ES544526A0 - Un procedimiento para la preparacion de nuevos derivados de bencenosulfonamida - Google Patents

Un procedimiento para la preparacion de nuevos derivados de bencenosulfonamida

Info

Publication number
ES544526A0
ES544526A0 ES544526A ES544526A ES544526A0 ES 544526 A0 ES544526 A0 ES 544526A0 ES 544526 A ES544526 A ES 544526A ES 544526 A ES544526 A ES 544526A ES 544526 A0 ES544526 A0 ES 544526A0
Authority
ES
Spain
Prior art keywords
procedure
preparation
benzene sulfonamide
sulfonamide derivatives
new benzene
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES544526A
Other languages
English (en)
Other versions
ES8604128A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of ES544526A0 publication Critical patent/ES544526A0/es
Publication of ES8604128A1 publication Critical patent/ES8604128A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/50Compounds containing any of the groups, X being a hetero atom, Y being any atom
    • C07C311/52Y being a hetero atom
    • C07C311/54Y being a hetero atom either X or Y, but not both, being nitrogen atoms, e.g. N-sulfonylurea
    • C07C311/57Y being a hetero atom either X or Y, but not both, being nitrogen atoms, e.g. N-sulfonylurea having sulfur atoms of the sulfonylurea groups bound to carbon atoms of six-membered aromatic rings
    • C07C311/60Y being a hetero atom either X or Y, but not both, being nitrogen atoms, e.g. N-sulfonylurea having sulfur atoms of the sulfonylurea groups bound to carbon atoms of six-membered aromatic rings having nitrogen atoms of the sulfonylurea groups bound to carbon atoms of six-membered aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES544526A 1984-06-27 1985-06-25 Un procedimiento para la preparacion de nuevos derivados de bencenosulfonamida Expired ES8604128A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US62528084A 1984-06-27 1984-06-27

Publications (2)

Publication Number Publication Date
ES544526A0 true ES544526A0 (es) 1986-01-16
ES8604128A1 ES8604128A1 (es) 1986-01-16

Family

ID=24505356

Family Applications (1)

Application Number Title Priority Date Filing Date
ES544526A Expired ES8604128A1 (es) 1984-06-27 1985-06-25 Un procedimiento para la preparacion de nuevos derivados de bencenosulfonamida

Country Status (19)

Country Link
US (1) US4845128A (es)
EP (1) EP0166615B1 (es)
JP (1) JPH0714881B2 (es)
KR (1) KR870000741B1 (es)
CN (1) CN1006548B (es)
AR (1) AR240916A1 (es)
AT (1) ATE89733T1 (es)
AU (1) AU571706B2 (es)
CA (1) CA1291163C (es)
DE (1) DE3587359T2 (es)
DK (1) DK288785A (es)
ES (1) ES8604128A1 (es)
GR (1) GR851538B (es)
HU (1) HU197298B (es)
IL (1) IL75616A0 (es)
NZ (1) NZ212521A (es)
PH (1) PH22825A (es)
PT (1) PT80708B (es)
ZA (1) ZA854744B (es)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5110830A (en) * 1984-06-27 1992-05-05 Eli Lilly And Company Benzenesulfonamides treatment of tumors susceptible to
US5260338A (en) * 1984-06-27 1993-11-09 Eli Lilly And Company Anti-tumor method and compounds
GR862353B (en) * 1985-09-23 1987-01-19 Lilly Co Eli Anti-tumor method and compounds
US5116874A (en) * 1985-09-23 1992-05-26 Eli Lilly And Company Anti-tumor method and compounds
US5216026A (en) * 1990-07-17 1993-06-01 Eli Lilly And Company Antitumor compositions and methods of treatment
NZ238911A (en) * 1990-07-17 1993-10-26 Lilly Co Eli Furyl, pyrrolyl and thienyl sulphonyl urea derivatives, pharmaceutical compositions and intermediates therefor
EP0493642A1 (en) * 1991-01-02 1992-07-08 Takeo Dr. Takayanagi Novel sulfonyl derivatives
US5254589A (en) * 1991-10-15 1993-10-19 Warner-Lambert Company Sulfonyl urea and carbamate ACAT inhibitors
US5262440A (en) * 1991-12-10 1993-11-16 Eli Lilly And Company Antitumor compositions and methods of treatment
US5258406A (en) * 1991-12-20 1993-11-02 Eli Lilly And Company Sulfonimidamides
US5234955A (en) * 1991-12-20 1993-08-10 Eli Lilly And Company Antitumor compositions and methods of treatment
US5254582A (en) * 1992-02-05 1993-10-19 Eli Lilly And Company Antitumor compositions and methods
US5169860A (en) * 1992-03-13 1992-12-08 Eli Lilly And Company Antitumor compositions and methods of treatment
US5387681A (en) * 1992-08-19 1995-02-07 Eli Lilly And Company Synthesis of bicyclic aromatic sulfonic acids sulfonyl chlorides and sulfonamides
US5270329A (en) * 1992-12-10 1993-12-14 Eli Lilly And Company Antitumor compositions and methods of treatment
CA2110524A1 (en) * 1992-12-10 1994-06-11 Gerald Burr Grindey Antitumor compositions and methods of treatment
US5529999A (en) * 1994-03-04 1996-06-25 Eli Lilly And Company Antitumor compositions and methods of treatment
JP3025860U (ja) * 1995-09-18 1996-06-25 将一 川▲崎▼ 野良猫回避板
ATE208774T1 (de) * 1996-08-22 2001-11-15 Dong Wha Pharm Ind Co Ltd Arylsulfonylimidazolon-derivate als antitumormittel
AU4734997A (en) * 1996-10-04 1998-04-24 Eli Lilly And Company Antitumor compositions and methods of treatment
WO1998014440A1 (en) * 1996-10-04 1998-04-09 Eli Lilly And Company Antitumor compositions and methods of treatment
US6174921B1 (en) 1997-10-02 2001-01-16 Eli Lilly And Company Antitumor compositions and methods of treatment
EA005810B1 (ru) * 2001-06-06 2005-06-30 Эли Лилли Энд Компани Бензоилсульфонамиды и сульфонилбензамидины для применения в качестве противоопухолевых агентов
AU2003224917A1 (en) * 2002-04-11 2003-10-27 Carbomer Diabetes imaging probes
WO2011009059A2 (en) * 2009-07-17 2011-01-20 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Method of treating or preventing cancer
CN114761379A (zh) * 2019-11-28 2022-07-15 三菱化学株式会社 显色剂及热敏记录材料

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1144259B (de) * 1956-05-29 1963-02-28 Hoechst Ag Verfahren zur Herstellung von Sulfonylharnstoffen
US3097241A (en) * 1956-08-10 1963-07-09 Hoechst Ag Nu-cyclohexane-sulphonyl-n'-(beta-phenylethyl)-urea
DE1159937B (de) * 1960-06-29 1963-12-27 Heyden Chem Fab Verfahren zur Herstellung von Hydrindensulfonylharnstoffen
US3097242A (en) * 1960-06-29 1963-07-09 Olin Mathieson Hydrindene sulfonylureas
DE1240866B (de) * 1961-06-29 1967-05-24 Heyden Chem Fab Verfahren zur Herstellung von Indolin-6-sulfonylharnstoffen
US3849110A (en) * 1963-01-07 1974-11-19 Lilly Co Eli Herbicidal method employing aryl-sulfonylureas or salts thereof
US3736122A (en) * 1969-04-10 1973-05-29 C Tung Method of controlling plant growth
US4276290A (en) * 1977-10-10 1981-06-30 Rohm And Haas Company Phosphonoureide and phosphonothioureide anthelmintics
US4634465A (en) * 1982-07-16 1987-01-06 Ciba-Geigy Corporation Fused N-phenylsulfonyl-N'-pyrimidinylureas and N-phenylsulfonyl-N'triazinylureas
IT1161220B (it) * 1983-04-21 1987-03-18 Montedison Spa Diidro-benzofurano derivati ad attivita' erbicida
CA1208561A (en) * 1984-01-19 1986-07-29 Marius S. Brouwer Pharmaceutical compositions containing benzoylurea compounds
GR862353B (en) * 1985-09-23 1987-01-19 Lilly Co Eli Anti-tumor method and compounds

Also Published As

Publication number Publication date
PT80708A (en) 1985-07-01
KR860000253A (ko) 1986-01-27
EP0166615A3 (en) 1990-03-21
PH22825A (en) 1989-01-19
GR851538B (es) 1985-11-25
DK288785A (da) 1985-12-28
DE3587359D1 (de) 1993-07-01
HU197298B (en) 1989-03-28
HUT38093A (en) 1986-04-28
KR870000741B1 (ko) 1987-04-13
CA1291163C (en) 1991-10-22
AU4419285A (en) 1986-01-02
DE3587359T2 (de) 1993-11-04
JPH0714881B2 (ja) 1995-02-22
DK288785D0 (da) 1985-06-26
EP0166615A2 (en) 1986-01-02
ZA854744B (en) 1987-02-25
CN85104893A (zh) 1987-01-07
JPS6118754A (ja) 1986-01-27
ES8604128A1 (es) 1986-01-16
IL75616A0 (en) 1985-10-31
EP0166615B1 (en) 1993-05-26
NZ212521A (en) 1989-02-24
CN1006548B (zh) 1990-01-24
PT80708B (pt) 1987-10-20
US4845128A (en) 1989-07-04
ATE89733T1 (de) 1993-06-15
AU571706B2 (en) 1988-04-21
AR240916A2 (es) 1991-03-27
AR240916A1 (es) 1991-03-27

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