ES2259379T3 - Inhibidores hidrazino carbociclicos de la amina oxidasas que contienen cobre. - Google Patents
Inhibidores hidrazino carbociclicos de la amina oxidasas que contienen cobre.Info
- Publication number
- ES2259379T3 ES2259379T3 ES02751224T ES02751224T ES2259379T3 ES 2259379 T3 ES2259379 T3 ES 2259379T3 ES 02751224 T ES02751224 T ES 02751224T ES 02751224 T ES02751224 T ES 02751224T ES 2259379 T3 ES2259379 T3 ES 2259379T3
- Authority
- ES
- Spain
- Prior art keywords
- hydrogen
- compound
- formula
- disease
- optionally substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
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Classifications
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- C07C243/26—Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids with acylating carboxyl groups bound to hydrogen atoms or to acyclic carbon atoms
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C243/00—Compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes
- C07C243/10—Hydrazines
- C07C243/20—Hydrazines having nitrogen atoms of hydrazine groups bound to carbon atoms of rings other than six-membered aromatic rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/04—One of the condensed rings being a six-membered aromatic ring
- C07C2602/08—One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
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- General Health & Medical Sciences (AREA)
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- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
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- Immunology (AREA)
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- Orthopedic Medicine & Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US902789 | 2001-07-12 | ||
| US09/902,789 US6982286B2 (en) | 2001-07-12 | 2001-07-12 | Carbocyclic hydrazino inhibitors of copper-containing amine oxidases |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2259379T3 true ES2259379T3 (es) | 2006-10-01 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| ES02751224T Expired - Lifetime ES2259379T3 (es) | 2001-07-12 | 2002-07-11 | Inhibidores hidrazino carbociclicos de la amina oxidasas que contienen cobre. |
Country Status (15)
| Country | Link |
|---|---|
| US (2) | US6982286B2 (https=) |
| EP (1) | EP1414426B1 (https=) |
| JP (1) | JP4377221B2 (https=) |
| KR (1) | KR20040017289A (https=) |
| CN (1) | CN1520290A (https=) |
| AT (1) | ATE318589T1 (https=) |
| CA (1) | CA2451569A1 (https=) |
| DE (1) | DE60209504T2 (https=) |
| ES (1) | ES2259379T3 (https=) |
| HU (1) | HUP0401097A3 (https=) |
| IL (1) | IL159205A0 (https=) |
| NO (1) | NO20035139D0 (https=) |
| RU (1) | RU2004103869A (https=) |
| WO (1) | WO2003006003A1 (https=) |
| ZA (1) | ZA200309112B (https=) |
Families Citing this family (48)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US6982286B2 (en) * | 2001-07-12 | 2006-01-03 | Biotie Therapies Corp. | Carbocyclic hydrazino inhibitors of copper-containing amine oxidases |
| FI20022007A0 (fi) * | 2002-11-08 | 2002-11-08 | Juvantia Pharma Ltd Oy | Oromukosaalinen valmiste ja menetelmä sen valmistamiseksi |
| EP1587800A1 (en) * | 2003-01-27 | 2005-10-26 | Astellas Pharma Inc. | Thiazole derivatives and their use as vap-1 inhibitors |
| JP4758337B2 (ja) * | 2003-03-31 | 2011-08-24 | 株式会社アールテック・ウエノ | 血管透過性亢進疾患を治療する方法 |
| ES2335769T3 (es) * | 2003-05-26 | 2010-04-05 | Biotie Therapies Corp. | Vap-1 cristalina y sus usos. |
| FI20031927A0 (fi) * | 2003-12-31 | 2003-12-31 | Faron Pharmaceuticals Oy | Terapeuttisesti vaikuttavia aineita ja niiden käyttö |
| FI20040136A0 (fi) * | 2004-01-30 | 2004-01-30 | Faron Pharmaceuticals Oy | Erityisesti diabeetikoille soveltuvia koostumuksia |
| US8119651B2 (en) * | 2004-01-30 | 2012-02-21 | Biotie Therapies Corp. | Compositions useful especially for treatment or prevention of metabolic syndrome |
| JP2007519688A (ja) * | 2004-01-30 | 2007-07-19 | ファロン ファーマシューティカルズ オサケ ユキチュア | メタボリックシンドロームの治療または予防に特に有効な組成物 |
| JP4140630B2 (ja) * | 2005-11-10 | 2008-08-27 | Ｔｄｋ株式会社 | 磁気ヘッドアセンブリ及び磁気ヘッドアセンブリの製造方法 |
| US8372399B2 (en) | 2006-08-31 | 2013-02-12 | Cardiac Pacemakers, Inc. | Bispecific antibodies and agents to enhance stem cell homing |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3105849A (en) | 1960-02-01 | 1963-10-01 | Ciba Geigy Corp | Bicyclic hydrazinium compounds |
| WO1998055447A1 (en) | 1997-06-05 | 1998-12-10 | Venantius Limited | 3-aminoindane derivatives, process for their preparation and pharmaceutical compositions containing them |
| AU8031698A (en) | 1997-06-05 | 1998-12-21 | Venantius Limited | Indane compounds and their pharmaceutical use |
| JP2004502682A (ja) | 2000-07-05 | 2004-01-29 | バイオティ セラピーズ コーポレイション | 銅含有アミン・オキシダーゼの阻害剤 |
| US6982286B2 (en) * | 2001-07-12 | 2006-01-03 | Biotie Therapies Corp. | Carbocyclic hydrazino inhibitors of copper-containing amine oxidases |
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- 2001-07-12 US US09/902,789 patent/US6982286B2/en not_active Expired - Fee Related
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2002
- 2002-07-11 DE DE60209504T patent/DE60209504T2/de not_active Expired - Lifetime
- 2002-07-11 KR KR10-2004-7000368A patent/KR20040017289A/ko not_active Withdrawn
- 2002-07-11 WO PCT/FI2002/000630 patent/WO2003006003A1/en not_active Ceased
- 2002-07-11 EP EP02751224A patent/EP1414426B1/en not_active Expired - Lifetime
- 2002-07-11 US US10/483,291 patent/US20040236108A1/en not_active Abandoned
- 2002-07-11 ES ES02751224T patent/ES2259379T3/es not_active Expired - Lifetime
- 2002-07-11 IL IL15920502A patent/IL159205A0/xx unknown
- 2002-07-11 JP JP2003511809A patent/JP4377221B2/ja not_active Expired - Fee Related
- 2002-07-11 RU RU2004103869/04A patent/RU2004103869A/ru not_active Application Discontinuation
- 2002-07-11 CN CNA028128915A patent/CN1520290A/zh active Pending
- 2002-07-11 HU HU0401097A patent/HUP0401097A3/hu unknown
- 2002-07-11 AT AT02751224T patent/ATE318589T1/de not_active IP Right Cessation
- 2002-07-11 CA CA002451569A patent/CA2451569A1/en not_active Abandoned
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2003
- 2003-11-19 NO NO20035139A patent/NO20035139D0/no not_active Application Discontinuation
- 2003-11-24 ZA ZA200309112A patent/ZA200309112B/en unknown
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| Publication number | Publication date |
|---|---|
| JP2005501035A (ja) | 2005-01-13 |
| DE60209504D1 (de) | 2006-04-27 |
| DE60209504T2 (de) | 2006-10-12 |
| US20040236108A1 (en) | 2004-11-25 |
| JP4377221B2 (ja) | 2009-12-02 |
| HUP0401097A2 (hu) | 2004-09-28 |
| CN1520290A (zh) | 2004-08-11 |
| ATE318589T1 (de) | 2006-03-15 |
| WO2003006003A1 (en) | 2003-01-23 |
| EP1414426A1 (en) | 2004-05-06 |
| EP1414426B1 (en) | 2006-03-01 |
| US20030125360A1 (en) | 2003-07-03 |
| CA2451569A1 (en) | 2003-01-23 |
| ZA200309112B (en) | 2004-07-23 |
| HUP0401097A3 (en) | 2006-02-28 |
| US6982286B2 (en) | 2006-01-03 |
| RU2004103869A (ru) | 2005-03-27 |
| IL159205A0 (en) | 2004-06-01 |
| KR20040017289A (ko) | 2004-02-26 |
| NO20035139D0 (no) | 2003-11-19 |
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