ES2620373T3 - Partículas que contienen un antagonista del receptor de opioides periférico - Google Patents
Partículas que contienen un antagonista del receptor de opioides periférico Download PDFInfo
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- ES2620373T3 ES2620373T3 ES09774028.6T ES09774028T ES2620373T3 ES 2620373 T3 ES2620373 T3 ES 2620373T3 ES 09774028 T ES09774028 T ES 09774028T ES 2620373 T3 ES2620373 T3 ES 2620373T3
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- opioid receptor
- receptor antagonist
- particles
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Classifications
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- A—HUMAN NECESSITIES
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
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- A—HUMAN NECESSITIES
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- A61K9/51—Nanocapsules; Nanoparticles
- A61K9/5107—Excipients; Inactive ingredients
- A61K9/513—Organic macromolecular compounds; Dendrimers
- A61K9/5138—Organic macromolecular compounds; Dendrimers obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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- A—HUMAN NECESSITIES
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| PCT/US2009/047372 WO2010002576A1 (en) | 2008-07-01 | 2009-06-15 | Particles containing an opioid receptor antagonist and methods of use |
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| WO2014007972A2 (en) | 2012-06-15 | 2014-01-09 | Nova Southeastern University | Epinephrine nanoparticles, methods of fabrication thereof, and methods for use thereof for treatment of conditions responsive to epinphrine |
| US20160045457A1 (en) | 2005-09-09 | 2016-02-18 | Ousama Rachid | Epinephrine fine particles and methods for use thereof for treatment of conditions responsive to epinephrine |
| US8829020B2 (en) | 2009-07-16 | 2014-09-09 | Mallinckrodt Llc | Compounds and compositions for use in phototherapy and in treatment of ocular neovascular disease and cancers |
| CA2853084C (en) | 2011-10-21 | 2022-04-26 | Nova Southeastern University | Epinephrine nanoparticles, methods of fabrication thereof, and methods for use thereof for treatment of conditions responsive to epinephrine |
| EP3326585B1 (en) | 2012-01-31 | 2019-06-19 | Mitral Valve Technologies Sàrl | Mitral valve docking devices and systems |
| CA2872400A1 (en) * | 2012-05-04 | 2013-11-07 | University Of Chicago | Bioavailability of oral methylnaltrexone increases with a phosphatidylcholine-based formulation |
| US10485798B2 (en) | 2012-08-22 | 2019-11-26 | Aptapharma Inc. | Methylnaltrexone nasal formulations, methods of making, and use thereof |
| ES2882530T3 (es) | 2013-03-22 | 2021-12-02 | Univ Nova Southeastern | Partículas finas de epinefrina y métodos para uso de las mismas para el tratamiento de condiciones que responden a la epinefrina |
| CN104274414B (zh) * | 2013-07-02 | 2018-03-09 | 天津康鸿医药科技发展有限公司 | 一种甲基纳曲酮复合物、口服片剂及其制备方法 |
| WO2016004290A1 (en) * | 2014-07-03 | 2016-01-07 | Bind Therapeutics, Inc. | Targeted therapeutic nanoparticles and methods of making and using same |
| JP2021512924A (ja) * | 2018-02-08 | 2021-05-20 | タイワンジェ ファーマシューティカルズ カンパニー リミテッドＴａｉｗａｎｊ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｃｏ．， Ｌｔｄ． | オピオイド受容体拮抗薬の固体剤形の医薬製剤 |
| WO2019169108A1 (en) * | 2018-02-28 | 2019-09-06 | Celista Pharmaceuticals Llc | Oxycodone and methylnaltrexone multi-particulates and suspensions containing them |
| WO2020081952A1 (en) | 2018-10-19 | 2020-04-23 | Nova Southeastern University | Sublingual epinephrine compositions including ph-modifying excipients and penetration enhancers and methods for use thereof |
| WO2021222545A1 (en) * | 2020-04-29 | 2021-11-04 | The Texas A&M University System | Naloxone nanoparticle compositions and methods thereof |
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| ES2114502B1 (es) * | 1996-07-29 | 1999-07-01 | Univ Santiago Compostela | Aplicacion de nanoparticulas a base de polimeros hidrofilicos como formas farmaceuticas. |
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| DE19651551C2 (de) * | 1996-12-11 | 2000-02-03 | Klinge Co Chem Pharm Fab | Opioidantagonisthaltige galenische Formulierung |
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| EP1404323B1 (en) | 2001-06-05 | 2009-10-28 | The University of Chicago | Use of methylnaltrexone to treat immune suppression |
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| EP1620078A2 (en) * | 2003-05-02 | 2006-02-01 | The Board Of Trustees Of The University Of Illinois | Biodegradable nanoparticles comprising an aminoglycoside and a polymer like a polysaccharide |
| CN101171010B (zh) | 2005-03-07 | 2014-09-17 | 芝加哥大学 | 阿片样物质拮抗剂用于减少内皮细胞增殖和迁移的用途 |
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| CA2609985A1 (en) | 2005-06-03 | 2007-05-10 | The University Of Chicago | Modulation of cell barrier dysfunction |
| PL116330U1 (en) * | 2005-10-31 | 2007-04-02 | Alza Corp | Method for the reduction of alcohol provoked rapid increase in the released dose of the orally administered opioide with prolonged liberation |
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| US20080113030A1 (en) | 2006-11-09 | 2008-05-15 | Ching-Fen Hsiao | Sustained release tamsulosin formulations |
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| US20200101026A1 (en) | 2020-04-02 |
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| EP2306829A4 (en) | 2011-08-24 |
| JP2015091825A (ja) | 2015-05-14 |
| AU2009265034A1 (en) | 2010-01-07 |
| EP2306829B1 (en) | 2017-01-04 |
| AU2009265034B2 (en) | 2015-09-03 |
| US20110250278A1 (en) | 2011-10-13 |
| WO2010002576A1 (en) | 2010-01-07 |
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