DK302883D0 - Allopurinol prodrugs - Google Patents

Allopurinol prodrugs

Info

Publication number
DK302883D0
DK302883D0 DK3028/83A DK302883A DK302883D0 DK 302883 D0 DK302883 D0 DK 302883D0 DK 3028/83 A DK3028/83 A DK 3028/83A DK 302883 A DK302883 A DK 302883A DK 302883 D0 DK302883 D0 DK 302883D0
Authority
DK
Denmark
Prior art keywords
allopurinol
products
allopurinol products
Prior art date
Application number
DK3028/83A
Other languages
English (en)
Inventor
Hans Bundgaard
Erik Falch
Original Assignee
Hans Bundgaard
Erik Falch
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hans Bundgaard, Erik Falch filed Critical Hans Bundgaard
Priority to DK3028/83A priority Critical patent/DK302883D0/da
Publication of DK302883D0 publication Critical patent/DK302883D0/da
Priority to DE8484902508T priority patent/DE3481369D1/de
Priority to US06/711,583 priority patent/US4694006A/en
Priority to AT84902508T priority patent/ATE50408T1/de
Priority to EP84902508A priority patent/EP0148883B1/en
Priority to JP84502551A priority patent/JPS60501708A/ja
Priority to PCT/DK1984/000057 priority patent/WO1985000368A1/en
Priority to ES533873A priority patent/ES533873A0/es
Priority to IE1659/84A priority patent/IE57696B1/en
Priority to IT8467669A priority patent/IT1214854B/it
Priority to NO850792A priority patent/NO164028C/no
Priority to DK089685A priority patent/DK162051C/da
Priority to FI850829A priority patent/FI83221C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK3028/83A 1983-06-30 1983-06-30 Allopurinol prodrugs DK302883D0 (da)

Priority Applications (13)

Application Number Priority Date Filing Date Title
DK3028/83A DK302883D0 (da) 1983-06-30 1983-06-30 Allopurinol prodrugs
PCT/DK1984/000057 WO1985000368A1 (en) 1983-06-30 1984-06-19 Allopurinol prodrugs
EP84902508A EP0148883B1 (en) 1983-06-30 1984-06-19 Allopurinol prodrugs
US06/711,583 US4694006A (en) 1983-06-30 1984-06-19 Acyl- or acyloxymethyl-allopurinol prodrugs
AT84902508T ATE50408T1 (de) 1983-06-30 1984-06-19 Allopurinol proheilmittel.
DE8484902508T DE3481369D1 (en) 1983-06-30 1984-06-19 Allopurinol proheilmittel.
JP84502551A JPS60501708A (ja) 1983-06-30 1984-06-19 アロプリノ−ル　プロドラツグ類
ES533873A ES533873A0 (es) 1983-06-30 1984-06-29 Un procedimiento para preparar profarmacos de alopurinol
IE1659/84A IE57696B1 (en) 1983-06-30 1984-06-29 Allopurinol prodrugs
IT8467669A IT1214854B (it) 1983-06-30 1984-06-29 Profarmaci costituiti da composti allopurinolici e procedimento per la loro preparazione
NO850792A NO164028C (no) 1983-06-30 1985-02-27 Analogifremgangsmaate for fremstilling av terapeutisk aktive allopurinol-derivater.
DK089685A DK162051C (da) 1983-06-30 1985-02-27 Allopurinol prodrugs
FI850829A FI83221C (fi) 1983-06-30 1985-02-28 Foerfarande foer framstaellning av som laekemedel anvaendbara 1-, 1,5- eller 2,5-substituerade 1,5- eller 2,5 -dihydro-4h-pyrazol-/3,4-d/-pyrimidin-4-oner.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK3028/83A DK302883D0 (da) 1983-06-30 1983-06-30 Allopurinol prodrugs

Publications (1)

Publication Number Publication Date
DK302883D0 true DK302883D0 (da) 1983-06-30

Family

ID=8118314

Family Applications (1)

Application Number Title Priority Date Filing Date
DK3028/83A DK302883D0 (da) 1983-06-30 1983-06-30 Allopurinol prodrugs

Country Status (10)

Country Link
US (1) US4694006A (da)
EP (1) EP0148883B1 (da)
JP (1) JPS60501708A (da)
DE (1) DE3481369D1 (da)
DK (1) DK302883D0 (da)
ES (1) ES533873A0 (da)
FI (1) FI83221C (da)
IE (1) IE57696B1 (da)
IT (1) IT1214854B (da)
WO (1) WO1985000368A1 (da)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4943579A (en) * 1987-10-06 1990-07-24 The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services Water soluble prodrugs of camptothecin
IT1244501B (it) * 1991-03-22 1994-07-15 Sigma Tau Ind Farmaceuti Derivati amminoacilici e oligopeptidici dell'allopurinolo dotati di attivita' immunostimolante e composizioni farmaceutiche che li contengono
US6110923A (en) * 1994-06-22 2000-08-29 Biochem Pharma Inc. Method for treating cancer using novel substituted purinyl derivatives with immunomodulating activity
US6908900B2 (en) * 2001-01-17 2005-06-21 Zimmer & Associates Ag Compositions and methods for enhanced pharmacological activity through oral and parenteral administration of compositions comprising polypeptide drug substances and other poorly absorbed active ingredients
US7671029B2 (en) * 1999-08-06 2010-03-02 Immupharma Sa Compositions and methods for enhanced pharmacological activity of compositions comprising peptide drug substances
WO2003020321A2 (en) * 2001-09-06 2003-03-13 Zimmer Robert H Derivatives of pseudo-peptides, their preparation and their biological uses
WO2004043396A2 (en) * 2002-11-09 2004-05-27 Nobex Corporation Modified carbamate-containing prodrugs and methods of synthesizing same
US8686009B2 (en) 2009-06-25 2014-04-01 Alkermes Pharma Ireland Limited Prodrugs of NH-acidic compounds
CA2802733C (en) * 2010-06-24 2017-11-21 Alkermes Pharma Ireland Limited Prodrugs of nh-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives
MX358344B (es) 2011-03-18 2018-08-15 Alkermes Pharma Ireland Ltd Composiciones farmaceuticas que comprenden un antipsicotico insoluble en agua y esteres de sorbitan.
WO2013088255A1 (en) 2011-12-15 2013-06-20 Alkermes Pharma Ireland Limited Prodrugs of secondary amine compounds
EP2827868B8 (en) 2012-03-19 2019-12-18 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising fatty acid esters
AU2013235523B9 (en) 2012-03-19 2018-01-04 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising glycerol esters
NZ630428A (en) 2012-03-19 2017-02-24 Alkermes Pharma Ireland Ltd Pharmaceutical compositions comprising benzyl alcohol
WO2014080285A2 (en) 2012-09-19 2014-05-30 Alkermes Pharma Ireland Limited Pharmaceutical compositions having improved storage stability
US8883857B2 (en) * 2012-12-07 2014-11-11 Baylor College Of Medicine Small molecule xanthine oxidase inhibitors and methods of use
CN110368360A (zh) 2014-03-20 2019-10-25 奥克梅斯制药爱尔兰有限公司 具有增加的注射速度的阿立哌唑制剂
CN105272984B (zh) * 2014-06-23 2019-06-14 湘北威尔曼制药股份有限公司 吡唑并[3,4-d]嘧啶-4-酮衍生物、其制备方法和应用
CN106459053B (zh) * 2014-06-23 2019-03-22 湘北威尔曼制药股份有限公司 吡唑并[3,4-d]嘧啶-4-酮衍生物、其制备方法和应用
WO2019173230A1 (en) 2018-03-05 2019-09-12 Alkermes Pharma Ireland Limited Aripiprazole dosing strategy

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2868803A (en) * 1956-02-10 1959-01-13 Ciba Pharm Prod Inc New pyrazoles and method of preparing same
US3474098A (en) * 1968-08-22 1969-10-21 Burroughs Wellcome Co Pyrazolo-(3,4-d) pyrimidines
GB1339748A (en) * 1970-07-02 1973-12-05 Ici Ltd Pyrimidine derivatives
DK172081A (da) * 1980-04-21 1981-10-22 Merck & Co Inc Mercaptoforbindelse og fremgangsmaade til fremstilling deraf
DE3131365A1 (de) * 1981-08-07 1983-02-24 Henkel KGaA, 4000 Düsseldorf Neue diglycidyl-substituierte heterocyclische verbindungen, verfahren zu ihrer herstellung und ihre verwendung in arzneimittelzubereitungen mit cytostatischer wirksamkeit
US4565868A (en) * 1983-02-07 1986-01-21 Syntex (U.S.A.) Inc. Process for preparing guanine derivatives
US4555579A (en) * 1983-03-24 1985-11-26 E. R. Squibb & Sons, Inc. Dioxolenylmethyl ester prodrugs of phosphinic acid ace inhibitors

Also Published As

Publication number Publication date
IE57696B1 (en) 1993-03-10
EP0148883B1 (en) 1990-02-14
IE841659L (en) 1984-12-30
WO1985000368A1 (en) 1985-01-31
ES8600293A1 (es) 1985-10-01
FI83221C (fi) 1991-06-10
DE3481369D1 (en) 1990-03-22
ES533873A0 (es) 1985-10-01
FI83221B (fi) 1991-02-28
IT8467669A0 (it) 1984-06-29
US4694006A (en) 1987-09-15
IT1214854B (it) 1990-01-18
EP0148883A1 (en) 1985-07-24
FI850829A0 (fi) 1985-02-28
JPS60501708A (ja) 1985-10-11
FI850829L (fi) 1985-02-28

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Legal Events

Date Code Title Description
AHS Application shelved for other reasons than non-payment