FI63033C - Foerfarande foer framstaellning av anxiolytiska tranquilliserande sedativa och/eller neuroleptiska substituerade 1-piperazinyl-4h-s-triazolo(3,4-c)tieno(2,3-e)-1,4-diazepiner - Google Patents

Foerfarande foer framstaellning av anxiolytiska tranquilliserande sedativa och/eller neuroleptiska substituerade 1-piperazinyl-4h-s-triazolo(3,4-c)tieno(2,3-e)-1,4-diazepiner Download PDF

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Publication number
FI63033C
FI63033C FI782025A FI782025A FI63033C FI 63033 C FI63033 C FI 63033C FI 782025 A FI782025 A FI 782025A FI 782025 A FI782025 A FI 782025A FI 63033 C FI63033 C FI 63033C
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FI
Finland
Prior art keywords
triazolo
thieno
piperazinyl
formula
compounds
Prior art date
Application number
FI782025A
Other languages
English (en)
Finnish (fi)
Other versions
FI63033B (fi
FI782025A (fi
Inventor
Karl-Heinz Weber
Adolf Langbein
Claus Schneider
Erich Lehr
Karin Boeke
Franz Josef Kuhn
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19772732921 external-priority patent/DE2732921A1/de
Priority claimed from DE19772732943 external-priority patent/DE2732943A1/de
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Publication of FI782025A publication Critical patent/FI782025A/fi
Application granted granted Critical
Publication of FI63033B publication Critical patent/FI63033B/fi
Publication of FI63033C publication Critical patent/FI63033C/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI782025A 1977-07-21 1978-06-26 Foerfarande foer framstaellning av anxiolytiska tranquilliserande sedativa och/eller neuroleptiska substituerade 1-piperazinyl-4h-s-triazolo(3,4-c)tieno(2,3-e)-1,4-diazepiner FI63033C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE19772732921 DE2732921A1 (de) 1977-07-21 1977-07-21 Neue substituierte 1-acyl-piperidino- bzw. -piperazino-4h-s-triazolo eckige klammer auf 3,4c eckige klammer zu thieno eckige klammer auf 2,3e eckige klammer zu 1,4- diazepine, verfahren zu ihrer herstellung und pharmazeutische zusammensetzungen
DE19772732943 DE2732943A1 (de) 1977-07-21 1977-07-21 Neue substituierte 1-piperazinyl- 4h-s-triazolo eckige klammer auf 3,4c eckige klammer zu thieno eckige klammer auf 2,3e eckige klammer zu 1,4-diazepine, verfahren zu ihrer herstellung und pharmazeutische zusammensetzungen
DE2732921 1977-07-21
DE2732943 1977-07-21

Publications (3)

Publication Number Publication Date
FI782025A FI782025A (fi) 1979-01-22
FI63033B FI63033B (fi) 1982-12-31
FI63033C true FI63033C (fi) 1983-04-11

Family

ID=25772369

Family Applications (1)

Application Number Title Priority Date Filing Date
FI782025A FI63033C (fi) 1977-07-21 1978-06-26 Foerfarande foer framstaellning av anxiolytiska tranquilliserande sedativa och/eller neuroleptiska substituerade 1-piperazinyl-4h-s-triazolo(3,4-c)tieno(2,3-e)-1,4-diazepiner

Country Status (30)

Country Link
US (1) US4180573A (xx)
EP (1) EP0000479B1 (xx)
JP (1) JPS5422395A (xx)
AT (1) AT363949B (xx)
AU (1) AU515885B2 (xx)
CA (1) CA1087182A (xx)
CH (1) CH642374A5 (xx)
CS (1) CS209897B2 (xx)
DD (1) DD137934A5 (xx)
DE (1) DE2860404D1 (xx)
DK (1) DK150306C (xx)
ES (2) ES471886A1 (xx)
FI (1) FI63033C (xx)
FR (1) FR2398070A1 (xx)
GB (1) GB2001972B (xx)
GR (1) GR65022B (xx)
HU (1) HU176485B (xx)
IE (1) IE47336B1 (xx)
IL (1) IL55169A (xx)
IT (1) IT1107490B (xx)
LU (1) LU80002A1 (xx)
NL (1) NL7807762A (xx)
NO (1) NO149889C (xx)
NZ (1) NZ187915A (xx)
PH (1) PH14236A (xx)
PL (1) PL115061B1 (xx)
PT (1) PT68330A (xx)
RO (1) RO75609A (xx)
SE (1) SE439920B (xx)
SU (2) SU725564A1 (xx)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2830782A1 (de) * 1978-07-13 1980-01-24 Boehringer Sohn Ingelheim Neue substituierte 4h-s-triazolo eckige klammer auf 3,4c eckige klammer zu thieno eckige klammer auf 2,3e eckige klammer zu 1,4-diazepine, verfahren zu ihrer herstellung und pharmazeutische zusammensetzungen
EP0230942B1 (de) * 1986-01-21 1992-04-29 Boehringer Ingelheim Kg Thieno-1,4-diazepine

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH12303A (en) * 1973-02-08 1979-01-16 Hoffmann La Roche Thienotriazolodiazepine derivatives
AT338799B (de) * 1974-03-02 1977-09-12 Boehringer Sohn Ingelheim Verfahren zur herstellung neuer substituierter 6-aryl-4h-s-triazolo-(3,4c)-thieno-(2,3e)-1,4-diazepine und ihrer salze
US3894025A (en) * 1974-03-21 1975-07-08 Upjohn Co 1-Piperazino-6-phenyl-4H-s-triazolo{8 4,3-a{9 {8 1,4{9 -benzodiazepine compounds
JPS5747916B2 (xx) * 1974-05-13 1982-10-13
DE2503235A1 (de) * 1975-01-27 1976-07-29 Boehringer Sohn Ingelheim Neues verfahren zur herstellung von 8-brom-thieno-triazolo-1,4-diazepinen
DE2533924C3 (de) * 1975-07-30 1979-05-03 C.H. Boehringer Sohn, 6507 Ingelheim Verfahren zur Herstellung von 6- Aryl-4H-striazolo [3,4-c] thieno [2,3-e] 1,4-diazepinen
DE2531678C3 (de) * 1975-07-16 1979-06-28 C.H. Boehringer Sohn, 6507 Ingelheim Thieno [2,3e] triazole [3,4c] 5,6-dihydro-l,4diazepine und Verfahren zu ihrer Herstellung

Also Published As

Publication number Publication date
EP0000479A1 (de) 1979-02-07
IT1107490B (it) 1985-11-25
NO149889C (no) 1984-07-11
IL55169A0 (en) 1978-09-29
ES471886A1 (es) 1979-02-01
JPS6254114B2 (xx) 1987-11-13
SE439920B (sv) 1985-07-08
IT7850381A0 (it) 1978-07-19
AU3820978A (en) 1980-01-24
AT363949B (de) 1981-09-10
NO782499L (no) 1979-01-23
NZ187915A (en) 1980-10-08
GB2001972A (en) 1979-02-14
FI63033B (fi) 1982-12-31
NL7807762A (nl) 1979-01-23
PH14236A (en) 1981-04-09
LU80002A1 (de) 1979-09-06
GR65022B (en) 1980-06-16
US4180573A (en) 1979-12-25
RO75609A (ro) 1981-01-30
SU725564A3 (en) 1980-03-30
FR2398070B1 (xx) 1982-05-21
PT68330A (de) 1978-08-01
PL115061B1 (en) 1981-03-31
FR2398070A1 (fr) 1979-02-16
SE7808019L (sv) 1979-01-22
CA1087182A (en) 1980-10-07
DK325178A (da) 1979-01-22
EP0000479B1 (de) 1981-01-07
ES472812A1 (es) 1979-02-16
IE47336B1 (en) 1984-02-22
FI782025A (fi) 1979-01-22
JPS5422395A (en) 1979-02-20
ATA498978A (de) 1981-02-15
GB2001972B (en) 1982-01-06
AU515885B2 (en) 1981-05-07
DE2860404D1 (en) 1981-02-26
SU793402A3 (ru) 1980-12-30
DK150306B (da) 1987-02-02
CH642374A5 (de) 1984-04-13
SU725564A1 (ru) 1980-03-30
DK150306C (da) 1987-11-09
IL55169A (en) 1982-04-30
HU176485B (en) 1981-03-28
NO149889B (no) 1984-04-02
CS209897B2 (en) 1981-12-31
DD137934A5 (de) 1979-10-03
IE781456L (en) 1979-01-21
PL208542A1 (pl) 1979-06-04

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Owner name: C.H. BOEHRINGER SOHN