ES401590A1 - Procedimiento para la preparacion de nuevas pirido (3,2-d) pirimidinas. - Google Patents

Procedimiento para la preparacion de nuevas pirido (3,2-d) pirimidinas.

Info

Publication number
ES401590A1
ES401590A1 ES401590A ES401590A ES401590A1 ES 401590 A1 ES401590 A1 ES 401590A1 ES 401590 A ES401590 A ES 401590A ES 401590 A ES401590 A ES 401590A ES 401590 A1 ES401590 A1 ES 401590A1
Authority
ES
Spain
Prior art keywords
general formula
radicals
radical
compound
salts
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES401590A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
Original Assignee
Dr Karl Thomae GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19712117657 external-priority patent/DE2117657B2/de
Priority claimed from DE19722208535 external-priority patent/DE2208535A1/de
Priority claimed from DE19722208534 external-priority patent/DE2208534A1/de
Application filed by Dr Karl Thomae GmbH filed Critical Dr Karl Thomae GmbH
Publication of ES401590A1 publication Critical patent/ES401590A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES401590A 1971-04-10 1972-04-08 Procedimiento para la preparacion de nuevas pirido (3,2-d) pirimidinas. Expired ES401590A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19712117657 DE2117657B2 (de) 1971-04-10 1971-04-10 Pyrido eckige klammer auf 3,2- d eckige klammer zu pyrimidine
DE19722208535 DE2208535A1 (de) 1972-02-23 1972-02-23 Neue pyrido eckige klammer auf 3,2-d eckige klammer zu pyrimidine
DE19722208534 DE2208534A1 (de) 1972-02-23 1972-02-23 Neue pyrido eckige klammer auf 3,2-d eckige klammer zu pyrimidin

Publications (1)

Publication Number Publication Date
ES401590A1 true ES401590A1 (es) 1975-02-16

Family

ID=27183344

Family Applications (2)

Application Number Title Priority Date Filing Date
ES401590A Expired ES401590A1 (es) 1971-04-10 1972-04-08 Procedimiento para la preparacion de nuevas pirido (3,2-d) pirimidinas.
ES405213A Expired ES405213A1 (es) 1971-04-10 1972-07-27 Procedimiento para la preparacion de nuevas pirido(3,2-d) pirimidinas.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES405213A Expired ES405213A1 (es) 1971-04-10 1972-07-27 Procedimiento para la preparacion de nuevas pirido(3,2-d) pirimidinas.

Country Status (7)

Country Link
US (1) US3843638A (es)
AT (1) AT319252B (es)
BG (1) BG19597A3 (es)
ES (2) ES401590A1 (es)
PL (1) PL84565B1 (es)
RO (1) RO63031A (es)
SU (2) SU474984A3 (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH075594B2 (ja) * 1986-03-25 1995-01-25 三井石油化学工業株式会社 新規ピリドピリミジン誘導体
ATE496035T1 (de) * 1998-03-31 2011-02-15 Kyowa Hakko Kirin Co Ltd Stickstoffenthaltende heterocyclische verbindungen
WO2004052862A1 (ja) * 2002-12-10 2004-06-24 Ono Pharmaceutical Co., Ltd. 含窒素複素環化合物およびその医薬用途
JP2008543888A (ja) * 2005-06-24 2008-12-04 ギリアード サイエンシーズ, インコーポレイテッド ピリド(3,2−d)ピリミジン、およびC型肝炎を治療するのに有用な医薬組成物
US8338435B2 (en) * 2006-07-20 2012-12-25 Gilead Sciences, Inc. Substituted pyrido(3,2-D) pyrimidines and pharmaceutical compositions for treating viral infections
TW200840584A (en) * 2006-12-26 2008-10-16 Gilead Sciences Inc Pyrido(3,2-d)pyrimidines useful for treating viral infections
BR112012019635A2 (pt) 2010-02-22 2016-05-03 Hoffmann La Roche compostos inibidores de pirido[3,2-d] pirimidina pi3k delta e métodos de uso
CN111171020A (zh) * 2018-11-13 2020-05-19 上海轶诺药业有限公司 一类六元并六元杂环化合物及其作为蛋白受体激酶抑制剂的用途

Also Published As

Publication number Publication date
BG19597A3 (es) 1975-06-25
SU474984A3 (ru) 1975-06-25
SU515450A3 (ru) 1976-05-25
AT319252B (de) 1974-12-10
ES405213A1 (es) 1976-01-01
PL84565B1 (es) 1976-04-30
RO63031A (fr) 1978-05-15
US3843638A (en) 1974-10-22

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