ES2693520T3 - Quinazolinas sustituidas con sulfoximina para composiciones farmacéuticas - Google Patents
Quinazolinas sustituidas con sulfoximina para composiciones farmacéuticas Download PDFInfo
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- ES2693520T3 ES2693520T3 ES14808895.8T ES14808895T ES2693520T3 ES 2693520 T3 ES2693520 T3 ES 2693520T3 ES 14808895 T ES14808895 T ES 14808895T ES 2693520 T3 ES2693520 T3 ES 2693520T3
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
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- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
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Landscapes
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| EP13195720 | 2013-12-04 | ||
| PCT/EP2014/075890 WO2015082324A1 (en) | 2013-12-04 | 2014-11-28 | Sulfoximine substituted quinazolines for pharmaceutical compositions |
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| UY38540A (es) * | 2019-01-14 | 2020-08-31 | Pi Industries Ltd | Compuestos de fenilamidina 3-sustituida, preparación y uso |
| CN112812136B (zh) * | 2019-11-15 | 2022-04-12 | 武汉光谷亚太医药研究院有限公司 | 新型2,3-二氢化茚衍生化合物、制备方法和应用 |
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| SE0102147D0 (sv) | 2001-06-18 | 2001-06-18 | Pharmacia Ab | New methods |
| DK1439863T3 (da) | 2001-10-29 | 2011-03-14 | Boehringer Ingelheim Int | MNK-kinase-homologe proteiner, som er involveret i reguleringen af energihomeostase og organelmetabolisme |
| AU2003206068A1 (en) | 2002-03-01 | 2003-09-16 | Pfizer Inc. | Indolyl-urea derivatives of thienopyridines useful as anti-angiogenic agents |
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| CA2558647C (en) | 2004-04-08 | 2013-05-28 | Dow Agrosciences Llc | Insecticidal n-substituted sulfoximines |
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| JP2010527951A (ja) | 2007-05-24 | 2010-08-19 | バイエル・シエーリング・ファーマ アクチエンゲゼルシャフト | キナーゼ阻害剤としての新規なスルホキシイミン置換型キノリン及びキナゾリン誘導体 |
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| UY33241A (es) * | 2010-02-26 | 2011-09-30 | Boehringer Ingelheim Int | ?Tienopirimidinas que contienen heterocicloalquilo para composiciones farmacéuticas?. |
| US8853193B2 (en) | 2010-02-26 | 2014-10-07 | Boehringer Ingelheim International Gmbh | Thienopyrimidines containing a substituted alkyl group for pharmaceutical compositions |
| AR088082A1 (es) | 2011-10-13 | 2014-05-07 | Lilly Co Eli | Moduladores selectivos del receptor androgeno |
| WO2014072244A1 (en) | 2012-11-09 | 2014-05-15 | Boehringer Ingelheim International Gmbh | Sulfoximine substituted quinazolines for pharmaceutical compositions |
| ES2663788T3 (es) * | 2013-06-28 | 2018-04-17 | Evotec International Gmbh | Quinazolinas sustituidas con sulfoximina y su uso como inhibidores de MNK1 y/o MNK2 quinasas |
-
2014
- 2014-11-28 EP EP14808895.8A patent/EP3077383B1/en active Active
- 2014-11-28 AU AU2014359456A patent/AU2014359456B2/en not_active Ceased
- 2014-11-28 JP JP2016536528A patent/JP6457523B2/ja not_active Expired - Fee Related
- 2014-11-28 CA CA2929742A patent/CA2929742C/en active Active
- 2014-11-28 WO PCT/EP2014/075890 patent/WO2015082324A1/en not_active Ceased
- 2014-11-28 ES ES14808895.8T patent/ES2693520T3/es active Active
- 2014-11-28 US US15/101,620 patent/US10093660B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| JP2016539148A (ja) | 2016-12-15 |
| JP6457523B2 (ja) | 2019-01-23 |
| CA2929742A1 (en) | 2015-06-11 |
| AU2014359456B2 (en) | 2019-01-24 |
| CA2929742C (en) | 2022-09-20 |
| US10093660B2 (en) | 2018-10-09 |
| EP3077383A1 (en) | 2016-10-12 |
| US20170174668A1 (en) | 2017-06-22 |
| WO2015082324A1 (en) | 2015-06-11 |
| AU2014359456A1 (en) | 2016-06-09 |
| EP3077383B1 (en) | 2018-08-22 |
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