ES2381117T3 - Derivados indolilalquilamínicos sustituidos como inhibidores novedosos de la histona-desacetilasa - Google Patents

Derivados indolilalquilamínicos sustituidos como inhibidores novedosos de la histona-desacetilasa Download PDF

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Publication number
ES2381117T3
ES2381117T3 ES05767934T ES05767934T ES2381117T3 ES 2381117 T3 ES2381117 T3 ES 2381117T3 ES 05767934 T ES05767934 T ES 05767934T ES 05767934 T ES05767934 T ES 05767934T ES 2381117 T3 ES2381117 T3 ES 2381117T3
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ES
Spain
Prior art keywords
alkyl
compound
formula
mol
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
ES05767934T
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English (en)
Spanish (es)
Inventor
Marc Gustaaf C Verdonck
Patrick René Angibaud
Bruno Roux
Isabelle Noëlle Constance PILATTE
Peter Ten Holte
Janine Arts
Kristof Van Emelen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Janssen Pharmaceutica NV
Original Assignee
Janssen Pharmaceutica NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Janssen Pharmaceutica NV filed Critical Janssen Pharmaceutica NV
Priority claimed from PCT/EP2005/053612 external-priority patent/WO2006010750A1/en
Application granted granted Critical
Publication of ES2381117T3 publication Critical patent/ES2381117T3/es
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ES05767934T 2004-07-28 2005-07-25 Derivados indolilalquilamínicos sustituidos como inhibidores novedosos de la histona-desacetilasa Active ES2381117T3 (es)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP04077172 2004-07-28
EP04077172 2004-07-28
US59218204P 2004-07-29 2004-07-29
US592182P 2004-07-29
PCT/EP2005/053612 WO2006010750A1 (en) 2004-07-28 2005-07-25 Substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylase

Publications (1)

Publication Number Publication Date
ES2381117T3 true ES2381117T3 (es) 2012-05-23

Family

ID=34928411

Family Applications (1)

Application Number Title Priority Date Filing Date
ES05767934T Active ES2381117T3 (es) 2004-07-28 2005-07-25 Derivados indolilalquilamínicos sustituidos como inhibidores novedosos de la histona-desacetilasa

Country Status (10)

Country Link
CN (1) CN1993353B (xx)
AT (1) ATE542812T1 (xx)
DK (1) DK1781639T3 (xx)
ES (1) ES2381117T3 (xx)
ME (1) ME01444B (xx)
PT (1) PT1781639E (xx)
RS (1) RS52304B (xx)
SI (1) SI1781639T1 (xx)
UA (1) UA93352C2 (xx)
ZA (1) ZA200700764B (xx)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107095871A (zh) * 2016-02-22 2017-08-29 中国科学院上海巴斯德研究所 Quisinostat,一种新型的高效抗疟药物
CN107721980B (zh) * 2017-08-25 2019-07-12 南京医科大学 一类氟尿嘧啶和Quisinosta的乏氧靶向前药及其应用
CN112485233B (zh) * 2020-11-03 2022-08-26 山东师范大学 一种检测去乙酰化酶用纳米传感器及其检测方法和应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE398105T1 (de) * 2002-03-13 2008-07-15 Janssen Pharmaceutica Nv Carbonylamino- derivativate als neue inhibitoren von histone deacetylase

Also Published As

Publication number Publication date
CN1993353B (zh) 2010-12-01
PT1781639E (pt) 2012-05-02
RS52304B (en) 2012-12-31
ATE542812T1 (de) 2012-02-15
UA93352C2 (ru) 2011-02-10
SI1781639T1 (sl) 2012-06-29
ZA200700764B (en) 2008-09-25
CN1993353A (zh) 2007-07-04
DK1781639T3 (da) 2012-05-14
ME01444B (me) 2013-12-20

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