ES546799A0 - Procedimiento para la obtencion de formulaciones medicionales solidas de nitrendipina cristalina. - Google Patents

Procedimiento para la obtencion de formulaciones medicionales solidas de nitrendipina cristalina.

Info

Publication number
ES546799A0
ES546799A0 ES546799A ES546799A ES546799A0 ES 546799 A0 ES546799 A0 ES 546799A0 ES 546799 A ES546799 A ES 546799A ES 546799 A ES546799 A ES 546799A ES 546799 A0 ES546799 A0 ES 546799A0
Authority
ES
Spain
Prior art keywords
weight
nitrendipine
crystal
procedure
parts
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES546799A
Other languages
English (en)
Other versions
ES8800153A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=6245068&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ES546799(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer AG filed Critical Bayer AG
Publication of ES546799A0 publication Critical patent/ES546799A0/es
Publication of ES8800153A1 publication Critical patent/ES8800153A1/es
Expired legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Hydrogenated Pyridines (AREA)
ES546799A 1984-09-11 1985-09-09 Procedimiento para la obtencion de formulaciones medicionales solidas de nitrendipina cristalina. Expired ES8800153A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19843433239 DE3433239A1 (de) 1984-09-11 1984-09-11 Feste arzneizubereitung enthaltend nitrendipin und verfahren zu ihrer herstellung

Publications (2)

Publication Number Publication Date
ES546799A0 true ES546799A0 (es) 1987-10-16
ES8800153A1 ES8800153A1 (es) 1987-10-16

Family

ID=6245068

Family Applications (1)

Application Number Title Priority Date Filing Date
ES546799A Expired ES8800153A1 (es) 1984-09-11 1985-09-09 Procedimiento para la obtencion de formulaciones medicionales solidas de nitrendipina cristalina.

Country Status (13)

Country Link
US (1) US4724141A (es)
EP (1) EP0176773B1 (es)
JP (1) JPH0761960B2 (es)
KR (1) KR920006909B1 (es)
AT (1) ATE48943T1 (es)
AU (1) AU578114B2 (es)
CA (1) CA1261271A (es)
DE (2) DE3433239A1 (es)
DK (1) DK411485A (es)
ES (1) ES8800153A1 (es)
GR (1) GR852176B (es)
IL (1) IL76332A0 (es)
ZA (1) ZA856916B (es)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1178511B (it) * 1984-09-14 1987-09-09 Pharmatec Spa Procedimento per la preparazione di una forma solida per uso orale a base di nifedipina con rilascio
US4771057A (en) * 1986-02-03 1988-09-13 University Of Alberta Reduced pyridyl derivatives with cardiovascular regulating properties
DE3639073A1 (de) * 1986-11-14 1988-05-26 Klinge Co Chem Pharm Fab Feste arzneizubereitungen und verfahren zu ihrer herstellung
US5571827A (en) * 1990-03-13 1996-11-05 Sepracor Inc. Methods and compositions for treating hypertension, angina and other disorders using optically pure s(-) nitrendipine
US5190962A (en) * 1990-03-13 1993-03-02 Sepracor, Inc. Treating hypertension
FR2661611B1 (fr) * 1990-05-04 1994-11-18 Theramex Nouvelles compositions pharmaceutiques a base de polycarbophil et leur procede d'obtention.
SI9300504A (en) * 1993-09-28 1995-04-30 Krka Process for preparation solid dispersions and deposits of calcium antagonist dihidropyrimidine derivates and pharmaceutical compositions comprising the same
JP2713549B2 (ja) * 1994-05-17 1998-02-16 財団法人工業技術研究院 防湿性漢方製剤
JP2656727B2 (ja) * 1994-05-17 1997-09-24 財団法人工業技術研究院 防湿性漢方顆粒製剤
AU776299B2 (en) * 1998-12-01 2004-09-02 Dr Reddy's Laboratories, Inc. New pharmaceutical composition and the process for its preparation
JP4748839B2 (ja) * 1999-03-25 2011-08-17 大塚製薬株式会社 シロスタゾール製剤
EG23951A (en) * 1999-03-25 2008-01-29 Otsuka Pharma Co Ltd Cilostazol preparation
AU2256702A (en) 2000-12-01 2002-06-11 Kyowa Hakko Kogyo Kk Composition improved in solubility or oral absorbability
FR2827517B1 (fr) 2001-07-23 2003-10-24 Bioalliance Pharma Systemes therapeutiques bioadhesifs a liberation prolongee
DE10355461A1 (de) 2003-11-27 2005-06-23 Bayer Healthcare Ag Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung
EP1837020A1 (en) 2006-03-24 2007-09-26 Bioalliance Pharma Mucosal bioadhesive slow release carrier for delivering active principles
EP3002005A1 (en) * 2014-09-30 2016-04-06 Molkerei Meggle Wasserburg GmbH & Co. Kg Direct compression excipient based on lactose, cellulose and starch
US11883404B2 (en) 2016-03-04 2024-01-30 Taiho Pharmaceuticals Co., Ltd. Preparation and composition for treatment of malignant tumors
EP3424505A4 (en) 2016-03-04 2019-10-16 Taiho Pharmaceutical Co., Ltd. PREPARATION AND COMPOSITION FOR TREATING MALIGNANT TUMORS
WO2019181876A1 (ja) * 2018-03-19 2019-09-26 大鵬薬品工業株式会社 アルキル硫酸ナトリウムを含む医薬組成物

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2837477A1 (de) * 1978-08-28 1980-03-13 Bayer Ag Sila-substituierte 1,4-dihydropyridin- derivate
JPS5547615A (en) * 1978-09-29 1980-04-04 Taiyo Yakuhin Kogyo Kk Stable solid drug of nifedipine
JPS56110612A (en) * 1980-02-08 1981-09-01 Yamanouchi Pharmaceut Co Ltd Readily disintegrable and absorbable compression molded article of slightly soluble drug
DE3142853A1 (de) * 1981-10-29 1983-05-11 Bayer Ag, 5090 Leverkusen Feste arzneizubereitungen mit nifedipin und verfahren zu ihrer herstellung
DE3212736A1 (de) * 1982-04-06 1983-10-13 Bayer Ag, 5090 Leverkusen Verwendung von dihydropyridinen in arzneimitteln mit salidiuretischer wirkung
DE3307422A1 (de) * 1983-03-03 1984-09-06 Bayer Ag, 5090 Leverkusen Fluessigzubereitungen von dihydropyridinen, ein verfahren zu ihrer herstellung, sowie ihre verwendung bei der bekaempfung von erkrankungen

Also Published As

Publication number Publication date
CA1261271A (en) 1989-09-26
DE3574933D1 (de) 1990-02-01
DK411485D0 (da) 1985-09-10
ES8800153A1 (es) 1987-10-16
US4724141A (en) 1988-02-09
DE3433239A1 (de) 1986-03-20
JPS6168431A (ja) 1986-04-08
JPH0761960B2 (ja) 1995-07-05
EP0176773B1 (de) 1989-12-27
IL76332A0 (en) 1986-01-31
ATE48943T1 (de) 1990-01-15
GR852176B (es) 1986-01-10
KR860002270A (ko) 1986-04-24
EP0176773A1 (de) 1986-04-09
ZA856916B (en) 1986-04-30
DK411485A (da) 1986-03-12
AU4733585A (en) 1986-03-20
AU578114B2 (en) 1988-10-13
KR920006909B1 (ko) 1992-08-22

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970401