ES8801650A1 - Un metodo para preparar derivados de acido (2-amino sustutuido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carboxilico. - Google Patents
Un metodo para preparar derivados de acido (2-amino sustutuido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carboxilico.Info
- Publication number
- ES8801650A1 ES8801650A1 ES557661A ES557661A ES8801650A1 ES 8801650 A1 ES8801650 A1 ES 8801650A1 ES 557661 A ES557661 A ES 557661A ES 557661 A ES557661 A ES 557661A ES 8801650 A1 ES8801650 A1 ES 8801650A1
- Authority
- ES
- Spain
- Prior art keywords
- stands
- hydrogen
- production
- organic residue
- antibiotic derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
METODO PARA LA PREPARACION DE DERIVADOS DE ACIDO (2-AMINO SUSTITUIDO-3-OXO-2-ISOXAZOLIDINIL)-5-OXO-2-TETRAHIDROFURAN-CARBOXILICO, DE FORMULA GENERAL (I). CONSISTE EN HACER REACCIONAR UN COMPUESTO DE FORMULA GENERAL (II), EN LA QUE R1 REPRESENTA UN GRUPO AMINO O UN RESTO ORGANICO UNIDO A TRAVES DE NITROGENO; R2 REPRESENTA UN GRUPO CARBOXILO; R3, R4, R5, R6, R7 Y R8 REPRESENTAN INDEPENDIENTEMENTE HIDROGENO O UN RESIDUO ORGANICO; Y X REPRESENTA HIDROGENO, METOXI O FORMILAMINO, CON UN COMPUESTO DE FORMULA GENERAL (III), EN LA QUE R2K REPRESENTA UN GRUPO DERIVABLE DEL GRUPO CARBOXILO; E Y REPRESENTA UN GRUPO ELIMINABLE, EFECTUANDOSE LA REACCION EN UN DISOLVENTE ORGANICO Y EN PRESENCIA DE UNA BASE A TEMPERATURA COMPRENDIDA ENTRE C20 Y 100 GRADOS. DE APLICACION EN MEDICINA COMO ANTIBIOTICOS.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/JP1985/000247 WO1986006380A1 (en) | 1985-04-30 | 1985-04-30 | Antibacterial compounds, use and preparation thereof |
PCT/JP1985/000394 WO1987000527A1 (en) | 1985-07-12 | 1985-07-12 | Antibacterial compounds, their use, and process for their preparation |
JP28415485 | 1985-12-16 | ||
JP61063735A JPS62228075A (ja) | 1985-04-30 | 1986-03-20 | 抗菌性化合物,その製造法および用途 |
Publications (2)
Publication Number | Publication Date |
---|---|
ES557661A0 ES557661A0 (es) | 1988-02-16 |
ES8801650A1 true ES8801650A1 (es) | 1988-02-16 |
Family
ID=27464357
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES554495A Expired ES8802317A1 (es) | 1985-04-30 | 1986-04-29 | Un procedimiento para preparar derivados de acido (2-aminosustituido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carboxilico |
ES557661A Expired ES8801650A1 (es) | 1985-04-30 | 1987-08-13 | Un metodo para preparar derivados de acido (2-amino sustutuido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carboxilico. |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES554495A Expired ES8802317A1 (es) | 1985-04-30 | 1986-04-29 | Un procedimiento para preparar derivados de acido (2-aminosustituido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carboxilico |
Country Status (6)
Country | Link |
---|---|
US (1) | US4851422A (es) |
EP (1) | EP0219923B1 (es) |
CN (1) | CN86102923A (es) |
CA (1) | CA1285950C (es) |
DE (1) | DE3686632T2 (es) |
ES (2) | ES8802317A1 (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4882434A (en) * | 1986-10-29 | 1989-11-21 | Takeda Chemical Industries, Ltd. | Gamma-lactonecarboxylic acid derivatives and their use as antibacterial agents or intermediates |
CA2305703A1 (en) | 1997-10-10 | 1999-04-22 | David W. Christianson | Compositions and methods for inhibiting arginase activity |
PL350128A1 (en) * | 1999-01-13 | 2002-11-04 | Jomaa Pharmaka Gmbh | Use of 3-isoxazolidinones and hydroxylamine acids for the treatment of infections |
AR057661A1 (es) * | 2005-07-11 | 2007-12-12 | Tanabe Seiyaku Co | Un derivado de oxima y sus preparaciones |
CA3213971A1 (en) * | 2021-03-31 | 2022-10-06 | Renata JANKOWSKA | Lactivicin compounds, their preparation and use as antibacterial agents |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1768114A1 (de) * | 1968-04-02 | 1971-10-07 | Bayer Ag | Verfahren zur Herstellung von alpha-Ketoglutarsaeure |
JPS57179133A (en) * | 1981-04-27 | 1982-11-04 | Mitsui Toatsu Chem Inc | Synthesis of gamma-ketocarboxylic acid and its ester |
IL67451A (en) * | 1981-12-25 | 1987-10-20 | Takeda Chemical Industries Ltd | 4-cyano-2-azetidinones and production thereof and process for the preparation of 4-carbamoyl-2-azetidinones using them |
US4546101A (en) * | 1982-09-10 | 1985-10-08 | Fujisawa Pharmaceutical Co., Ltd. | New cephem compounds useful for treating infectious diseases in human being and animals and processes for preparation thereof |
US4595532A (en) * | 1983-02-02 | 1986-06-17 | University Of Notre Dame Du Lac | N-(substituted-methyl)-azetidin-2-ones |
EP0146735A1 (de) * | 1983-11-23 | 1985-07-03 | F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft | Optisch einheitliche beta-Lactame |
EP0157544A3 (en) * | 1984-03-29 | 1987-08-05 | Takeda Chemical Industries, Ltd. | Antibiotics, their production and use |
JPH0473775A (ja) * | 1990-07-13 | 1992-03-09 | Mutoh Ind Ltd | 電子写真装置 |
JPH0473772A (ja) * | 1990-07-13 | 1992-03-09 | Toshiba Corp | 画像形成装置 |
-
1986
- 1986-04-16 DE DE8686302819T patent/DE3686632T2/de not_active Expired - Fee Related
- 1986-04-16 EP EP86302819A patent/EP0219923B1/en not_active Expired - Lifetime
- 1986-04-29 CA CA000507875A patent/CA1285950C/en not_active Expired - Lifetime
- 1986-04-29 ES ES554495A patent/ES8802317A1/es not_active Expired
- 1986-04-30 CN CN198686102923A patent/CN86102923A/zh active Pending
- 1986-04-30 US US06/857,834 patent/US4851422A/en not_active Expired - Fee Related
-
1987
- 1987-08-13 ES ES557661A patent/ES8801650A1/es not_active Expired
Also Published As
Publication number | Publication date |
---|---|
DE3686632T2 (de) | 1993-01-21 |
CN86102923A (zh) | 1986-11-12 |
DE3686632D1 (de) | 1992-10-08 |
EP0219923A1 (en) | 1987-04-29 |
ES8802317A1 (es) | 1988-05-01 |
EP0219923B1 (en) | 1992-09-02 |
US4851422A (en) | 1989-07-25 |
ES554495A0 (es) | 1988-05-01 |
ES557661A0 (es) | 1988-02-16 |
CA1285950C (en) | 1991-07-09 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD1A | Patent lapsed |
Effective date: 19970519 |