ES2427628T3 - Nuevas composiciones de 1-[2-(2,4-dimetil-fenilsulfanil)-fenil]piperazina - Google Patents
Nuevas composiciones de 1-[2-(2,4-dimetil-fenilsulfanil)-fenil]piperazina Download PDFInfo
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- ES2427628T3 ES2427628T3 ES10805414T ES10805414T ES2427628T3 ES 2427628 T3 ES2427628 T3 ES 2427628T3 ES 10805414 T ES10805414 T ES 10805414T ES 10805414 T ES10805414 T ES 10805414T ES 2427628 T3 ES2427628 T3 ES 2427628T3
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- piperazine
- phenyl
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- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Pain & Pain Management (AREA)
- Hematology (AREA)
- Addiction (AREA)
- Rheumatology (AREA)
- Nutrition Science (AREA)
- Hospice & Palliative Care (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23622309P | 2009-08-24 | 2009-08-24 | |
| DK200900950 | 2009-08-24 | ||
| US236223P | 2009-08-24 | ||
| DKPA200900950 | 2009-08-24 | ||
| PCT/DK2010/050216 WO2011023194A2 (en) | 2009-08-24 | 2010-08-23 | New compositions of 1-[2-(2,4-dimethyl-phenylsulfanyl)-phenyl]piperazine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2427628T3 true ES2427628T3 (es) | 2013-10-31 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES10805414T Active ES2427628T3 (es) | 2009-08-24 | 2010-08-23 | Nuevas composiciones de 1-[2-(2,4-dimetil-fenilsulfanil)-fenil]piperazina |
Country Status (32)
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| TW200932233A (en) | 2007-11-13 | 2009-08-01 | Lundbeck & Co As H | Therapeutic uses of compounds having combined SERT, 5-HT3 and 5-HT1a activity |
| BR112012027794A2 (pt) * | 2010-04-30 | 2016-08-02 | Takeda Pharmaceutical | tablete entérico |
| EP2564837B1 (en) | 2010-04-30 | 2019-01-30 | Takeda Pharmaceutical Company Limited | Enteric tablet |
| CN104146953A (zh) * | 2014-07-24 | 2014-11-19 | 李雪梅 | 一种氢溴酸沃替西汀注射液 |
| CN104610195B (zh) * | 2015-01-30 | 2017-06-27 | 上虞京新药业有限公司 | 沃替西汀的天冬氨酸盐或其水合物及其制备方法和用途 |
| JO3456B1 (ar) | 2015-05-13 | 2020-07-05 | H Lundbeck As | فيروتيوكسيتين بيروجلوتامات |
| EP3184102A1 (en) | 2015-12-23 | 2017-06-28 | Hexal AG | Pharmaceutical composition of vortioxetine hydrobromide comprising an inert core formed of an acidic reacting compound |
| EP3184104B1 (en) | 2015-12-23 | 2018-09-12 | Hexal AG | Pharmaceutical composition of vortioxetine hydrobromide comprising vortioxetine hydrobromide in a polyethylene oxide matrix |
| KR20190025556A (ko) | 2016-07-01 | 2019-03-11 | 하. 룬드벡 아크티에셀스카브 | 항우울 효과의 신속한 개시를 위한 보티옥세틴 투여 요법 |
| WO2018065348A1 (en) | 2016-10-05 | 2018-04-12 | Hexal Ag | Novel enteric-coated tablet comprising vortioxetine |
| WO2020087031A1 (en) | 2018-10-26 | 2020-04-30 | The Research Foundation For The State University Of New York | Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia |
| CN112006995A (zh) * | 2020-08-14 | 2020-12-01 | 石药集团中奇制药技术（石家庄）有限公司 | 一种氢溴酸伏硫西汀片的制备方法 |
| CN113398131B (zh) * | 2020-11-05 | 2022-03-01 | 东南大学 | 1-二苯甲基-4-甲基哌嗪类化合物在制备改善肠道菌群紊乱药物中的应用 |
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| GB9514842D0 (en) * | 1995-07-20 | 1995-09-20 | Smithkline Beecham Plc | Novel formulation |
| UA81749C2 (uk) | 2001-10-04 | 2008-02-11 | Х. Луннбек А/С | Фенілпіперазинові похідні як інгібітори зворотного захоплення серотоніну |
| US6866146B2 (en) | 2001-10-09 | 2005-03-15 | Christian M. Heesch | Protective case for string instruments |
| CA2590802A1 (en) * | 2004-12-20 | 2006-06-29 | Collegium Pharmaceutical, Inc. | Pharmaceutical compositions for sleep disorders |
| EP1888550B1 (en) * | 2005-05-12 | 2014-06-25 | AbbVie Bahamas Ltd. | Apoptosis promoters |
| WO2007015270A2 (en) * | 2005-08-02 | 2007-02-08 | Lupin Limited | Novel controlled release compositions of selective serotonin reuptake inhibitors |
| EA015287B1 (ru) * | 2006-06-16 | 2011-06-30 | Х. Лундбекк А/С | 1-[2-(2,4-диметилфенилсульфанил)фенил]пиперазин в качестве соединения с сочетанием активности в отношении повторного захвата серотонина, 5-нти 5-нтдля лечения когнитивного нарушения |
| TW200848411A (en) | 2007-03-20 | 2008-12-16 | Lundbeck & Co As H | Novel therapeutic uses of 1-[2-(2, 4-dimethylphenylsulfanyl)phenyl]-piperazine |
| TW200932233A (en) * | 2007-11-13 | 2009-08-01 | Lundbeck & Co As H | Therapeutic uses of compounds having combined SERT, 5-HT3 and 5-HT1a activity |
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2010
- 2010-08-23 BR BR112012003280A patent/BR112012003280A2/pt not_active IP Right Cessation
- 2010-08-23 HR HRP20130819AT patent/HRP20130819T1/hr unknown
- 2010-08-23 EA EA201290116A patent/EA021321B1/ru not_active IP Right Cessation
- 2010-08-23 GE GEAP201012633A patent/GEP20135950B/en unknown
- 2010-08-23 UA UAA201203101A patent/UA105057C2/uk unknown
- 2010-08-23 SG SG2012008868A patent/SG178325A1/en unknown
- 2010-08-23 JP JP2012525884A patent/JP2013502446A/ja active Pending
- 2010-08-23 NZ NZ598083A patent/NZ598083A/xx not_active IP Right Cessation
- 2010-08-23 ES ES10805414T patent/ES2427628T3/es active Active
- 2010-08-23 US US13/388,750 patent/US20120189697A1/en not_active Abandoned
- 2010-08-23 CA CA2769872A patent/CA2769872A1/en not_active Abandoned
- 2010-08-23 MX MX2012002199A patent/MX2012002199A/es active IP Right Grant
- 2010-08-23 SI SI201030343T patent/SI2470166T1/sl unknown
- 2010-08-23 PT PT108054149T patent/PT2470166E/pt unknown
- 2010-08-23 ME MEP-2013-99A patent/ME01602B/me unknown
- 2010-08-23 DK DK10805414.9T patent/DK2470166T3/da active
- 2010-08-23 CN CN2010800376999A patent/CN102639117A/zh active Pending
- 2010-08-23 KR KR1020127004405A patent/KR20120065328A/ko not_active Withdrawn
- 2010-08-23 EP EP10805414.9A patent/EP2470166B1/en not_active Revoked
- 2010-08-23 PL PL10805414T patent/PL2470166T3/pl unknown
- 2010-08-23 AU AU2010289022A patent/AU2010289022B2/en not_active Ceased
- 2010-08-23 RS RS20130404A patent/RS52959B/sr unknown
- 2010-08-23 WO PCT/DK2010/050216 patent/WO2011023194A2/en not_active Ceased
-
2012
- 2012-01-25 TN TNP2012000038A patent/TN2012000038A1/en unknown
- 2012-02-02 IL IL217914A patent/IL217914A0/en unknown
- 2012-02-07 CR CR20120058A patent/CR20120058A/es unknown
- 2012-02-17 CO CO12028578A patent/CO6612204A2/es not_active Application Discontinuation
- 2012-02-22 CL CL2012000457A patent/CL2012000457A1/es unknown
- 2012-02-23 DO DO2012000050A patent/DOP2012000050A/es unknown
- 2012-02-23 ZA ZA2012/01360A patent/ZA201201360B/en unknown
- 2012-03-21 MA MA34709A patent/MA33598B1/fr unknown
-
2013
- 2013-09-30 SM SM201300108T patent/SMT201300108B/xx unknown
-
2015
- 2015-02-04 US US14/613,693 patent/US20150150867A1/en not_active Abandoned
- 2015-10-19 US US14/886,333 patent/US20160256398A1/en not_active Abandoned
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