DK0788500T3 - Fremgangsmåder og mellemprodukter til fremstilling af 5,7-dihydro-3-[2-(1-benzylpiperidin-4-yl)ethyl]-6H-pyrrolo-[4,5-f],2-benzisoxazol-6-on - Google Patents

Fremgangsmåder og mellemprodukter til fremstilling af 5,7-dihydro-3-[2-(1-benzylpiperidin-4-yl)ethyl]-6H-pyrrolo-[4,5-f],2-benzisoxazol-6-on

Info

Publication number
DK0788500T3
DK0788500T3 DK95929199T DK95929199T DK0788500T3 DK 0788500 T3 DK0788500 T3 DK 0788500T3 DK 95929199 T DK95929199 T DK 95929199T DK 95929199 T DK95929199 T DK 95929199T DK 0788500 T3 DK0788500 T3 DK 0788500T3
Authority
DK
Denmark
Prior art keywords
benzisoxazol
benzylpiperidin
pyrrolo
dihydro
intermediates
Prior art date
Application number
DK95929199T
Other languages
English (en)
Inventor
Keith M Devries
Anabella Villalobos
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of DK0788500T3 publication Critical patent/DK0788500T3/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK95929199T 1994-10-26 1995-09-13 Fremgangsmåder og mellemprodukter til fremstilling af 5,7-dihydro-3-[2-(1-benzylpiperidin-4-yl)ethyl]-6H-pyrrolo-[4,5-f],2-benzisoxazol-6-on DK0788500T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32935294A 1994-10-26 1994-10-26
PCT/IB1995/000755 WO1996013505A1 (en) 1994-10-26 1995-09-13 PROCESSES AND INTERMEDIATES FOR PREPARING 5,7-DIHYDRO-3-[2-{1-BENZYLPIPERIDIN-4-YL}ETHYL]-6H-PYRROLO-[4,5-f]-1,2-BENZISOXAZOL-6-ONE

Publications (1)

Publication Number Publication Date
DK0788500T3 true DK0788500T3 (da) 2004-06-07

Family

ID=23284993

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95929199T DK0788500T3 (da) 1994-10-26 1995-09-13 Fremgangsmåder og mellemprodukter til fremstilling af 5,7-dihydro-3-[2-(1-benzylpiperidin-4-yl)ethyl]-6H-pyrrolo-[4,5-f],2-benzisoxazol-6-on

Country Status (10)

Country Link
EP (1) EP0788500B1 (da)
JP (1) JP3048643B2 (da)
AT (1) ATE260922T1 (da)
CA (1) CA2200607C (da)
DE (1) DE69532641T2 (da)
DK (1) DK0788500T3 (da)
ES (1) ES2214506T3 (da)
FI (2) FI113869B (da)
PT (1) PT788500E (da)
WO (1) WO1996013505A1 (da)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1048302A3 (en) * 1999-04-30 2002-07-17 Pfizer Products Inc. Radiotracers for in vivo study of acetylcholinesterase and Alzheimer's disease

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CZ289756B6 (cs) * 1991-03-28 2002-04-17 Eisai Co., Ltd. Heterocyklicko-cyklické aminové deriváty, meziprodukty postupu přípravy těchto sloučenin, farmaceutický prostředek a pouľití uvedených derivátů

Also Published As

Publication number Publication date
JPH10502939A (ja) 1998-03-17
FI115301B (fi) 2005-04-15
FI971785A0 (fi) 1997-04-25
CA2200607C (en) 2003-03-18
FI20040505A (fi) 2004-04-06
MX9703076A (es) 1997-07-31
DE69532641T2 (de) 2004-08-05
ATE260922T1 (de) 2004-03-15
PT788500E (pt) 2004-05-31
CA2200607A1 (en) 1996-05-09
FI113869B (fi) 2004-06-30
ES2214506T3 (es) 2004-09-16
WO1996013505A1 (en) 1996-05-09
EP0788500B1 (en) 2004-03-03
JP3048643B2 (ja) 2000-06-05
FI971785A (fi) 1997-04-25
EP0788500A1 (en) 1997-08-13
DE69532641D1 (de) 2004-04-08

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