ES519832A0 - Un procedimiento para preparar pirazolo (4,3-c)piridinas. - Google Patents

Un procedimiento para preparar pirazolo (4,3-c)piridinas.

Info

Publication number
ES519832A0
ES519832A0 ES519832A ES519832A ES519832A0 ES 519832 A0 ES519832 A0 ES 519832A0 ES 519832 A ES519832 A ES 519832A ES 519832 A ES519832 A ES 519832A ES 519832 A0 ES519832 A0 ES 519832A0
Authority
ES
Spain
Prior art keywords
piridines
procedure
preparing pyrazolo
pyrazolo
preparing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES519832A
Other languages
English (en)
Spanish (es)
Other versions
ES8500273A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gruppo Lepetit SpA
Original Assignee
Gruppo Lepetit SpA
Lepetit SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruppo Lepetit SpA, Lepetit SpA filed Critical Gruppo Lepetit SpA
Publication of ES8500273A1 publication Critical patent/ES8500273A1/es
Publication of ES519832A0 publication Critical patent/ES519832A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/74—Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Anesthesiology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ES519832A 1982-02-17 1983-02-16 Un procedimiento para preparar pirazolo (4,3-c)piridinas. Granted ES519832A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8204722 1982-02-17

Publications (2)

Publication Number Publication Date
ES8500273A1 ES8500273A1 (es) 1984-10-01
ES519832A0 true ES519832A0 (es) 1984-10-01

Family

ID=10528419

Family Applications (3)

Application Number Title Priority Date Filing Date
ES519832A Granted ES519832A0 (es) 1982-02-17 1983-02-16 Un procedimiento para preparar pirazolo (4,3-c)piridinas.
ES531981A Expired ES8507547A1 (es) 1982-02-17 1984-04-27 Un procedimiento para preparar pirazolo (4,3-c) piridinas
ES531980A Granted ES531980A0 (es) 1982-02-17 1984-04-27 Un procedimiento para preparar pirazolo (4,3-c) piridinas

Family Applications After (2)

Application Number Title Priority Date Filing Date
ES531981A Expired ES8507547A1 (es) 1982-02-17 1984-04-27 Un procedimiento para preparar pirazolo (4,3-c) piridinas
ES531980A Granted ES531980A0 (es) 1982-02-17 1984-04-27 Un procedimiento para preparar pirazolo (4,3-c) piridinas

Country Status (16)

Country Link
US (1) US4500525A (enExample)
EP (1) EP0086422B1 (enExample)
JP (1) JPS58152885A (enExample)
KR (1) KR900006853B1 (enExample)
AT (1) ATE30027T1 (enExample)
AU (1) AU563591B2 (enExample)
CA (1) CA1225646A (enExample)
DE (1) DE3373904D1 (enExample)
DK (1) DK27383A (enExample)
ES (3) ES519832A0 (enExample)
GR (1) GR78080B (enExample)
IE (1) IE55156B1 (enExample)
IL (1) IL67785A0 (enExample)
NZ (1) NZ203302A (enExample)
PH (1) PH23645A (enExample)
ZA (1) ZA83628B (enExample)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5137890A (en) * 1990-02-14 1992-08-11 Ortho Pharmaceutical Corporation 4-phenyl tetrahydropyrido(4,3-d)pyrimidines
US5264576A (en) * 1992-10-22 1993-11-23 Hoechst-Roussel Pharmaceuticals Incorporated Pyrazolo[4,3-c]pyridines which are intermediates
DE19834044A1 (de) * 1998-07-29 2000-02-03 Bayer Ag Neue substituierte Pyrazolderivate
EP1309593B1 (en) 2000-08-14 2006-03-15 Ortho-McNeil Pharmaceutical, Inc. Substituted pyrazoles
HK1052509B (en) * 2000-08-14 2007-09-07 Ortho-Mcneil Pharmaceutical, Inc. Substituted pyrazole
US7332494B2 (en) 2000-08-14 2008-02-19 Janssen Pharmaceutica, N.V. Method for treating allergies using substituted pyrazoles
US20070117785A1 (en) * 2000-08-14 2007-05-24 Butler Christopher R Substituted pyrazoles and methods of treatment with substituted pyrazoles
JP4911864B2 (ja) * 2000-08-14 2012-04-04 オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド 置換ピラゾール
US20070105841A1 (en) * 2000-08-14 2007-05-10 Breitenbucher J G Method for treating allergies using substituted pyrazoles
US20050101587A9 (en) * 2000-08-14 2005-05-12 Butler Christopher R. Method for treating allergies using substituted pyrazoles
CN1642973A (zh) 2000-09-06 2005-07-20 奥索-麦克尼尔药品公司 治疗变态反应的方法
CN100384420C (zh) * 2000-09-06 2008-04-30 奥索-麦克尼尔药品公司 取代的吡唑在制备用于治疗变应性疾病的药物组合物中的应用
RU2286343C2 (ru) * 2001-08-10 2006-10-27 Орто-Макнейл Фармасьютикал, Инк. Замещенные пиразолы
AU2003231880A1 (en) * 2002-05-30 2003-12-19 Vertex Pharmaceuticals Incorporated Inhibitors of jak and cdk2 protein kinases
EP1526852A1 (en) * 2002-07-25 2005-05-04 Pharmacia Italia S.p.A. Bicyclo-pyrazoles active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
EP2243781A1 (en) * 2003-05-30 2010-10-27 Vertex Pharmaceuticals, Inc. Pyrazolopyridine derivatives as inhibitors of JAK and CDK2 protein kinases
PL1668014T3 (pl) 2003-09-17 2009-06-30 Janssen Pharmaceutica Nv Skondensowane związki heterocykliczne jako modulatory receptora serotoninowego
WO2005030776A1 (en) 2003-09-23 2005-04-07 Vertex Pharmaceuticals Incorporated Pyrazolopyrrole derivatives as protein kinase inhibitors
KR100838692B1 (ko) 2007-07-11 2008-06-16 한국화학연구원 7-(3′,4′-디알콕시페닐)-4,5,6,7-테트라히드로피라졸로[1,5-ａ]피리미딘 화합물, 이의 제조방법 및 이를 포함하는천식 및 만성폐쇄성 폐질환을 포함한 염증관련 질환,관절염, 아토피 피부염, 암 및 뇌질환의 치료 및 예방을위한 약제학적 조성물
US9242981B2 (en) 2010-09-16 2016-01-26 Merck Sharp & Dohme Corp. Fused pyrazole derivatives as novel ERK inhibitors
DK2755972T3 (en) 2011-09-12 2016-01-25 Sanofi Sa INDANYL SUBSTITUTED 4,5,6,7-TETRAHYDRO-1H-PYRAZOLE [4,3-C] PYRIDINES, THEIR USE AS MEDICINE AND PHARMACEUTICAL PREPARATIONS CONTAINING THESE
MX2014002968A (es) 2011-09-12 2014-07-09 Sanofi Sa 4,5,6,7 - tetrahidro - 1h - pirazolo [4,3 -c] piridinas sustituidas con indanilo, su uso como medicamento, y preparaciones farmaceuticas que las comprenden.
EA025240B1 (ru) * 2011-09-16 2016-12-30 Санофи ЗАМЕЩЕННЫЕ 4,5,6,7-ТЕТРАГИДРО-1H-ПИРАЗОЛО[4,3-c]ПИРИДИНЫ, ИХ ПРИМЕНЕНИЕ В КАЧЕСТВЕ ЛЕКАРСТВЕННОГО СРЕДСТВА И ФАРМАЦЕВТИЧЕСКИЕ ПРЕПАРАТЫ, СОДЕРЖАЩИЕ ИХ
DK2755973T3 (en) 2011-09-16 2016-01-25 Sanofi Sa SUBSTITUTED 4,5,6,7-TETRAHYDRO-1H-PYRAZOLE [4,3-C] PYRIDINES, THEIR USE AS MEDICINES AND PHARMACEUTICAL PREPARATIONS CONTAINING THESE
JP6713465B2 (ja) 2014-12-30 2020-06-24 ノヴィラ・セラピューティクス・インコーポレイテッド Ｂ型肝炎感染症治療のための誘導体及び方法
EP3464286B1 (en) * 2016-05-24 2021-08-18 Genentech, Inc. Pyrazolopyridine derivatives for the treatment of cancer
CA3029566A1 (en) 2016-06-29 2018-01-04 Novira Therapeutics, Inc. Diazepinone derivatives and their use in the treatment of hepatitis b infections
WO2018005881A1 (en) 2016-06-29 2018-01-04 Novira Therapeutics, Inc. Oxadiazepinone derivatives and their use in the treatment of hepatitis b infections
MA48803A (fr) 2017-05-31 2020-04-08 Chemocentryx Inc Cycles 6-5 fusionnés utilisés en tant qu'inhibiteurs de c5a
US10828285B2 (en) * 2017-12-22 2020-11-10 Chemocentryx, Inc. Diaryl substituted 6,5-fused ring compounds as C5aR inhibitors

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3852279A (en) * 1973-03-12 1974-12-03 Squibb & Sons Inc 7-substituted -3,3a,4,5,6,7-hexahydro-3-substituted-2h- pyrazolo (4,3-c)pyridines

Also Published As

Publication number Publication date
CA1225646A (en) 1987-08-18
NZ203302A (en) 1986-08-08
AU563591B2 (en) 1987-07-16
PH23645A (en) 1989-09-27
DK27383A (da) 1983-08-18
IL67785A0 (en) 1983-05-15
ZA83628B (en) 1983-12-28
EP0086422A2 (en) 1983-08-24
ES8507546A1 (es) 1985-09-01
DE3373904D1 (en) 1987-11-05
JPS58152885A (ja) 1983-09-10
EP0086422B1 (en) 1987-09-30
EP0086422A3 (en) 1984-03-28
KR840003636A (ko) 1984-09-15
ES531981A0 (es) 1985-09-01
ES8500273A1 (es) 1984-10-01
IE55156B1 (en) 1990-06-20
ES531980A0 (es) 1985-09-01
US4500525A (en) 1985-02-19
ES8507547A1 (es) 1985-09-01
ATE30027T1 (de) 1987-10-15
DK27383D0 (da) 1983-01-25
IE830328L (en) 1983-08-17
GR78080B (enExample) 1984-09-26
KR900006853B1 (ko) 1990-09-22
AU1130583A (en) 1983-08-25
JPH0412269B2 (enExample) 1992-03-04

Similar Documents

Publication Publication Date Title
ES519832A0 (es) Un procedimiento para preparar pirazolo (4,3-c)piridinas.
IL72120A (en) 2-pyrimidinyl-1-piperazine derivatives,their preparation and pharmaceutical compositions containing them
ATE22562T1 (de) 6-substituierte s-triazolo(3,4-a)phthalazinderivate.
DE3571982D1 (en) Benzisoselenazolethiones,process for their preparation and pharmaceutical products containing these compounds
PT77370B (en) Process for preparing new pyrazolo <3,4-b> piridine derivatives and pharmaceutical preparations containing the same
JO1406B1 (en) Chemical compounds
ZA848140B (en) New benzenesulfonyl-lactams,process for their preparation and their use as active substances of pharmaceutical compositions
ES478048A1 (es) Procedimiento para la obtencion de difenil-imidazolil-meta- nos sustituidos.
ATE69228T1 (de) Amidabkoemmlinge.
SE8405588D0 (sv) New compounds
ES8800217A1 (es) Procedimiento para la preparacion de acidos 4-(isoxazolil)-tiazol-2-oxamicos y sus derivados
ES8305783A1 (es) Procedimiento para la obtencion de derivados de aminociclitol saturados.
SE8404334L (sv) 16-fluoro-16,17-didehydro-prostanoider och forfarande for deras framstellning
ES8200871A1 (es) Procedimiento para la obtencion de derivados de 2-amino-3,4-dihidropiridina
ES2000716A6 (es) Un procedimiento para preparar derivados de tetrahidroisoquinoleina
ATE44149T1 (de) N,n-dialkylaminoalkyl-hexahydro-5-oxo-1hpyrrolizin-3-carboxamide.

Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970303