FI56386C - Foerfarande foer framstaellning av oktahydro-oxazolo(3,2-a)pyrrolo(2,1-c)pyrazin-derivat - Google Patents

Foerfarande foer framstaellning av oktahydro-oxazolo(3,2-a)pyrrolo(2,1-c)pyrazin-derivat Download PDF

Info

Publication number
FI56386C
FI56386C FI2010/74A FI201074A FI56386C FI 56386 C FI56386 C FI 56386C FI 2010/74 A FI2010/74 A FI 2010/74A FI 201074 A FI201074 A FI 201074A FI 56386 C FI56386 C FI 56386C
Authority
FI
Finland
Prior art keywords
formula
benzyl
compounds
hydroxy
ester
Prior art date
Application number
FI2010/74A
Other languages
English (en)
Finnish (fi)
Other versions
FI201074A (da
FI56386B (fi
Inventor
Peter Stuetz
Paul Stadler
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of FI201074A publication Critical patent/FI201074A/fi
Application granted granted Critical
Publication of FI56386B publication Critical patent/FI56386B/fi
Publication of FI56386C publication Critical patent/FI56386C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
FI2010/74A 1973-07-09 1974-07-01 Foerfarande foer framstaellning av oktahydro-oxazolo(3,2-a)pyrrolo(2,1-c)pyrazin-derivat FI56386C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH995473 1973-07-09
CH995473 1973-07-09
CH132574 1974-01-31
CH132574 1974-01-31

Publications (3)

Publication Number Publication Date
FI201074A FI201074A (da) 1975-01-10
FI56386B FI56386B (fi) 1979-09-28
FI56386C true FI56386C (fi) 1980-01-10

Family

ID=25687336

Family Applications (1)

Application Number Title Priority Date Filing Date
FI2010/74A FI56386C (fi) 1973-07-09 1974-07-01 Foerfarande foer framstaellning av oktahydro-oxazolo(3,2-a)pyrrolo(2,1-c)pyrazin-derivat

Country Status (14)

Country Link
US (1) US4000139A (da)
JP (1) JPS5833877B2 (da)
AT (1) AT347957B (da)
DD (1) DD113235A5 (da)
DE (1) DE2431963C2 (da)
DK (1) DK140017B (da)
ES (1) ES428030A1 (da)
FI (1) FI56386C (da)
FR (1) FR2236868B1 (da)
GB (1) GB1479007A (da)
NL (1) NL7409117A (da)
SE (1) SE397093B (da)
SU (1) SU593664A3 (da)
YU (1) YU36962B (da)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH619468A5 (da) * 1976-01-12 1980-09-30 Sandoz Ag
GB1584464A (en) * 1977-04-19 1981-02-11 Farmaceutici Italia Ergot alkaloids
LU78804A1 (de) * 1977-12-30 1979-07-20 Byk Gulden Lomberg Chem Fab N-substituierte w-aminoalkanoyl-w-aminoalkansaeuren,ihre verwendung und verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel
EP0003286B1 (de) * 1978-01-20 1982-03-24 Sandoz Ag Ergopeptidalkaloid-Derivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zusammensetzungen
DE3116257A1 (de) * 1980-05-30 1982-01-07 GAO Gesellschaft für Automation und Organisation mbH, 8000 München "wertpapier mit echtheitsmerkmalen"
DE3303616A1 (de) * 1982-02-12 1983-08-25 Sandoz-Patent-GmbH, 7850 Lörrach Mutterkornalkaloide, verfahren zu deren herstellung sowie diese verbindungen enthaltende pharmazeutische zubereitungen

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3314959A (en) * 1961-05-10 1967-04-18 Sandoz Ltd Intermediates for the synthesis of ergot alkaloids
CH395119A (de) * 1961-05-10 1965-07-15 Sandoz Ag Verfahren zur Herstellung von heterocyclischen Verbindungen
DE1194868B (de) * 1961-05-10 1965-06-16 Sandoz Ag Verfahren zur Herstellung von Octahydro-oxazolo [3, 2-a] pyrrolo[2, 1-c] pyrazinderivaten
FR1583797A (da) * 1967-04-12 1969-12-05
CH541564A (de) * 1967-08-02 1973-09-15 Sandoz Ag Verfahren zur Herstellung von bisher unbekannten heterocyclischen Verbindungen
JPS4735440A (da) * 1971-03-29 1972-11-25

Also Published As

Publication number Publication date
GB1479007A (en) 1977-07-06
DD113235A5 (da) 1975-05-20
AT347957B (de) 1979-01-25
JPS5833877B2 (ja) 1983-07-22
DK140017B (da) 1979-06-05
ATA559774A (de) 1978-06-15
FI201074A (da) 1975-01-10
DE2431963C2 (de) 1986-04-17
YU189974A (en) 1982-06-18
JPS5040594A (da) 1975-04-14
US4000139A (en) 1976-12-28
SE397093B (sv) 1977-10-17
FR2236868A1 (da) 1975-02-07
SE7408688L (da) 1975-01-10
SU593664A3 (ru) 1978-02-15
AU7097874A (en) 1976-01-08
FI56386B (fi) 1979-09-28
DK352874A (da) 1975-03-03
DK140017C (da) 1979-11-05
NL7409117A (nl) 1975-01-13
ES428030A1 (es) 1976-09-16
FR2236868B1 (da) 1978-04-28
YU36962B (en) 1984-08-31
DE2431963A1 (de) 1975-01-30

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