-04-10 2008-10-16 Achaogen Inc. Antibacterial 1,4,5-substituted aminoglycoside analogs
WO2010030704A2 (en) 2008-09-10 2010-03-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010030690A1 (en) 2008-09-10 2010-03-18 Isis Pharmaceuticals, Inc. Antibacterial 4,6-substituted 6', 6" and 1 modified aminoglycoside analogs
WO2010042851A1 (en) 2008-10-09 2010-04-15 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010042850A1 (en) 2008-10-09 2010-04-15 Achaogen, Inc. Antibacterial aminoglycoside analogs
JP2013507391A (ja) 2009-10-09 2013-03-04 アカオジェン インコーポレイテッド 抗ウイルスアミノグリコシド類似体
WO2011044538A1 (en) * 2009-10-09 2011-04-14 Achaogen, Inc. Antibacterial aminoglycoside analogs
TW201304784A (zh) 2010-11-17 2013-02-01 Achaogen Inc 抗菌性胺基糖苷類似物

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3920628A (en) * 1972-10-24 1975-11-18 Schering Corp 2{41 -Deoxyaminoglycosides and 2{41 -epi-amino-3{41 -desamino derivatives thereof, methods for their manufacture and novel intermediates useful therein
US4029883A (en) * 1972-12-29 1977-06-14 Takeda Chemical Industries, Ltd. Dehydroxylation of aminosugars
US4051315A (en) * 1974-11-13 1977-09-27 Bristol-Myers Company 6"-Deoxykanamycin B and 6"-deoxytobramycin
JPS5850235B2 (ja) * 1974-12-11 1983-11-09 明治製菓株式会社 ３′，４′−α−エポキシ−リボスタマイシン又は−カナマイシンＢの製造法
US4247687A (en) * 1979-06-12 1981-01-27 Farmitalia Carlo Erba S.P.A. Aminoglycoside antibiotic derivatives and process for their preparation

Also Published As

Publication number Publication date
EP0021150B1 (en) 1983-05-18
ZA803031B (en) 1981-05-27
AU534470B2 (en) 1984-02-02
EP0021150A1 (en) 1981-01-07
IE50057B1 (en) 1986-02-05
FR2458556A1 (fr) 1981-01-02
CA1137982A (en) 1982-12-21
DK246180A (da) 1980-12-08
FI801769A (fi) 1980-12-08
AU5895580A (en) 1980-12-11
ATE3429T1 (de) 1983-06-15
US4337248A (en) 1982-06-29
FI69082B (fi) 1985-08-30
CS226412B2 (en) 1984-03-19
IT8022594A0 (it) 1980-06-06
IE801163L (en) 1980-12-07
IL60217A (en) 1983-11-30
IT1201934B (it) 1989-02-02
DE3063288D1 (en) 1983-07-07
IL60217A0 (en) 1980-09-16
BE883686A (fr) 1980-12-08
JPS55164697A (en) 1980-12-22
SU1103796A3 (ru) 1984-07-15
FR2458556B1 (xx) 1983-07-08

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: FARMITALIA CARLO ERBA S.P.A.