ES2732437T3 - Moduladores del receptor de CXCR7 - Google Patents
Moduladores del receptor de CXCR7 Download PDFInfo
- Publication number
- ES2732437T3 ES2732437T3 ES15801467T ES15801467T ES2732437T3 ES 2732437 T3 ES2732437 T3 ES 2732437T3 ES 15801467 T ES15801467 T ES 15801467T ES 15801467 T ES15801467 T ES 15801467T ES 2732437 T3 ES2732437 T3 ES 2732437T3
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- Prior art keywords
- lam
- benzo
- ethyl
- tetrahydro
- alkyl
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
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- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
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- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP2014076126 | 2014-12-01 | ||
| PCT/EP2015/078058 WO2016087370A1 (en) | 2014-12-01 | 2015-11-30 | Cxcr7 receptor modulators |
Publications (1)
| Publication Number | Publication Date |
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| ES2732437T3 true ES2732437T3 (es) | 2019-11-22 |
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| JP (1) | JP6582056B2 (https=) |
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| ES (1) | ES2732437T3 (https=) |
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| EA028604B1 (ru) | 2013-05-30 | 2017-12-29 | Идорсиа Фармасьютиклз Лтд. | Модуляторы рецептора cxcr7 |
| HRP20230313T1 (hr) * | 2016-07-28 | 2023-05-12 | Idorsia Pharmaceuticals Ltd | Modulatori receptora cxcr7 piperidina |
| CN112266368B (zh) * | 2017-11-15 | 2024-03-19 | 中山光禾医疗科技有限公司 | 光交联水凝胶材料的制备、原料、产品及应用 |
| KR102502046B1 (ko) * | 2018-01-26 | 2023-02-20 | 이도르시아 파마슈티컬스 리미티드 | Cxcr7 수용체 작동제 (3s,4s)-1-시클로프로필메틸-4-｛[5-(2,4-디플루오로-페닐)-이속사졸-3-카르보닐]-아미노｝-피페리딘-3-카르복실산 (1-피리미딘-2-일-시클로프로필)-아미드의 결정질 형태 |
| WO2020207263A1 (zh) * | 2019-04-08 | 2020-10-15 | 四川科伦博泰生物医药股份有限公司 | 苯并咪唑化合物、其制备方法及其用途 |
| MX2023012365A (es) * | 2021-04-19 | 2023-11-27 | Chemocentryx Inc | Azetidinil-acetamidas como inhibidores de cxcr7. |
| CN120202196A (zh) | 2022-11-16 | 2025-06-24 | 巴斯夫欧洲公司 | 作为杀真菌剂的取代的苯并二氮杂䓬类 |
| WO2024104822A1 (en) | 2022-11-16 | 2024-05-23 | Basf Se | Substituted tetrahydrobenzodiazepine as fungicides |
| CN120202195A (zh) | 2022-11-16 | 2025-06-24 | 巴斯夫欧洲公司 | 作为杀真菌剂的取代的苯并二氮杂䓬类 |
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| US5639748A (en) * | 1991-08-05 | 1997-06-17 | Smithkline Beecham Corporation | 6,9-disubstituted benzazepines having α-adrenoceptor blocking activity |
| GB9116824D0 (en) * | 1991-08-05 | 1991-09-18 | Smithkline Beecham Corp | Chemical compounds |
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| WO2002046164A1 (en) | 2000-12-07 | 2002-06-13 | Astrazeneca Ab | Therapeutic compounds |
| JP2002371042A (ja) * | 2001-06-12 | 2002-12-26 | Takeda Chem Ind Ltd | ジアミン化合物、その製造法および用途 |
| ATE427933T1 (de) * | 2002-12-20 | 2009-04-15 | Chemocentryx Inc | Inhibitoren der bindungder chemokine i-tac bzw. sdf-1 an den ccxckr2-rezeptor |
| EP1575874B1 (en) | 2002-12-23 | 2010-09-08 | Council of Scientific and Industrial Research | Process for preparing hydrotalcite and brucite type posite charged layers |
| US20050192272A1 (en) * | 2003-12-22 | 2005-09-01 | Garland Marshall | Substituted benzodiazepines as inhibitors of the chemokine receptor CXCR4 |
| DE602006018057D1 (de) | 2005-11-10 | 2010-12-16 | Chemocentryx Inc | Substituierte chinolone und verwendungsverfahren |
| EP2069347A2 (en) | 2006-09-27 | 2009-06-17 | Merck & Co., Inc. | Novel inhibitors of beta-lactamase |
| CN101535276B (zh) * | 2006-10-23 | 2013-08-28 | 赛福伦公司 | 作为ALK和c-MET抑制剂的2,4-二氨基嘧啶稠合双环衍生物 |
| US20100331298A1 (en) | 2007-12-10 | 2010-12-30 | Cytopathfinder, Inc. | Carboxamide Compounds and Their Use |
| PE20091339A1 (es) * | 2007-12-21 | 2009-09-26 | Glaxo Group Ltd | Derivados de oxadiazol con actividad sobre receptores s1p1 |
| US8748623B2 (en) * | 2009-02-17 | 2014-06-10 | Syntrix Biosystems, Inc. | Pyridinecarboxamides as CXCR2 modulators |
| AR091516A1 (es) | 2012-06-22 | 2015-02-11 | Actelion Pharmaceuticals Ltd | Derivados de 1-[m-carboxamido(hetero)aril-metil]-heterociclil-carboxamida |
| EA028604B1 (ru) | 2013-05-30 | 2017-12-29 | Идорсиа Фармасьютиклз Лтд. | Модуляторы рецептора cxcr7 |
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| US20170327493A1 (en) | 2017-11-16 |
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| EP3227263A1 (en) | 2017-10-11 |
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