ES8604239A1 - Un procedimiento para la obtencion de imidazotiadiazolal- quen-carboxiamidas - Google Patents
Un procedimiento para la obtencion de imidazotiadiazolal- quen-carboxiamidasInfo
- Publication number
- ES8604239A1 ES8604239A1 ES544217A ES544217A ES8604239A1 ES 8604239 A1 ES8604239 A1 ES 8604239A1 ES 544217 A ES544217 A ES 544217A ES 544217 A ES544217 A ES 544217A ES 8604239 A1 ES8604239 A1 ES 8604239A1
- Authority
- ES
- Spain
- Prior art keywords
- opt
- alkyl
- substd
- aryl
- ring
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
PROCEDIMIENTO PARA LA OBTENCION DE IMIDAZOTIADIAZOLAL-QUENCARBOXIAMIDAS, DE SUS FORMAS ESTEREOISOMERAS DE LOS ENANTIOMEROS, DIASTEREOMEROS E ISOMEROS E/Z Y DE SUS SALES DE ADICION DE ACIDO FISIOLOGICAMENTE COMPATIBLES DE FORMULA (I), EN LA QUE A Y R1-R7 PUEDEN SER VARIOS TIPOS DE RADICALES. COMPRENDE LA REACCION DE IMIDAZOTIADIAZOL-ALQUENCARBOXIAMIDAS, DE FORMULA (II), CON UNA AMINA DE FORMULA R1R2NH, EN LAS QUE HAL ES UN ATOMO DE CLORO, BROMO O YODO, Y LOS DEMAS SIMBOLOS TIENEN EL MISMO SIGNIFICADO QUE EN LA FORMULA (I). LA REACCION SE LLEVA A CABO EN UN DISOLVENTE ORGANICO INERTE, EN PRESENCIA DE UNA BASE, A TEMPERATURA COMPRENDIDA ENTRE 0JC Y 150JC. ESTOS COMPUESTOS TIENEN APLICACIONES FARMACOLOGICAS COMO ANTIHIPERTENSIVOS, DIURETICOS Y URICOSURICOS.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE3329621A DE3329621A1 (de) | 1983-08-17 | 1983-08-17 | Aminoalkyl-imidazothiadiazol-alkencarbonsaeureamide, neue zwischenprodukte zu ihrer herstellung, ihre herstellung und ihre verwendung in arzneimitteln |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES544217A0 ES544217A0 (es) | 1986-01-16 |
| ES8604239A1 true ES8604239A1 (es) | 1986-01-16 |
Family
ID=6206712
Family Applications (7)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES535054A Granted ES535054A0 (es) | 1983-08-17 | 1984-08-10 | Imidazotiadiazolalquencarboxiamidas |
| ES544216A Expired ES8604238A1 (es) | 1983-08-17 | 1985-06-14 | Un procedimiento para la obtencion de imidazotiadiazolal- quen-carboxiamidas |
| ES544215A Expired ES8604237A1 (es) | 1983-08-17 | 1985-06-14 | Un procedimiento para la obtencion de imidazotiadiazolal- quen-carboxiamidas |
| ES544217A Expired ES8604239A1 (es) | 1983-08-17 | 1985-06-14 | Un procedimiento para la obtencion de imidazotiadiazolal- quen-carboxiamidas |
| ES544218A Expired ES8604240A1 (es) | 1983-08-17 | 1985-06-14 | Un procedimiento para la obtencion de carbonil compuestos |
| ES544220A Expired ES8604242A1 (es) | 1983-08-17 | 1985-06-14 | Un procedimiento para la obtencion de acidos alquencarboxi- licos |
| ES544219A Expired ES8604241A1 (es) | 1983-08-17 | 1985-06-14 | Un procedimiento para la obtencion de acidos alquencarboxi- licos |
Family Applications Before (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES535054A Granted ES535054A0 (es) | 1983-08-17 | 1984-08-10 | Imidazotiadiazolalquencarboxiamidas |
| ES544216A Expired ES8604238A1 (es) | 1983-08-17 | 1985-06-14 | Un procedimiento para la obtencion de imidazotiadiazolal- quen-carboxiamidas |
| ES544215A Expired ES8604237A1 (es) | 1983-08-17 | 1985-06-14 | Un procedimiento para la obtencion de imidazotiadiazolal- quen-carboxiamidas |
Family Applications After (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES544218A Expired ES8604240A1 (es) | 1983-08-17 | 1985-06-14 | Un procedimiento para la obtencion de carbonil compuestos |
| ES544220A Expired ES8604242A1 (es) | 1983-08-17 | 1985-06-14 | Un procedimiento para la obtencion de acidos alquencarboxi- licos |
| ES544219A Expired ES8604241A1 (es) | 1983-08-17 | 1985-06-14 | Un procedimiento para la obtencion de acidos alquencarboxi- licos |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US4588723A (es) |
| EP (1) | EP0141072A3 (es) |
| JP (1) | JPS6058989A (es) |
| KR (1) | KR850001762A (es) |
| AU (1) | AU3111184A (es) |
| CA (1) | CA1234113A (es) |
| DE (1) | DE3329621A1 (es) |
| DK (1) | DK394384A (es) |
| ES (7) | ES535054A0 (es) |
| FI (1) | FI843226A (es) |
| GR (1) | GR80133B (es) |
| HU (1) | HU190969B (es) |
| IL (1) | IL72678A0 (es) |
| NO (1) | NO843108L (es) |
| PT (1) | PT79084B (es) |
| ZA (1) | ZA846378B (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0232612B1 (en) * | 1985-12-23 | 1990-04-04 | Dr. Lo. Zambeletti S.p.A. | Azacyclic compounds, processes for their preparation, and their use as pharmaceuticals |
| DE102005010215A1 (de) * | 2005-03-05 | 2006-09-07 | Bayer Cropscience Ag | Heterobicyclische Acrylamide |
| EP2682395A1 (en) * | 2012-07-04 | 2014-01-08 | Laboratorios Del. Dr. Esteve, S.A. | Imidazo[2,1-b]thiazole derivatives, their preparation and use as medicaments |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NO811630L (no) * | 1980-05-29 | 1981-11-30 | Bayer Ag | Imidazoazolalkensyreamider, nye mellomprodukter for deres fremstilling, deres fremstilling og deres anvendelse som legemiddel |
-
1983
- 1983-08-17 DE DE3329621A patent/DE3329621A1/de not_active Withdrawn
-
1984
- 1984-07-24 AU AU31111/84A patent/AU3111184A/en not_active Abandoned
- 1984-07-26 US US06/634,851 patent/US4588723A/en not_active Expired - Fee Related
- 1984-08-02 NO NO843108A patent/NO843108L/no unknown
- 1984-08-06 EP EP84109291A patent/EP0141072A3/de not_active Withdrawn
- 1984-08-10 ES ES535054A patent/ES535054A0/es active Granted
- 1984-08-14 IL IL72678A patent/IL72678A0/xx unknown
- 1984-08-14 PT PT79084A patent/PT79084B/pt unknown
- 1984-08-15 FI FI843226A patent/FI843226A/fi not_active Application Discontinuation
- 1984-08-15 CA CA000461031A patent/CA1234113A/en not_active Expired
- 1984-08-16 JP JP59170086A patent/JPS6058989A/ja active Pending
- 1984-08-16 HU HU843114A patent/HU190969B/hu unknown
- 1984-08-16 ZA ZA846378A patent/ZA846378B/xx unknown
- 1984-08-16 KR KR1019840004913A patent/KR850001762A/ko not_active Application Discontinuation
- 1984-08-16 DK DK394384A patent/DK394384A/da not_active Application Discontinuation
- 1984-08-17 GR GR80133A patent/GR80133B/el unknown
-
1985
- 1985-06-14 ES ES544216A patent/ES8604238A1/es not_active Expired
- 1985-06-14 ES ES544215A patent/ES8604237A1/es not_active Expired
- 1985-06-14 ES ES544217A patent/ES8604239A1/es not_active Expired
- 1985-06-14 ES ES544218A patent/ES8604240A1/es not_active Expired
- 1985-06-14 ES ES544220A patent/ES8604242A1/es not_active Expired
- 1985-06-14 ES ES544219A patent/ES8604241A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| ES544215A0 (es) | 1986-01-16 |
| ES8600768A1 (es) | 1985-10-16 |
| ES544217A0 (es) | 1986-01-16 |
| US4588723A (en) | 1986-05-13 |
| EP0141072A3 (de) | 1986-01-08 |
| EP0141072A2 (de) | 1985-05-15 |
| ES8604237A1 (es) | 1986-01-16 |
| ES544219A0 (es) | 1986-01-16 |
| HU190969B (en) | 1986-12-28 |
| ES535054A0 (es) | 1985-10-16 |
| HUT36130A (en) | 1985-08-28 |
| ES544220A0 (es) | 1986-01-16 |
| KR850001762A (ko) | 1985-04-01 |
| JPS6058989A (ja) | 1985-04-05 |
| IL72678A0 (en) | 1984-11-30 |
| FI843226A (fi) | 1985-02-18 |
| ES544218A0 (es) | 1986-01-16 |
| FI843226A0 (fi) | 1984-08-15 |
| CA1234113A (en) | 1988-03-15 |
| AU3111184A (en) | 1985-02-21 |
| DK394384A (da) | 1985-02-18 |
| GR80133B (en) | 1984-12-19 |
| ZA846378B (en) | 1985-05-29 |
| ES8604238A1 (es) | 1986-01-16 |
| ES544216A0 (es) | 1986-01-16 |
| PT79084B (en) | 1986-08-14 |
| DE3329621A1 (de) | 1985-02-28 |
| ES8604240A1 (es) | 1986-01-16 |
| ES8604242A1 (es) | 1986-01-16 |
| NO843108L (no) | 1985-02-18 |
| DK394384D0 (da) | 1984-08-16 |
| ES8604241A1 (es) | 1986-01-16 |
| PT79084A (en) | 1984-09-01 |
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