ES2134563T3 - Cianofenilsulfenil halogenuro y su utilizacion en el procedimiento de preparacion de benzoisotiazol 3-sustituido. - Google Patents
Cianofenilsulfenil halogenuro y su utilizacion en el procedimiento de preparacion de benzoisotiazol 3-sustituido.Info
- Publication number
- ES2134563T3 ES2134563T3 ES96302851T ES96302851T ES2134563T3 ES 2134563 T3 ES2134563 T3 ES 2134563T3 ES 96302851 T ES96302851 T ES 96302851T ES 96302851 T ES96302851 T ES 96302851T ES 2134563 T3 ES2134563 T3 ES 2134563T3
- Authority
- ES
- Spain
- Prior art keywords
- substituted
- halogenuro
- cyanofenilsulfenil
- benzoisotiazole
- preparation procedure
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 150000001875 compounds Chemical class 0.000 abstract 4
- GLUUGHFHXGJENI-UHFFFAOYSA-N Piperazine Chemical compound C1CNCCN1 GLUUGHFHXGJENI-UHFFFAOYSA-N 0.000 abstract 2
- 238000006243 chemical reaction Methods 0.000 abstract 1
- 230000026030 halogenation Effects 0.000 abstract 1
- 238000005658 halogenation reaction Methods 0.000 abstract 1
- 239000002184 metal Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C313/00—Sulfinic acids; Sulfenic acids; Halides, esters or anhydrides thereof; Amides of sulfinic or sulfenic acids, i.e. compounds having singly-bound oxygen atoms of sulfinic or sulfenic groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C313/08—Sulfenic acids; Derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C313/00—Sulfinic acids; Sulfenic acids; Halides, esters or anhydrides thereof; Amides of sulfinic or sulfenic acids, i.e. compounds having singly-bound oxygen atoms of sulfinic or sulfenic groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C313/08—Sulfenic acids; Derivatives thereof
- C07C313/10—Sulfenic acids; Esters thereof
- C07C313/16—Sulfenic acids; Esters thereof having sulfur atoms of sulfenic groups bound to carbon atoms of six-membered aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
UN COMPUESTO DE 2-CIANOBENCENOSULFENIL ESTA REPRESENTADO POR LA FORMULA GENERAL (I): EN DONDE X REPRESENTA CL O BR Y PUEDE SER UTILIZADO PARA LA PREPARACION DE BENCISOTIAZOL 3-SUBSTITUIDO POR LA REACCION DEL COMPUESTO (I) CON UN COMPUESTO DE PIPERAZINA. EL COMPUESTO (I) PUEDE SER PREPARADO POR HALOGENACION DE UN DERIVADO DE 2-CIANOFENILTIO DE LA FORMULA (II): EN DONDE R REPRESENTA H, METAL ALCALINO, 2-CIANOFENILTIO O ALQUILO C{SUB,1-4}.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP09838795A JP3701044B2 (ja) | 1995-04-24 | 1995-04-24 | シアノベンゼンスルフェニルハライドおよびそれを用いる3−置換ベンゾイソチアゾールの製造方法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2134563T3 true ES2134563T3 (es) | 1999-10-01 |
Family
ID=14218454
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES96302851T Expired - Lifetime ES2134563T3 (es) | 1995-04-24 | 1996-04-24 | Cianofenilsulfenil halogenuro y su utilizacion en el procedimiento de preparacion de benzoisotiazol 3-sustituido. |
Country Status (9)
| Country | Link |
|---|---|
| US (2) | US5679827A (es) |
| EP (1) | EP0741129B1 (es) |
| JP (1) | JP3701044B2 (es) |
| KR (1) | KR100387538B1 (es) |
| CN (2) | CN1187346C (es) |
| CA (1) | CA2174797C (es) |
| DE (1) | DE69602802T2 (es) |
| ES (1) | ES2134563T3 (es) |
| TW (1) | TW326033B (es) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0874834B1 (en) * | 1995-11-07 | 2000-12-13 | Pfizer Inc. | Processes and intermediates for preparing 3-(1-piperazinyl)-1,2-benzisothiazole |
| JP3996228B2 (ja) * | 1996-10-11 | 2007-10-24 | 住友精化株式会社 | 3−ピペラジニルベンズイソチアゾール類の製造法 |
| TWI232214B (en) * | 1998-04-16 | 2005-05-11 | Shionogi & Co | Preparation of aryl sulfenyl halide |
| AU5197199A (en) * | 1999-08-12 | 2001-03-13 | Nippon Fine Chemical Co., Ltd. | Processes for the preparation of aromatic sulfenyl chlorides and so forth |
| WO2004002950A1 (ja) * | 2002-06-28 | 2004-01-08 | Shimadzu Corporation | スルフェニル化合物、ラベル化試薬、及びペプチドの解析方法 |
| WO2013014665A1 (en) | 2011-07-28 | 2013-01-31 | Mapi Pharma Ltd. | Intermediate compounds and process for the preparation of lurasidone and salts thereof |
| CN105669588B (zh) * | 2016-03-16 | 2017-11-07 | 天津大学 | 苯并异噻唑类衍生物的制备方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2609864C2 (de) * | 1976-03-10 | 1984-02-16 | Basf Ag, 6700 Ludwigshafen | Verfahren zur Herstellung von 3-Amino-1,2-benzisothiazolen |
| EP0053652A1 (de) * | 1980-11-10 | 1982-06-16 | Klaus Arlt | Energie-Erzeuger: Maschinelle Vorrichtung zur Erzeugung von Energie durch Schwerkraftwirkung |
| US4590196A (en) * | 1984-08-23 | 1986-05-20 | Bristol-Myers Company | Analgesic 1,2-benzisothiazol-3-ylpiperazine derivatives |
| JPH0625181B2 (ja) * | 1985-03-27 | 1994-04-06 | 住友製薬株式会社 | 新規なイミド誘導体 |
| JPS6383085A (ja) * | 1986-09-26 | 1988-04-13 | Sumitomo Pharmaceut Co Ltd | 新規なイミド誘導体 |
| JPS6383067A (ja) * | 1986-09-26 | 1988-04-13 | Sumitomo Pharmaceut Co Ltd | 新規コハク酸イミド誘導体 |
| TW241263B (es) * | 1991-08-22 | 1995-02-21 | Hoechst Roussel Pharma | |
| US5359068A (en) * | 1993-06-28 | 1994-10-25 | Pfizer Inc. | Processes and intermediates for the preparation of 5-[2-(4-(benzoisothiazol-3-yl)-piperazin-1-yl)ethyl]-6-chloro-1,3-dihydro-indol-2-one |
-
1995
- 1995-04-24 JP JP09838795A patent/JP3701044B2/ja not_active Expired - Fee Related
-
1996
- 1996-04-10 US US08/630,730 patent/US5679827A/en not_active Expired - Lifetime
- 1996-04-12 TW TW085104333A patent/TW326033B/zh not_active IP Right Cessation
- 1996-04-23 CA CA002174797A patent/CA2174797C/en not_active Expired - Fee Related
- 1996-04-23 KR KR1019960012366A patent/KR100387538B1/ko not_active Expired - Fee Related
- 1996-04-24 CN CNB001086383A patent/CN1187346C/zh not_active Expired - Fee Related
- 1996-04-24 EP EP96302851A patent/EP0741129B1/en not_active Expired - Lifetime
- 1996-04-24 CN CN96106019A patent/CN1061975C/zh not_active Expired - Fee Related
- 1996-04-24 ES ES96302851T patent/ES2134563T3/es not_active Expired - Lifetime
- 1996-04-24 DE DE69602802T patent/DE69602802T2/de not_active Expired - Lifetime
-
1997
- 1997-05-21 US US08/861,426 patent/US5756806A/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| EP0741129B1 (en) | 1999-06-09 |
| JPH08291134A (ja) | 1996-11-05 |
| CN1061975C (zh) | 2001-02-14 |
| DE69602802T2 (de) | 1999-10-21 |
| CA2174797C (en) | 2007-01-09 |
| CN1138032A (zh) | 1996-12-18 |
| CN1187346C (zh) | 2005-02-02 |
| US5679827A (en) | 1997-10-21 |
| US5756806A (en) | 1998-05-26 |
| DE69602802D1 (de) | 1999-07-15 |
| CN1289770A (zh) | 2001-04-04 |
| JP3701044B2 (ja) | 2005-09-28 |
| TW326033B (en) | 1998-02-01 |
| EP0741129A2 (en) | 1996-11-06 |
| EP0741129A3 (en) | 1997-05-07 |
| KR100387538B1 (ko) | 2003-11-28 |
| KR960037647A (ko) | 1996-11-19 |
| CA2174797A1 (en) | 1996-10-25 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ES2173477T3 (es) | Derivados de tetrahidronaftaleno y su utilizacion terapeutica. | |
| DK0674642T3 (da) | Pyrazolopyrimidiner som CRF-antagonister | |
| EE03869B1 (et) | Sulfiinhappe derivaadid, nende valmistamine ja kasutamine | |
| YU49312B (sh) | Kristalni hidratni derivati 3,4,4-trisupstituisanih - peperidinil-n-alkilkarboksilata, njihovi intermedijari i postupak za dobijanje | |
| ES8206440A1 (es) | Un procedimiento para la preparacion del enantiomero (-) de la n-metil-3-(2metilfenoxi)-3-fenilpropilamina. | |
| AU6613896A (en) | Chemical compounds | |
| ES2140565T3 (es) | Nuevos derivados de pirazina-carboxamida, su preparacion y su utilizacion en medicamentos. | |
| IT1269176B (it) | Eterobicicli ad attivita' fungicida | |
| AR248010A1 (es) | Un procedimiento de preparacion del 4-metil-2'-ciano-bifenilo | |
| ES2157992T3 (es) | Alcoxi-alquil-carbamatos de imidazo(1,2-a)piridinas. | |
| BR0115501A (pt) | Processo quìmico e novos intermediários | |
| IT1271026B (it) | Derivati dell'acido b-amminopropionico ad attivita' fungicida | |
| FI860073A0 (fi) | 6,7-disubstituerade 1-cyklopropyl-1,4-dihydro-4-oxo-1,8-naftyridin-3-karboxylsyror. | |
| NZ504084A (en) | Processes for producing 7-isoindolinequinolonecarboxylic derivatives and its intermediates, as well as salts of 7-isoindolinequinolonecarboxylic acid derivatives, its hydrates and composition comprising the same as active ingredient | |
| ES2134563T3 (es) | Cianofenilsulfenil halogenuro y su utilizacion en el procedimiento de preparacion de benzoisotiazol 3-sustituido. | |
| AU1079283A (en) | A fungicidal indanylbenzamide | |
| FI872636A0 (fi) | Substituerade 4-bensyl -piperazinylfoereningar. | |
| MX9200003A (es) | Procedimiento e intermediarios para preparar azabiciclo (2.2.2)octan-3-iminas. | |
| MX9204179A (es) | Derivados de imidazo(2,1-b)benzotiazola-3-acetamida, su preparacion y su aplicacion en terapeutica. | |
| DE60121048D1 (de) | PYRAZINOi1'2':1,6öPYRIDOi3,4-BöINDOLDERIVATE | |
| AR248126A1 (es) | Nuevos derivados sustituidos de bicicloheptanodiona, procedimiento para obtenerlos y composiciones herbicidas que los contienen. | |
| ES2043738T3 (es) | Procedimiento para la reduccion de cetonas. | |
| IT1271443B (it) | Derivati eterobiciclici ad attivita' fungicida | |
| FI930092A0 (fi) | Indanopyrrolidinkarbamater | |
| ES8801669A1 (es) | Un procedimiento para preparar nuevos compuestos de 2-oxa-0 aza-pregnano. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG2A | Definitive protection |
Ref document number: 741129 Country of ref document: ES |