ES533873A0 - Un procedimiento para preparar profarmacos de alopurinol - Google Patents

Un procedimiento para preparar profarmacos de alopurinol

Info

Publication number
ES533873A0
ES533873A0 ES533873A ES533873A ES533873A0 ES 533873 A0 ES533873 A0 ES 533873A0 ES 533873 A ES533873 A ES 533873A ES 533873 A ES533873 A ES 533873A ES 533873 A0 ES533873 A0 ES 533873A0
Authority
ES
Spain
Prior art keywords
alopurinol
drugs
preparing
procedure
preparing alopurinol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES533873A
Other languages
English (en)
Other versions
ES8600293A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
A-S GEA
Hexal AS
Original Assignee
A-S GEA
Gea AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by A-S GEA, Gea AS filed Critical A-S GEA
Publication of ES533873A0 publication Critical patent/ES533873A0/es
Publication of ES8600293A1 publication Critical patent/ES8600293A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ES533873A 1983-06-30 1984-06-29 Un procedimiento para preparar profarmacos de alopurinol Expired ES8600293A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK3028/83A DK302883D0 (da) 1983-06-30 1983-06-30 Allopurinol prodrugs

Publications (2)

Publication Number Publication Date
ES533873A0 true ES533873A0 (es) 1985-10-01
ES8600293A1 ES8600293A1 (es) 1985-10-01

Family

ID=8118314

Family Applications (1)

Application Number Title Priority Date Filing Date
ES533873A Expired ES8600293A1 (es) 1983-06-30 1984-06-29 Un procedimiento para preparar profarmacos de alopurinol

Country Status (10)

Country Link
US (1) US4694006A (es)
EP (1) EP0148883B1 (es)
JP (1) JPS60501708A (es)
DE (1) DE3481369D1 (es)
DK (1) DK302883D0 (es)
ES (1) ES8600293A1 (es)
FI (1) FI83221C (es)
IE (1) IE57696B1 (es)
IT (1) IT1214854B (es)
WO (1) WO1985000368A1 (es)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4943579A (en) * 1987-10-06 1990-07-24 The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services Water soluble prodrugs of camptothecin
IT1244501B (it) * 1991-03-22 1994-07-15 Sigma Tau Ind Farmaceuti Derivati amminoacilici e oligopeptidici dell'allopurinolo dotati di attivita' immunostimolante e composizioni farmaceutiche che li contengono
US5994361A (en) * 1994-06-22 1999-11-30 Biochem Pharma Substituted purinyl derivatives with immunomodulating activity
US7671029B2 (en) * 1999-08-06 2010-03-02 Immupharma Sa Compositions and methods for enhanced pharmacological activity of compositions comprising peptide drug substances
US20030060413A1 (en) * 2001-09-06 2003-03-27 Zimmer Robert H. Derivatives of pseudo-peptides, their preparation and their biological uses
US6908900B2 (en) * 2001-01-17 2005-06-21 Zimmer & Associates Ag Compositions and methods for enhanced pharmacological activity through oral and parenteral administration of compositions comprising polypeptide drug substances and other poorly absorbed active ingredients
WO2004043396A2 (en) * 2002-11-09 2004-05-27 Nobex Corporation Modified carbamate-containing prodrugs and methods of synthesizing same
WO2010151711A1 (en) 2009-06-25 2010-12-29 Alkermes, Inc. Prodrugs of nh-acidic compounds
WO2011163594A2 (en) * 2010-06-24 2011-12-29 Alkermes, Inc. Prodrugs of nh-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives
CN103561746B (zh) 2011-03-18 2018-05-29 奥克梅斯制药爱尔兰有限公司 包含脱水山梨糖醇酯的药物组合物
NZ722096A (en) 2011-12-15 2016-11-25 Alkermes Pharma Ireland Ltd Prodrugs of secondary amine compounds
EP2827868B8 (en) 2012-03-19 2019-12-18 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising fatty acid esters
CA2867137C (en) 2012-03-19 2020-12-08 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising aripiprazole prodrugs and benzyl alcohol
CA2867123C (en) 2012-03-19 2021-02-16 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising water-insoluble antipsychotic agents and glycerol esters
CA2885196C (en) 2012-09-19 2021-06-22 Alkermes Pharma Ireland Limited Pharmaceutical compositions having improved storage stability
US8883857B2 (en) 2012-12-07 2014-11-11 Baylor College Of Medicine Small molecule xanthine oxidase inhibitors and methods of use
CN110368360A (zh) 2014-03-20 2019-10-25 奥克梅斯制药爱尔兰有限公司 具有增加的注射速度的阿立哌唑制剂
CN105272984B (zh) * 2014-06-23 2019-06-14 湘北威尔曼制药股份有限公司 吡唑并[3,4-d]嘧啶-4-酮衍生物、其制备方法和应用
WO2016015177A1 (zh) * 2014-06-23 2016-02-04 北京新天宇科技开发有限公司 吡唑并[3，4-d]嘧啶-4-酮衍生物、其制备方法和应用
CN112423754A (zh) 2018-03-05 2021-02-26 奥克梅斯制药爱尔兰有限公司 阿立哌唑的给药策略

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2868803A (en) * 1956-02-10 1959-01-13 Ciba Pharm Prod Inc New pyrazoles and method of preparing same
US3474098A (en) * 1968-08-22 1969-10-21 Burroughs Wellcome Co Pyrazolo-(3,4-d) pyrimidines
GB1339748A (en) * 1970-07-02 1973-12-05 Ici Ltd Pyrimidine derivatives
GR75219B (es) * 1980-04-21 1984-07-13 Merck & Co Inc
DE3131365A1 (de) * 1981-08-07 1983-02-24 Henkel KGaA, 4000 Düsseldorf Neue diglycidyl-substituierte heterocyclische verbindungen, verfahren zu ihrer herstellung und ihre verwendung in arzneimittelzubereitungen mit cytostatischer wirksamkeit
US4565868A (en) * 1983-02-07 1986-01-21 Syntex (U.S.A.) Inc. Process for preparing guanine derivatives
US4555579A (en) * 1983-03-24 1985-11-26 E. R. Squibb & Sons, Inc. Dioxolenylmethyl ester prodrugs of phosphinic acid ace inhibitors

Also Published As

Publication number Publication date
WO1985000368A1 (en) 1985-01-31
FI83221B (fi) 1991-02-28
FI850829A0 (fi) 1985-02-28
EP0148883B1 (en) 1990-02-14
DK302883D0 (da) 1983-06-30
IT8467669A0 (it) 1984-06-29
IT1214854B (it) 1990-01-18
US4694006A (en) 1987-09-15
FI850829L (fi) 1985-02-28
IE57696B1 (en) 1993-03-10
IE841659L (en) 1984-12-30
DE3481369D1 (en) 1990-03-22
FI83221C (fi) 1991-06-10
EP0148883A1 (en) 1985-07-24
ES8600293A1 (es) 1985-10-01
JPS60501708A (ja) 1985-10-11

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970519