FI111130B - Menetelmä syklosporiinijohdannaista sisältävän farmaseuttisen koostumuksen valmistamiseksi - Google Patents

Menetelmä syklosporiinijohdannaista sisältävän farmaseuttisen koostumuksen valmistamiseksi Download PDF

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Publication number
FI111130B
FI111130B FI944978A FI944978A FI111130B FI 111130 B FI111130 B FI 111130B FI 944978 A FI944978 A FI 944978A FI 944978 A FI944978 A FI 944978A FI 111130 B FI111130 B FI 111130B
Authority
FI
Finland
Prior art keywords
weight
carrier medium
pharmaceutical composition
hydrophilic phase
composition
Prior art date
Application number
FI944978A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI944978A (fi
FI944978A0 (fi
Inventor
Jacky Vonderscher
Friedrich Richter
Armin Meinzer
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of FI944978A publication Critical patent/FI944978A/fi
Publication of FI944978A0 publication Critical patent/FI944978A0/fi
Application granted granted Critical
Publication of FI111130B publication Critical patent/FI111130B/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A61K38/13Cyclosporins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Dispersion Chemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Peptides Or Proteins (AREA)
FI944978A 1992-04-22 1994-10-21 Menetelmä syklosporiinijohdannaista sisältävän farmaseuttisen koostumuksen valmistamiseksi FI111130B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB9208712 1992-04-22
GB929208712A GB9208712D0 (en) 1992-04-22 1992-04-22 Pharmaceutical compositions containing cyclosporin derivates
PCT/EP1993/000955 WO1993020833A1 (en) 1992-04-22 1993-04-20 Pharmaceutical composition containing cyclosporin derivative
EP9300955 1993-04-20

Publications (3)

Publication Number Publication Date
FI944978A FI944978A (fi) 1994-10-21
FI944978A0 FI944978A0 (fi) 1994-10-21
FI111130B true FI111130B (fi) 2003-06-13

Family

ID=10714386

Family Applications (1)

Application Number Title Priority Date Filing Date
FI944978A FI111130B (fi) 1992-04-22 1994-10-21 Menetelmä syklosporiinijohdannaista sisältävän farmaseuttisen koostumuksen valmistamiseksi

Country Status (22)

Country Link
EP (1) EP0637248B1 (uk)
JP (1) JP2818298B2 (uk)
KR (2) KR950701227A (uk)
AT (1) ATE219940T1 (uk)
AU (1) AU672793B2 (uk)
CA (1) CA2132740C (uk)
CY (1) CY2399B1 (uk)
CZ (1) CZ287359B6 (uk)
DE (1) DE69332078T2 (uk)
DK (1) DK0637248T3 (uk)
ES (1) ES2179052T3 (uk)
FI (1) FI111130B (uk)
GB (1) GB9208712D0 (uk)
HU (1) HU218279B (uk)
NO (1) NO315075B1 (uk)
NZ (1) NZ252681A (uk)
PT (1) PT637248E (uk)
RU (1) RU2126263C1 (uk)
SG (1) SG50692A1 (uk)
SK (1) SK282745B6 (uk)
UA (1) UA34454C2 (uk)
WO (1) WO1993020833A1 (uk)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2222770B (en) 1988-09-16 1992-07-29 Sandoz Ltd Pharmaceutical compositions containing cyclosporins
US6007840A (en) * 1988-09-16 1999-12-28 Novartis Ag Pharmaceutical compositions comprising cyclosporins
US6262022B1 (en) 1992-06-25 2001-07-17 Novartis Ag Pharmaceutical compositions containing cyclosporin as the active agent
JP3631490B2 (ja) 1992-05-13 2005-03-23 ノバルティス ファーマ株式会社 シクロスポリン含有眼科用組成物
DK0589843T3 (da) * 1992-09-25 2002-04-02 Novartis Ag Cyclosporinholdige farmaceutiske præparater
GB2278780B (en) * 1993-05-27 1998-10-14 Sandoz Ltd Macrolide formulations
CH686761A5 (de) 1993-05-27 1996-06-28 Sandoz Ag Galenische Formulierungen.
GB2315216B (en) * 1993-10-05 1998-10-14 Ciba Geigy Ag Microemulsion preconcentrates comprising FK506 or 33-epi-chloro-33-desoxy-ascomycin
HUT77283A (hu) 1994-11-03 1998-03-30 Novartis Ag. Egyszerű összetételű, a hatóanyagot biológiailag jól hozzáférhetően tartalmazó, orális alkalmazásra szánt új ciklosporinkészítmény és eljárás az előállítására
HU215966B (hu) * 1994-11-21 1999-07-28 BIOGAL Gyógyszergyár Rt. Orálisan alkalmazható, ciklosporint tartalmazó, összetett emulzió-előkoncentrátum
US5962019A (en) * 1995-08-25 1999-10-05 Sangstat Medical Corporation Oral cyclosporin formulations
US5766629A (en) 1995-08-25 1998-06-16 Sangstat Medical Corporation Oral cyclosporin formulations
DE19544507B4 (de) 1995-11-29 2007-11-15 Novartis Ag Cyclosporin enthaltende Präparate
GB9601120D0 (en) * 1996-01-19 1996-03-20 Sandoz Ltd Organic compounds
DK0989851T3 (da) * 1997-07-29 2003-01-27 Upjohn Co Selvemulgerende formulering indeholdende sure lipofile forbindelser
CA2294031E (en) * 1997-07-29 2012-04-03 Pharmacia & Upjohn Company Self-emulsifying formulation for lipophilic compounds
US6187747B1 (en) 1997-09-08 2001-02-13 Panacea Biotech Limited Pharmaceutical composition comprising cyclosporin
US6346511B1 (en) 1997-09-08 2002-02-12 Panacea Biotec Limited Pharmaceutical composition comprising cyclosporin
US6008191A (en) * 1997-09-08 1999-12-28 Panacea Biotec Limited Pharmaceutical compositions containing cyclosporin
US6294192B1 (en) * 1999-02-26 2001-09-25 Lipocine, Inc. Triglyceride-free compositions and methods for improved delivery of hydrophobic therapeutic agents
CZ20033341A3 (cs) 2001-06-21 2004-10-13 Pfizeráproductsáinc Samoemulgující se kompozice inhibitorů přenosového proteinu cholesterylesteru
US6828301B2 (en) 2002-02-07 2004-12-07 Boehringer Ingelheim International Gmbh Pharmaceutical compositions for hepatitis C viral protease inhibitors
EP2204167A1 (en) 2009-01-05 2010-07-07 Azad Pharma AG Pharmaceutical microemulsion for preventing supramolecular aggregation of amphiphilic molecules
MA33491B1 (fr) 2009-07-07 2012-08-01 Boehringer Ingelheim Int Composition pharmaceutique pour un inhibiteur de protease virale de l'hépatite c

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2907460A1 (de) * 1978-03-07 1979-09-13 Sandoz Ag Neue resorbierbare galenische kompositionen
ATE95193T1 (de) * 1987-06-17 1993-10-15 Sandoz Ag Cyclosporine und deren benutzung als arzneimittel.
GB2222770B (en) * 1988-09-16 1992-07-29 Sandoz Ltd Pharmaceutical compositions containing cyclosporins

Also Published As

Publication number Publication date
EP0637248B1 (en) 2002-07-03
AU672793B2 (en) 1996-10-17
ATE219940T1 (de) 2002-07-15
NZ252681A (en) 1996-02-27
UA34454C2 (uk) 2001-03-15
DK0637248T3 (da) 2002-10-28
RU94046413A (ru) 1996-11-10
HU9403055D0 (en) 1994-12-28
NO315075B1 (no) 2003-07-07
NO943998D0 (no) 1994-10-21
CY2399B1 (en) 2004-09-10
SK127294A3 (en) 1995-04-12
SK282745B6 (sk) 2002-12-03
ES2179052T3 (es) 2003-01-16
DE69332078T2 (de) 2002-12-19
HUT71580A (en) 1995-12-28
KR100414853B1 (uk) 2004-01-13
PT637248E (pt) 2002-11-29
JPH07505872A (ja) 1995-06-29
EP0637248A1 (en) 1995-02-08
CA2132740C (en) 2008-01-15
CZ287359B6 (en) 2000-11-15
WO1993020833A1 (en) 1993-10-28
HU218279B (en) 2000-07-28
CZ261794A3 (en) 1995-02-15
NO943998L (no) 1994-10-21
JP2818298B2 (ja) 1998-10-30
AU4261193A (en) 1993-11-18
DE69332078D1 (de) 2002-08-08
RU2126263C1 (ru) 1999-02-20
SG50692A1 (en) 1999-05-25
FI944978A (fi) 1994-10-21
FI944978A0 (fi) 1994-10-21
GB9208712D0 (en) 1992-06-10
KR950701227A (ko) 1995-03-23
CA2132740A1 (en) 1993-10-28

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Owner name: NOVARTIS AG