FI59097C - Foerfarande foer framstaellning av terapeutiskt anvaendbara pyrimido(4,5-b)kinolin-4(3h)-oni-2-karboxylsyraderivat - Google Patents

Foerfarande foer framstaellning av terapeutiskt anvaendbara pyrimido(4,5-b)kinolin-4(3h)-oni-2-karboxylsyraderivat Download PDF

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Publication number
FI59097C
FI59097C FI751628A FI751628A FI59097C FI 59097 C FI59097 C FI 59097C FI 751628 A FI751628 A FI 751628A FI 751628 A FI751628 A FI 751628A FI 59097 C FI59097 C FI 59097C
Authority
FI
Finland
Prior art keywords
quinolin
pyrimido
compounds
preparation
acid
Prior art date
Application number
FI751628A
Other languages
English (en)
Finnish (fi)
Other versions
FI59097B (fi
FI751628A (sv
Inventor
Thomas Henry Althuis
Leonard Joseph Czuba
Saul Bernard Kadin
Hans-Juergen Ernst Hess
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/485,945 external-priority patent/US3974161A/en
Application filed by Pfizer filed Critical Pfizer
Publication of FI751628A publication Critical patent/FI751628A/fi
Publication of FI59097B publication Critical patent/FI59097B/fi
Application granted granted Critical
Publication of FI59097C publication Critical patent/FI59097C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
    • C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D265/24—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in positions 2 and 4
    • C07D265/26—Two oxygen atoms, e.g. isatoic anhydride
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI751628A 1974-07-05 1975-06-03 Foerfarande foer framstaellning av terapeutiskt anvaendbara pyrimido(4,5-b)kinolin-4(3h)-oni-2-karboxylsyraderivat FI59097C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/485,945 US3974161A (en) 1974-02-20 1974-07-05 Fused pyrimidin-4(3H)-ones as antiallergy agents
US48594574 1974-07-05

Publications (3)

Publication Number Publication Date
FI751628A FI751628A (sv) 1976-01-06
FI59097B FI59097B (fi) 1981-02-27
FI59097C true FI59097C (fi) 1981-06-10

Family

ID=23930024

Family Applications (1)

Application Number Title Priority Date Filing Date
FI751628A FI59097C (fi) 1974-07-05 1975-06-03 Foerfarande foer framstaellning av terapeutiskt anvaendbara pyrimido(4,5-b)kinolin-4(3h)-oni-2-karboxylsyraderivat

Country Status (20)

Country Link
JP (1) JPS518280A (sv)
AR (1) AR214389A1 (sv)
AT (1) AT351546B (sv)
BE (1) BE829987R (sv)
BG (1) BG25226A3 (sv)
CA (1) CA1053674A (sv)
CH (1) CH619951A5 (sv)
DD (1) DD118093A6 (sv)
DE (1) DE2525050A1 (sv)
DK (1) DK250275A (sv)
ES (1) ES437966A2 (sv)
FI (1) FI59097C (sv)
GB (1) GB1501438A (sv)
IE (1) IE42746B1 (sv)
LU (1) LU72672A1 (sv)
NO (1) NO751594L (sv)
RO (1) RO69550A (sv)
SE (1) SE420610B (sv)
YU (1) YU145675A (sv)
ZA (1) ZA752908B (sv)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5510896U (sv) * 1979-08-03 1980-01-24
JPS5510894U (sv) * 1979-08-03 1980-01-24
JPS5510891U (sv) * 1979-08-03 1980-01-24
JPS5510892U (sv) * 1979-08-03 1980-01-24
JPS59210071A (ja) * 1982-12-30 1984-11-28 バイオメジヤ−・インコ−ポレ−テツド 抗ウイルス作用を有する化合物
JP2006503094A (ja) * 2002-10-16 2006-01-26 スミスクライン ビーチャム コーポレーション 化合物

Also Published As

Publication number Publication date
RO69550A (ro) 1981-08-30
GB1501438A (en) 1978-02-15
ATA432675A (de) 1979-01-15
CH619951A5 (en) 1980-10-31
YU145675A (en) 1982-08-31
SE7504599L (sv) 1976-01-07
FI59097B (fi) 1981-02-27
AU8095575A (en) 1976-11-11
NO751594L (sv) 1976-01-06
SE420610B (sv) 1981-10-19
BE829987R (fr) 1975-12-08
AR214389A1 (es) 1979-06-15
DK250275A (da) 1976-01-06
FI751628A (sv) 1976-01-06
DD118093A6 (sv) 1976-02-12
LU72672A1 (sv) 1976-03-17
JPS518280A (sv) 1976-01-23
ES437966A2 (es) 1977-02-16
AT351546B (de) 1979-07-25
BG25226A3 (en) 1978-08-10
CA1053674A (en) 1979-05-01
IE42746B1 (en) 1980-10-08
IE42746L (en) 1976-01-05
DE2525050A1 (de) 1976-01-22
ZA752908B (en) 1976-04-28

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Owner name: PFIZER INC.