ES2191350T3 - Mitogenos especificos de osteoblastos y medicamentos que contienen estos compuestos. - Google Patents
Mitogenos especificos de osteoblastos y medicamentos que contienen estos compuestos.Info
- Publication number
- ES2191350T3 ES2191350T3 ES98954302T ES98954302T ES2191350T3 ES 2191350 T3 ES2191350 T3 ES 2191350T3 ES 98954302 T ES98954302 T ES 98954302T ES 98954302 T ES98954302 T ES 98954302T ES 2191350 T3 ES2191350 T3 ES 2191350T3
- Authority
- ES
- Spain
- Prior art keywords
- compounds
- osteoblasts
- medicines containing
- well
- general formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 239000003814 drug Substances 0.000 title abstract 2
- 239000003226 mitogen Substances 0.000 title 1
- 210000000963 osteoblast Anatomy 0.000 title 1
- 239000002253 acid Substances 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 230000004097 bone metabolism Effects 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 238000001727 in vivo Methods 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/06—Phosphorus compounds without P—C bonds
- C07F9/08—Esters of oxyacids of phosphorus
- C07F9/09—Esters of phosphoric acids
- C07F9/091—Esters of phosphoric acids with hydroxyalkyl compounds with further substituents on alkyl
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
- A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Physical Education & Sports Medicine (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Utilización de derivados del ácido lisofosfatidílico de la Fórmula General (I): **fórmula** en donde: R1 =significa alquilo, alquenilo o alquinilo con 6 a 24 átomos de carbono, N = 0 - 12, X = significa oxígeno o NH, así como también de sus sales fisiológicamente aceptables, ésteres, formas ópticamente activas, racematos así como sus derivados, que pueden ser metabolizados in vivo para dar compuestos de la Fórmula general (I), en la producción de medicamentos para el tratamiento de los trastornos del metabolismo óseo.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP97117124A EP0906759A1 (de) | 1997-10-02 | 1997-10-02 | Neue Osteoblastenspezifische Mitogene: Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2191350T3 true ES2191350T3 (es) | 2003-09-01 |
Family
ID=8227430
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES98954302T Expired - Lifetime ES2191350T3 (es) | 1997-10-02 | 1998-09-30 | Mitogenos especificos de osteoblastos y medicamentos que contienen estos compuestos. |
Country Status (16)
Country | Link |
---|---|
US (1) | US6197759B1 (es) |
EP (2) | EP0906759A1 (es) |
JP (2) | JP2001518511A (es) |
KR (1) | KR100392207B1 (es) |
CN (1) | CN1191070C (es) |
AR (1) | AR013538A1 (es) |
AT (1) | ATE232103T1 (es) |
AU (1) | AU738479B2 (es) |
BR (1) | BR9813020A (es) |
CA (1) | CA2304821C (es) |
DE (1) | DE69811253T2 (es) |
DK (1) | DK1019062T3 (es) |
ES (1) | ES2191350T3 (es) |
TR (1) | TR200000875T2 (es) |
WO (1) | WO1999017781A1 (es) |
ZA (1) | ZA988952B (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPWO2003041717A1 (ja) * | 2001-11-12 | 2005-03-03 | 小野薬品工業株式会社 | プロスタグランジン誘導体を有効成分とする局所投与用持続性フィルム状製剤 |
WO2004000232A2 (en) | 2002-06-24 | 2003-12-31 | New York Society For The Ruptured And Crippled Maintaining The Hospital For Special Surgery | Complexed-acidic-phospholipid-collagen composites for bone induction |
KR100789323B1 (ko) * | 2005-07-20 | 2007-12-28 | 주식회사 엔지켐 | 글리세롤 유도체의 위치 선택적 제조방법 및 그 중간체 |
US20100266691A1 (en) * | 2009-04-15 | 2010-10-21 | Battelle Memorial Institute | Agents and Methods to Stimulate Bone Healing |
CN113842504B (zh) * | 2021-09-22 | 2022-12-09 | 苏州大学附属第二医院 | 一种用于骨再生的多功能电纺支架的制备方法 |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4164560A (en) | 1977-01-05 | 1979-08-14 | Folkman Moses J | Systems for the controlled release of macromolecules |
PL151315B1 (pl) * | 1987-04-17 | 1990-08-31 | Sposób wytwarzania nowych związków powierzchniowo czynnych | |
US5645591A (en) | 1990-05-29 | 1997-07-08 | Stryker Corporation | Synthetic bone matrix |
US5238965A (en) * | 1991-05-31 | 1993-08-24 | The Procter & Gamble Company | Methods of using lysophosphatidic acids for regulating skin wrinkles |
MX9203083A (es) | 1991-06-21 | 1994-08-31 | Genetics Inst | Formulaciones farmaceuticas de proteinas osteogenicas. |
US5300687A (en) * | 1991-07-18 | 1994-04-05 | Ortho Pharmaceutical Corporation | Trifluoromethylbenzylphosphonates useful in treating osteoporosis |
WO1993020859A1 (en) | 1992-04-20 | 1993-10-28 | Board Of Regents Of The University Of Washington | Sustained release compositions for delivery of growth factors |
CA2093836A1 (en) | 1992-04-24 | 1993-10-25 | Wayne Gombotz | Biodegradable tgf-.beta. delivery system for bone regeneration |
US5565439A (en) * | 1992-11-24 | 1996-10-15 | The Procter & Gamble Company | Methods of using lysophosphatidic acid for treating hyperproliferative conditions |
NO940913L (no) | 1993-03-26 | 1994-09-27 | Bristol Myers Squibb Co | Preparater for kontrollert frigivelse av biologisk aktiv TGF- |
DE69412538T2 (de) * | 1993-05-18 | 1998-12-24 | Takeda Chemical Industries, Ltd., Osaka | Benzopyran-Derivate und ihre Verwendung |
ES2065855B1 (es) * | 1993-05-31 | 1995-09-01 | Menarini Lab | Procedimiento para la preparacion de nuevos derivados desoxiazafosfolipidicos con accion inhibidora de la fosfolipasa a2, nuevos derivados desoxiazafosfolipidicos obtenidos y utilizacion de los mismos. |
DE19544635A1 (de) | 1995-11-30 | 1997-06-05 | Boehringer Mannheim Gmbh | Neue Aminoalkoholderivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel |
-
1997
- 1997-10-02 EP EP97117124A patent/EP0906759A1/de not_active Withdrawn
-
1998
- 1998-09-30 DE DE69811253T patent/DE69811253T2/de not_active Expired - Fee Related
- 1998-09-30 CN CNB988094193A patent/CN1191070C/zh not_active Expired - Fee Related
- 1998-09-30 KR KR10-2000-7003443A patent/KR100392207B1/ko not_active IP Right Cessation
- 1998-09-30 US US09/508,714 patent/US6197759B1/en not_active Expired - Lifetime
- 1998-09-30 WO PCT/EP1998/006214 patent/WO1999017781A1/en active IP Right Grant
- 1998-09-30 JP JP2000514652A patent/JP2001518511A/ja active Pending
- 1998-09-30 TR TR2000/00875T patent/TR200000875T2/xx unknown
- 1998-09-30 ES ES98954302T patent/ES2191350T3/es not_active Expired - Lifetime
- 1998-09-30 BR BR9813020-0A patent/BR9813020A/pt not_active Application Discontinuation
- 1998-09-30 AT AT98954302T patent/ATE232103T1/de not_active IP Right Cessation
- 1998-09-30 DK DK98954302T patent/DK1019062T3/da active
- 1998-09-30 CA CA002304821A patent/CA2304821C/en not_active Expired - Fee Related
- 1998-09-30 EP EP98954302A patent/EP1019062B1/en not_active Expired - Lifetime
- 1998-09-30 AU AU11483/99A patent/AU738479B2/en not_active Ceased
- 1998-10-01 ZA ZA9808952A patent/ZA988952B/xx unknown
- 1998-10-02 AR ARP980104917A patent/AR013538A1/es unknown
-
2004
- 2004-03-22 JP JP2004082628A patent/JP2004217667A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
ZA988952B (en) | 2000-04-03 |
ATE232103T1 (de) | 2003-02-15 |
EP1019062A1 (en) | 2000-07-19 |
JP2004217667A (ja) | 2004-08-05 |
KR100392207B1 (ko) | 2003-07-23 |
CN1271289A (zh) | 2000-10-25 |
DK1019062T3 (da) | 2003-05-26 |
EP1019062B1 (en) | 2003-02-05 |
DE69811253D1 (de) | 2003-03-13 |
CA2304821A1 (en) | 1999-04-15 |
CN1191070C (zh) | 2005-03-02 |
AR013538A1 (es) | 2000-12-27 |
EP0906759A1 (de) | 1999-04-07 |
JP2001518511A (ja) | 2001-10-16 |
US6197759B1 (en) | 2001-03-06 |
CA2304821C (en) | 2005-08-02 |
AU1148399A (en) | 1999-04-27 |
DE69811253T2 (de) | 2003-12-04 |
BR9813020A (pt) | 2000-08-15 |
KR20010030822A (ko) | 2001-04-16 |
WO1999017781A1 (en) | 1999-04-15 |
AU738479B2 (en) | 2001-09-20 |
TR200000875T2 (tr) | 2000-11-21 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AR038045A1 (es) | Agentes terapeuticos | |
CR6726A (es) | Compuestos azapoliciclicos condensados con arilo | |
PA8487601A1 (es) | Derivados biciclicos sustituidos utiles como agentes contra el cancer | |
UY26332A1 (es) | Nuevos derivados del ácido aminodicarboxílico con propiedades farmacéuticas. | |
ECSP034914A (es) | "azaindoles" | |
AR007118A1 (es) | 4(3h)-quinazolinonas 2,3 disustituidas y composiciones farmaceuticas que las contienen | |
ES2139638T3 (es) | 1,4-piperazinas disustituidas para el tratamiento de las enfermedades del sistema nervioso central y de las enfermedades neuroendocrinas. | |
AR010328A1 (es) | Ester-amidas de acido 3-hidroxi-piridina-2-carboxilico, procedimiento para su preparacion, medicamentos y su utilizacion para la fabricacion demedicamentos | |
ECSP045229A (es) | Piridinonas sustituidas como moduladores de la p38 map quinasa | |
ES2161290T3 (es) | Derivados de quinazolina. | |
ES2139132T3 (es) | Composiciones farmaceuticas activas en la terapia de desordenes del sueño. | |
SV2002000232A (es) | Derivados nuevos de benzoimidazole utiles como agentes antiproliferativos ref. pc 10608abcz/bb | |
PA8432901A1 (es) | Compuestos de piridilpirrol | |
ES2213732T3 (es) | Nuevos esteres derivados de compuestos fenil-ciclohexil sustituidos. | |
AR030541A1 (es) | Acidos aminopropilfosfinicos, su utilizacion para la manufactura de medicamentos, y formulacion farmaceutica | |
ES2164465T3 (es) | Uso de aminometil-cromanos sustituidos para evitar la degeneracion neuronal y para estimular la regeneracion neuronal. | |
AR013462A1 (es) | Nuevos peptidomimeticos para el tratamiento de trastornos oseos, metodos para su produccion y drogas que contienen estos compuestos | |
AR019859A1 (es) | Derivados diaza-espiro[3,5]nonano, un procedimiento para su preparacion, composiciones farmaceuticas que los comprenden y el uso de los mismos para la preparacion de un medicamento | |
ES2191350T3 (es) | Mitogenos especificos de osteoblastos y medicamentos que contienen estos compuestos. | |
AR041865A1 (es) | Derivados terapeuticos de prolina y su uso en el tratamiento de epilepsia y dolor | |
AR005102A1 (es) | Compuestos derivados de octahidro-pirrolo [1,2-a]-pirazina 2,7-sustituidos, composiciones farmaceuticas y uso de dichos compuestos para la fabricacion deun medicamento. | |
AR008244A1 (es) | Compuestos heterociclicos, procedimiento para prepararlos, composiciones farmaceuticas que los comprenden, uso de dichos compuestos en la fabricacion de medicamentos, e intermediarios utiles en la preparacion de dichos compuestos | |
AR016382A1 (es) | Uso de un derivado del acido bencil-indazol metoxialcanoico. | |
ES2052776T3 (es) | Derivados o-alcanoilo del acido 3-amino-2-hidroxipropansulfonico con actividad anticonvulsiva y composiciones farmaceuticas que los contienen para el tratamiento terapeutico de epilepsia. | |
HN2003000015A (es) | Sales estables del acido o acetilsalicilico con aminoacidos basicos i i. |