ES8506009A1 - Un procedimiento para la preparacion de derivados de oxacefalosporina - Google Patents
Un procedimiento para la preparacion de derivados de oxacefalosporinaInfo
- Publication number
- ES8506009A1 ES8506009A1 ES527804A ES527804A ES8506009A1 ES 8506009 A1 ES8506009 A1 ES 8506009A1 ES 527804 A ES527804 A ES 527804A ES 527804 A ES527804 A ES 527804A ES 8506009 A1 ES8506009 A1 ES 8506009A1
- Authority
- ES
- Spain
- Prior art keywords
- hydrogen
- protecting group
- derivatives
- preparation
- combating
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 229910052739 hydrogen Inorganic materials 0.000 abstract 3
- 239000001257 hydrogen Substances 0.000 abstract 3
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
- 241000894006 Bacteria Species 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 230000003115 biocidal effect Effects 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000009472 formulation Methods 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical group 0.000 abstract 1
- 125000001072 heteroaryl group Chemical group 0.000 abstract 1
- 150000002431 hydrogen Chemical class 0.000 abstract 1
- 208000015181 infectious disease Diseases 0.000 abstract 1
- 239000002184 metal Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- JUJWROOIHBZHMG-UHFFFAOYSA-O pyridinium Chemical group C1=CC=[NH+]C=C1 JUJWROOIHBZHMG-UHFFFAOYSA-O 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP57214112A JPS59104389A (ja) | 1982-12-06 | 1982-12-06 | オキサセファム誘導体 |
Publications (2)
Publication Number | Publication Date |
---|---|
ES527804A0 ES527804A0 (es) | 1985-06-16 |
ES8506009A1 true ES8506009A1 (es) | 1985-06-16 |
Family
ID=16650427
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES527804A Expired ES8506009A1 (es) | 1982-12-06 | 1983-12-05 | Un procedimiento para la preparacion de derivados de oxacefalosporina |
Country Status (8)
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6489319B2 (en) * | 1999-08-16 | 2002-12-03 | Revaax Pharmaceuticals, Llc | Neurotherapeutic use of carboxypeptidase inhibitors |
US6426342B2 (en) * | 1999-08-16 | 2002-07-30 | Revaax Pharmaceuticals, Llc | Use of β-lactamase inhibitors as neuroprotectants |
US6610681B1 (en) * | 1999-08-16 | 2003-08-26 | Revaax Pharmaceuticals, Llc | Neurotherapeutic clavulanate composition and method |
JP2004168775A (ja) * | 2002-11-08 | 2004-06-17 | Orchid Chemicals & Pharmaceuticals Ltd | オキサセファロスポリンの改良合成法 |
KR100749163B1 (ko) | 2005-11-10 | 2007-08-14 | 주식회사 엔지켐 | 7α-메톡시옥사세펨 유도체의 제조방법 |
KR20120012823A (ko) * | 2009-04-29 | 2012-02-10 | 렉산 파마슈티컬스, 인코포레이티드 | 신경보호 및 퇴행성 신경 질환 치료용 클라블라네이트 제제 |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NL7314706A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * | 1972-11-06 | 1974-05-08 | ||
NL178005C (nl) * | 1972-11-06 | 1986-01-02 | Merck & Co Inc | Werkwijze voor het bereiden van een farmaceutisch preparaat met antibacteriele werking, alsmede werkwijze ter bereiding van een cefalosporine-antibioticum. |
GB1510794A (en) * | 1974-08-06 | 1978-05-17 | Univ Kingston | 1-oxacephems and intermediates therefor |
US4096329A (en) * | 1976-03-05 | 1978-06-20 | E. R. Squibb & Sons, Inc. | 7-Cyanoalkylureido 3 heterocylic thio methyl cephalosporins |
JPS609515B2 (ja) * | 1976-08-09 | 1985-03-11 | 塩野義製薬株式会社 | 3′−ノルオキサセファロスポリン類 |
JPS5331690A (en) * | 1976-09-01 | 1978-03-25 | Shionogi & Co Ltd | Oxadithiacephalosporins |
DE2714880A1 (de) * | 1977-04-02 | 1978-10-26 | Hoechst Ag | Cephemderivate und verfahren zu ihrer herstellung |
JPS5419990A (en) * | 1977-07-14 | 1979-02-15 | Shionogi & Co Ltd | Dihydrotriazinylthioxacephalosporin |
JPS54117494A (en) * | 1978-03-03 | 1979-09-12 | Takeda Chem Ind Ltd | Cephalosporin compound and its preparation |
JPS56103185A (en) * | 1980-01-22 | 1981-08-18 | Shionogi & Co Ltd | Malonamidoxa-dethia-cephem compound |
DE3045331A1 (de) * | 1980-12-02 | 1982-07-01 | Dr. Karl Thomae Gmbh, 7950 Biberach | Neue cephalosporine, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
DE3047082A1 (de) * | 1980-12-13 | 1982-07-29 | Dr. Karl Thomae Gmbh, 7950 Biberach | Neue cephalosporine, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
-
1982
- 1982-12-06 JP JP57214112A patent/JPS59104389A/ja active Granted
-
1983
- 1983-12-05 ES ES527804A patent/ES8506009A1/es not_active Expired
- 1983-12-05 US US06/559,293 patent/US4529722A/en not_active Expired - Lifetime
- 1983-12-06 DE DE8383307426T patent/DE3365480D1/de not_active Expired
- 1983-12-06 EP EP83307426A patent/EP0111421B1/en not_active Expired
- 1983-12-06 KR KR1019830005770A patent/KR840007005A/ko not_active Withdrawn
- 1983-12-06 CA CA000442647A patent/CA1209997A/en not_active Expired
- 1983-12-06 GB GB08332551A patent/GB2131803B/en not_active Expired
Also Published As
Publication number | Publication date |
---|---|
CA1209997A (en) | 1986-08-19 |
GB2131803A (en) | 1984-06-27 |
ES527804A0 (es) | 1985-06-16 |
EP0111421B1 (en) | 1986-08-20 |
GB8332551D0 (en) | 1984-01-11 |
GB2131803B (en) | 1986-06-04 |
US4529722A (en) | 1985-07-16 |
KR840007005A (ko) | 1984-12-04 |
JPH0354673B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1991-08-20 |
DE3365480D1 (en) | 1986-09-25 |
JPS59104389A (ja) | 1984-06-16 |
EP0111421A1 (en) | 1984-06-20 |
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