FI113869B - Menetelmä 5,7-dihydro-3-[2-(1-bentsyylipiperidin-4-yyli)etyyli]-6H-pyrrolo[4,5-f]-1,2-bentsioksatsol-6-onin valmistamiseksi - Google Patents

Menetelmä 5,7-dihydro-3-[2-(1-bentsyylipiperidin-4-yyli)etyyli]-6H-pyrrolo[4,5-f]-1,2-bentsioksatsol-6-onin valmistamiseksi Download PDF

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Publication number
FI113869B
FI113869B FI971785A FI971785A FI113869B FI 113869 B FI113869 B FI 113869B FI 971785 A FI971785 A FI 971785A FI 971785 A FI971785 A FI 971785A FI 113869 B FI113869 B FI 113869B
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FI
Finland
Prior art keywords
compound
formula
acid
temperature
base
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Application number
FI971785A
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English (en)
Finnish (fi)
Swedish (sv)
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FI971785A0 (fi
FI971785A (fi
Inventor
Anabella Villalobos
Keith M Devries
Original Assignee
Pfizer
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Publication of FI971785A0 publication Critical patent/FI971785A0/fi
Publication of FI971785A publication Critical patent/FI971785A/fi
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Publication of FI113869B publication Critical patent/FI113869B/fi

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI971785A 1994-10-26 1997-04-25 Menetelmä 5,7-dihydro-3-[2-(1-bentsyylipiperidin-4-yyli)etyyli]-6H-pyrrolo[4,5-f]-1,2-bentsioksatsol-6-onin valmistamiseksi FI113869B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US32935294A 1994-10-26 1994-10-26
US32935294 1994-10-26
IB9500755 1995-09-13
PCT/IB1995/000755 WO1996013505A1 (fr) 1994-10-26 1995-09-13 PROCEDES ET INTERMEDIAIRES POUR PREPARER LA 5,7-DIHYDRO-3-[2{1-BENZYLPIPERIDIN-4-YL}ETHYL]-6H-PYRROLO-[4,5-f]-1,2-BENZISOXAZOL-6-ONE

Publications (3)

Publication Number Publication Date
FI971785A0 FI971785A0 (fi) 1997-04-25
FI971785A FI971785A (fi) 1997-04-25
FI113869B true FI113869B (fi) 2004-06-30

Family

ID=23284993

Family Applications (2)

Application Number Title Priority Date Filing Date
FI971785A FI113869B (fi) 1994-10-26 1997-04-25 Menetelmä 5,7-dihydro-3-[2-(1-bentsyylipiperidin-4-yyli)etyyli]-6H-pyrrolo[4,5-f]-1,2-bentsioksatsol-6-onin valmistamiseksi
FI20040505A FI115301B (fi) 1994-10-26 2004-04-06 Menetelmä 1,3-dihydro-6-hydroksi-2H-indol-2-oni-johdannaisten valmistamiseksi

Family Applications After (1)

Application Number Title Priority Date Filing Date
FI20040505A FI115301B (fi) 1994-10-26 2004-04-06 Menetelmä 1,3-dihydro-6-hydroksi-2H-indol-2-oni-johdannaisten valmistamiseksi

Country Status (10)

Country Link
EP (1) EP0788500B1 (fr)
JP (1) JP3048643B2 (fr)
AT (1) ATE260922T1 (fr)
CA (1) CA2200607C (fr)
DE (1) DE69532641T2 (fr)
DK (1) DK0788500T3 (fr)
ES (1) ES2214506T3 (fr)
FI (2) FI113869B (fr)
PT (1) PT788500E (fr)
WO (1) WO1996013505A1 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU767726B2 (en) * 1999-04-30 2003-11-20 Pfizer Products Inc. Radiotracers for in vivo study of acetylcholinesterase and Alzheimer's disease

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2188584T3 (es) * 1991-03-28 2003-07-01 Eisai Co Ltd Derivados heterociclicos de amina.

Also Published As

Publication number Publication date
DE69532641T2 (de) 2004-08-05
CA2200607C (fr) 2003-03-18
DK0788500T3 (da) 2004-06-07
JP3048643B2 (ja) 2000-06-05
EP0788500B1 (fr) 2004-03-03
FI20040505A (fi) 2004-04-06
ES2214506T3 (es) 2004-09-16
WO1996013505A1 (fr) 1996-05-09
PT788500E (pt) 2004-05-31
DE69532641D1 (de) 2004-04-08
FI971785A0 (fi) 1997-04-25
ATE260922T1 (de) 2004-03-15
JPH10502939A (ja) 1998-03-17
MX9703076A (es) 1997-07-31
FI115301B (fi) 2005-04-15
CA2200607A1 (fr) 1996-05-09
FI971785A (fi) 1997-04-25
EP0788500A1 (fr) 1997-08-13

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