ES457473A1 - Un procedimiento para preparar derivados de cefalosporina. - Google Patents
Un procedimiento para preparar derivados de cefalosporina.Info
- Publication number
- ES457473A1 ES457473A1 ES457473A ES457473A ES457473A1 ES 457473 A1 ES457473 A1 ES 457473A1 ES 457473 A ES457473 A ES 457473A ES 457473 A ES457473 A ES 457473A ES 457473 A1 ES457473 A1 ES 457473A1
- Authority
- ES
- Spain
- Prior art keywords
- proteus
- formula
- group
- carbamoyloxy
- acyloxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 229930186147 Cephalosporin Natural products 0.000 title abstract 2
- 229940124587 cephalosporin Drugs 0.000 title abstract 2
- 150000001780 cephalosporins Chemical class 0.000 title abstract 2
- 241000894006 Bacteria Species 0.000 abstract 2
- 241000588919 Citrobacter freundii Species 0.000 abstract 1
- 241000588724 Escherichia coli Species 0.000 abstract 1
- 241000588747 Klebsiella pneumoniae Species 0.000 abstract 1
- 241000588772 Morganella morganii Species 0.000 abstract 1
- 241000588770 Proteus mirabilis Species 0.000 abstract 1
- 241000588767 Proteus vulgaris Species 0.000 abstract 1
- 241000588777 Providencia rettgeri Species 0.000 abstract 1
- 125000004423 acyloxy group Chemical group 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 230000003115 biocidal effect Effects 0.000 abstract 1
- -1 carbamoyloxy Chemical group 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
- 229940007042 proteus vulgaris Drugs 0.000 abstract 1
- 125000001453 quaternary ammonium group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP51037374A JPS5946237B2 (ja) | 1976-04-02 | 1976-04-02 | セフアロスポリン誘導体およびその製造法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES457473A1 true ES457473A1 (es) | 1978-07-01 |
Family
ID=12495730
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES457473A Expired ES457473A1 (es) | 1976-04-02 | 1977-04-01 | Un procedimiento para preparar derivados de cefalosporina. |
Country Status (22)
| Country | Link |
|---|---|
| US (2) | US4172891A (OSRAM) |
| JP (1) | JPS5946237B2 (OSRAM) |
| AT (1) | AT351677B (OSRAM) |
| AU (1) | AU510278B2 (OSRAM) |
| BE (1) | BE853073A (OSRAM) |
| CA (1) | CA1127149A (OSRAM) |
| CH (1) | CH631717A5 (OSRAM) |
| DE (1) | DE2714419C2 (OSRAM) |
| DK (1) | DK144577A (OSRAM) |
| ES (1) | ES457473A1 (OSRAM) |
| FI (1) | FI66006C (OSRAM) |
| FR (2) | FR2361403A1 (OSRAM) |
| GB (1) | GB1525687A (OSRAM) |
| GR (1) | GR66409B (OSRAM) |
| HU (1) | HU179596B (OSRAM) |
| MX (1) | MX4409E (OSRAM) |
| NL (1) | NL7703474A (OSRAM) |
| NO (1) | NO153259C (OSRAM) |
| PH (1) | PH13024A (OSRAM) |
| PT (1) | PT66392B (OSRAM) |
| SE (1) | SE433354B (OSRAM) |
| ZA (1) | ZA771993B (OSRAM) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5946237B2 (ja) * | 1976-04-02 | 1984-11-10 | 武田薬品工業株式会社 | セフアロスポリン誘導体およびその製造法 |
| IL61458A0 (en) * | 1979-12-07 | 1980-12-31 | Erba Farmitalia | N-substituted thiazolyl derivatives of oximino-substituted cephalosporins, their preparation and pharmalceutical compositions containing them |
| IT1148888B (it) * | 1980-07-15 | 1986-12-03 | Schiena Ricerche Di | Composti antibiotici |
| NZ198350A (en) * | 1980-09-25 | 1985-02-28 | Toyama Chemical Co Ltd | Cephalosporins and intermediates;pharmaceutical compositions |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2518130A (en) * | 1945-04-26 | 1950-08-08 | Evans | N-oxides of tertiary amines and process of preparing same |
| US2500131A (en) * | 1945-06-27 | 1950-03-07 | Ralph L Evans | Di-nu-oxides of amino-substituted acridines and quinolines |
| NZ176206A (en) * | 1973-12-25 | 1978-03-06 | Takeda Chemical Industries Ltd | Cephalosporins |
| JPS5119765A (en) * | 1974-08-09 | 1976-02-17 | Takeda Chemical Industries Ltd | Aminochiazoorujudotaino seizoho |
| DK154939C (da) * | 1974-12-19 | 1989-06-12 | Takeda Chemical Industries Ltd | Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf |
| JPS5946237B2 (ja) * | 1976-04-02 | 1984-11-10 | 武田薬品工業株式会社 | セフアロスポリン誘導体およびその製造法 |
-
1976
- 1976-04-02 JP JP51037374A patent/JPS5946237B2/ja not_active Expired
-
1977
- 1977-03-25 MX MX775580U patent/MX4409E/es unknown
- 1977-03-26 GR GR53093A patent/GR66409B/el unknown
- 1977-03-29 NO NO771111A patent/NO153259C/no unknown
- 1977-03-29 AU AU23723/77A patent/AU510278B2/en not_active Expired
- 1977-03-30 NL NL7703474A patent/NL7703474A/xx not_active Application Discontinuation
- 1977-03-30 SE SE7703689A patent/SE433354B/xx not_active IP Right Cessation
- 1977-03-30 CH CH397277A patent/CH631717A5/de not_active IP Right Cessation
- 1977-03-31 FR FR7709744A patent/FR2361403A1/fr active Granted
- 1977-03-31 DE DE2714419A patent/DE2714419C2/de not_active Expired
- 1977-03-31 BE BE1008055A patent/BE853073A/xx not_active IP Right Cessation
- 1977-03-31 GB GB13688/77A patent/GB1525687A/en not_active Expired
- 1977-03-31 US US05/783,230 patent/US4172891A/en not_active Expired - Lifetime
- 1977-04-01 HU HU77TA1433A patent/HU179596B/hu not_active IP Right Cessation
- 1977-04-01 ZA ZA00771993A patent/ZA771993B/xx unknown
- 1977-04-01 FI FI771023A patent/FI66006C/fi not_active IP Right Cessation
- 1977-04-01 ES ES457473A patent/ES457473A1/es not_active Expired
- 1977-04-01 PH PH19619A patent/PH13024A/en unknown
- 1977-04-01 DK DK144577A patent/DK144577A/da not_active Application Discontinuation
- 1977-04-01 CA CA275,315A patent/CA1127149A/en not_active Expired
- 1977-04-02 PT PT66392A patent/PT66392B/pt unknown
- 1977-04-04 AT AT234677A patent/AT351677B/de active
-
1978
- 1978-01-10 FR FR7800580A patent/FR2369282A1/fr active Granted
-
1979
- 1979-05-31 US US06/044,215 patent/US4239758A/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| MX4409E (es) | 1982-04-27 |
| NO153259B (no) | 1985-11-04 |
| PT66392B (en) | 1978-09-11 |
| BE853073A (fr) | 1977-09-30 |
| FI66006B (fi) | 1984-04-30 |
| FR2361403B1 (OSRAM) | 1981-11-13 |
| DE2714419C2 (de) | 1985-12-05 |
| AU510278B2 (en) | 1980-06-19 |
| CA1127149A (en) | 1982-07-06 |
| AT351677B (de) | 1979-08-10 |
| US4239758A (en) | 1980-12-16 |
| FR2369282A1 (fr) | 1978-05-26 |
| FI66006C (fi) | 1984-08-10 |
| ATA234677A (de) | 1979-01-15 |
| DK144577A (da) | 1977-10-03 |
| HU179596B (en) | 1982-11-29 |
| JPS52122389A (en) | 1977-10-14 |
| FR2361403A1 (fr) | 1978-03-10 |
| GR66409B (OSRAM) | 1981-03-20 |
| US4172891A (en) | 1979-10-30 |
| NL7703474A (nl) | 1977-10-04 |
| PT66392A (en) | 1977-05-01 |
| FI771023A7 (OSRAM) | 1977-10-03 |
| PH13024A (en) | 1979-11-15 |
| DE2714419A1 (de) | 1977-10-13 |
| FR2369282B1 (OSRAM) | 1981-05-08 |
| AU2372377A (en) | 1978-10-05 |
| SE7703689L (sv) | 1977-10-03 |
| GB1525687A (en) | 1978-09-20 |
| JPS5946237B2 (ja) | 1984-11-10 |
| CH631717A5 (de) | 1982-08-31 |
| ZA771993B (en) | 1978-03-29 |
| NO153259C (no) | 1986-02-12 |
| SE433354B (sv) | 1984-05-21 |
| NO771111L (no) | 1977-10-04 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19971103 |