CA2929742C - Sulfoximine substituted quinazolines for pharmaceutical compositions - Google Patents
Sulfoximine substituted quinazolines for pharmaceutical compositions Download PDFInfo
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- CA2929742C CA2929742C CA2929742A CA2929742A CA2929742C CA 2929742 C CA2929742 C CA 2929742C CA 2929742 A CA2929742 A CA 2929742A CA 2929742 A CA2929742 A CA 2929742A CA 2929742 C CA2929742 C CA 2929742C
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- 101710138999 MAP kinase-interacting serine/threonine-protein kinase 2 Proteins 0.000 claims abstract description 38
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- 101710139011 MAP kinase-interacting serine/threonine-protein kinase 1 Proteins 0.000 claims abstract 3
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Landscapes
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- Hematology (AREA)
- Obesity (AREA)
- Epidemiology (AREA)
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- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Hospice & Palliative Care (AREA)
- Emergency Medicine (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Urology & Nephrology (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP13195720.1 | 2013-12-04 | ||
| EP13195720 | 2013-12-04 | ||
| PCT/EP2014/075890 WO2015082324A1 (en) | 2013-12-04 | 2014-11-28 | Sulfoximine substituted quinazolines for pharmaceutical compositions |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CA2929742A1 CA2929742A1 (en) | 2015-06-11 |
| CA2929742C true CA2929742C (en) | 2022-09-20 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2929742A Active CA2929742C (en) | 2013-12-04 | 2014-11-28 | Sulfoximine substituted quinazolines for pharmaceutical compositions |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US10093660B2 (cg-RX-API-DMAC7.html) |
| EP (1) | EP3077383B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP6457523B2 (cg-RX-API-DMAC7.html) |
| AU (1) | AU2014359456B2 (cg-RX-API-DMAC7.html) |
| CA (1) | CA2929742C (cg-RX-API-DMAC7.html) |
| ES (1) | ES2693520T3 (cg-RX-API-DMAC7.html) |
| WO (1) | WO2015082324A1 (cg-RX-API-DMAC7.html) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3140300B1 (en) * | 2014-05-07 | 2019-08-14 | Evotec International GmbH | Sulfoximine substituted quinazolines for pharmaceutical compositions |
| UY38540A (es) * | 2019-01-14 | 2020-08-31 | Pi Industries Ltd | Compuestos de fenilamidina 3-sustituida, preparación y uso |
| CN112812136B (zh) * | 2019-11-15 | 2022-04-12 | 武汉光谷亚太医药研究院有限公司 | 新型2,3-二氢化茚衍生化合物、制备方法和应用 |
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| US3987192A (en) | 1974-01-07 | 1976-10-19 | The Upjohn Company | Compositions and process of treatment |
| US5602118A (en) | 1993-03-16 | 1997-02-11 | American Cyanamid Company | 2-thiosubstituted carbapenems |
| EP0765324A1 (en) | 1994-06-08 | 1997-04-02 | E.I. Du Pont De Nemours And Company | Cyclic sulfonamide herbicides |
| SE0102147D0 (sv) | 2001-06-18 | 2001-06-18 | Pharmacia Ab | New methods |
| DK1439863T3 (da) | 2001-10-29 | 2011-03-14 | Boehringer Ingelheim Int | MNK-kinase-homologe proteiner, som er involveret i reguleringen af energihomeostase og organelmetabolisme |
| AU2003206068A1 (en) | 2002-03-01 | 2003-09-16 | Pfizer Inc. | Indolyl-urea derivatives of thienopyridines useful as anti-angiogenic agents |
| GB0315587D0 (en) | 2003-07-03 | 2003-08-13 | Univ Dundee | Anti-inflammatory assay and compounds |
| CA2558647C (en) | 2004-04-08 | 2013-05-28 | Dow Agrosciences Llc | Insecticidal n-substituted sulfoximines |
| EP1746099A1 (en) | 2004-12-23 | 2007-01-24 | DeveloGen Aktiengesellschaft | Mnk1 or Mnk2 inhibitors |
| JP5301986B2 (ja) * | 2005-06-22 | 2013-09-25 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 医薬組成物用のチエノピリミジン類 |
| AU2007222982A1 (en) | 2006-03-09 | 2007-09-13 | Pharmacopeia, Inc. | 8-Heteroarylpurine Mnk2 inhibitors for treating metabolic disorders |
| CA2651898A1 (en) * | 2006-04-07 | 2007-10-18 | Develogen Aktiengesellschaft | Thienopyrimidines having mnk1/mnk2 inhibiting activity for pharmaceutical compositions |
| EP2044051B1 (en) | 2006-06-22 | 2010-01-27 | BIOVITRUM AB (publ) | Pyridine and pyrazine derivatives as mnk kinase inhibitors |
| JP2010527951A (ja) | 2007-05-24 | 2010-08-19 | バイエル・シエーリング・ファーマ アクチエンゲゼルシャフト | キナーゼ阻害剤としての新規なスルホキシイミン置換型キノリン及びキナゾリン誘導体 |
| DE102007024470A1 (de) | 2007-05-24 | 2008-11-27 | Bayer Schering Pharma Aktiengesellschaft | Neue Sulfoximin-substituierte Chinolin- bzw. Chinazolinderivate als Kinase-Inhibitoren |
| CN101925588B (zh) | 2008-01-25 | 2014-01-15 | 先正达参股股份有限公司 | 用作杀虫剂的2-氰基苯基磺酰胺衍生物 |
| WO2011062885A1 (en) | 2009-11-23 | 2011-05-26 | Schering Corporation | Fused bicyclic pyrimidine derivatives and methods of use thereof |
| UY33241A (es) * | 2010-02-26 | 2011-09-30 | Boehringer Ingelheim Int | ?Tienopirimidinas que contienen heterocicloalquilo para composiciones farmacéuticas?. |
| US8853193B2 (en) | 2010-02-26 | 2014-10-07 | Boehringer Ingelheim International Gmbh | Thienopyrimidines containing a substituted alkyl group for pharmaceutical compositions |
| AR088082A1 (es) | 2011-10-13 | 2014-05-07 | Lilly Co Eli | Moduladores selectivos del receptor androgeno |
| WO2014072244A1 (en) | 2012-11-09 | 2014-05-15 | Boehringer Ingelheim International Gmbh | Sulfoximine substituted quinazolines for pharmaceutical compositions |
| ES2663788T3 (es) * | 2013-06-28 | 2018-04-17 | Evotec International Gmbh | Quinazolinas sustituidas con sulfoximina y su uso como inhibidores de MNK1 y/o MNK2 quinasas |
-
2014
- 2014-11-28 EP EP14808895.8A patent/EP3077383B1/en active Active
- 2014-11-28 AU AU2014359456A patent/AU2014359456B2/en not_active Ceased
- 2014-11-28 JP JP2016536528A patent/JP6457523B2/ja not_active Expired - Fee Related
- 2014-11-28 CA CA2929742A patent/CA2929742C/en active Active
- 2014-11-28 WO PCT/EP2014/075890 patent/WO2015082324A1/en not_active Ceased
- 2014-11-28 ES ES14808895.8T patent/ES2693520T3/es active Active
- 2014-11-28 US US15/101,620 patent/US10093660B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| JP2016539148A (ja) | 2016-12-15 |
| JP6457523B2 (ja) | 2019-01-23 |
| CA2929742A1 (en) | 2015-06-11 |
| AU2014359456B2 (en) | 2019-01-24 |
| US10093660B2 (en) | 2018-10-09 |
| EP3077383A1 (en) | 2016-10-12 |
| ES2693520T3 (es) | 2018-12-12 |
| US20170174668A1 (en) | 2017-06-22 |
| WO2015082324A1 (en) | 2015-06-11 |
| AU2014359456A1 (en) | 2016-06-09 |
| EP3077383B1 (en) | 2018-08-22 |
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