ES2087130T3 - Procedimiento para la preparacion de compuestos de purina. - Google Patents

Procedimiento para la preparacion de compuestos de purina.

Info

Publication number
ES2087130T3
ES2087130T3 ES90310444T ES90310444T ES2087130T3 ES 2087130 T3 ES2087130 T3 ES 2087130T3 ES 90310444 T ES90310444 T ES 90310444T ES 90310444 T ES90310444 T ES 90310444T ES 2087130 T3 ES2087130 T3 ES 2087130T3
Authority
ES
Spain
Prior art keywords
formula
compound
chem
alkoxy
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES90310444T
Other languages
English (en)
Inventor
Graham Richard Geen
Trevor John Grinter
Stephen Moore
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beecham Group PLC
Original Assignee
Beecham Group PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group PLC filed Critical Beecham Group PLC
Application granted granted Critical
Publication of ES2087130T3 publication Critical patent/ES2087130T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/40Heterocyclic compounds containing purine ring systems with halogen atoms or perhalogeno-alkyl radicals directly attached in position 2 or 6
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Catalysts (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Compounds Of Unknown Constitution (AREA)

Abstract

UN PROCESO PARA PREPARAR UN COMPONENTE DE FORMULA (A): EN LA QUE X ES HIDROGENO, HIDROXIDO, CLORO, C1-6 ALCOXI, O ALCOXI FENIL C1-6 Y; RA Y RB SON HIDROGENO, DERIVADOS DE LOS ANTERIORES QUE INCLUYEN ACILO Y FOSFATO. TAL PROCESO COMPRENDE PREPARAR UN COMPONENTE DE LA FORMULA I.
ES90310444T 1989-09-28 1990-09-25 Procedimiento para la preparacion de compuestos de purina. Expired - Lifetime ES2087130T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB898922076A GB8922076D0 (en) 1989-09-28 1989-09-28 Novel process

Publications (1)

Publication Number Publication Date
ES2087130T3 true ES2087130T3 (es) 1996-07-16

Family

ID=10663861

Family Applications (1)

Application Number Title Priority Date Filing Date
ES90310444T Expired - Lifetime ES2087130T3 (es) 1989-09-28 1990-09-25 Procedimiento para la preparacion de compuestos de purina.

Country Status (19)

Country Link
US (1) US5220024A (es)
EP (1) EP0420559B1 (es)
JP (1) JP2877931B2 (es)
KR (1) KR0158208B1 (es)
AT (1) ATE138379T1 (es)
AU (1) AU627939B2 (es)
CA (1) CA2026238A1 (es)
DE (1) DE69027084T2 (es)
ES (1) ES2087130T3 (es)
FI (1) FI904774A0 (es)
GB (1) GB8922076D0 (es)
GR (1) GR3020455T3 (es)
HU (1) HU207319B (es)
IE (1) IE903465A1 (es)
MA (1) MA21960A1 (es)
NO (1) NO904191L (es)
NZ (1) NZ235465A (es)
PT (1) PT95427B (es)
ZA (1) ZA907682B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8817607D0 (en) * 1988-07-23 1988-09-01 Beecham Group Plc Novel process
AT412211B (de) * 1996-07-20 2004-11-25 Novartis Int Pharm Ltd Verfahren zur herstellung von penciclovir und famciclovir
GB9615276D0 (en) * 1996-07-20 1996-09-04 Smithkline Beecham Plc Pharmaceuticals
GB9615275D0 (en) * 1996-07-20 1996-09-04 Smithkline Beecham Plc Pharmaceuticals
GB9615253D0 (en) * 1996-07-20 1996-09-04 Smithkline Beecham Plc Pharmaceuticals
CA2251481A1 (en) 1997-11-12 1999-05-12 Junichi Yasuoka Purine derivatives having cyclopropane ring
MY141789A (en) * 2001-01-19 2010-06-30 Lg Chem Investment Ltd Novel acyclic nucleoside phosphonate derivatives, salts thereof and process for the preparation of the same.
KR100573860B1 (ko) * 2003-06-13 2006-04-25 경동제약 주식회사 2-아미노-9-(2-치환에틸)푸린을 이용한 9-[4-아세톡시-3-(아세톡시메틸)부트-1-일]-2-아미노푸린의 제조방법
KR102043754B1 (ko) 2018-04-25 2019-11-12 (주)세원물산 코일 휨 방지 금형장치

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL73682A (en) * 1983-12-20 1991-08-16 Medivir Ab Antiviral pharmaceutical compositions containing 9-hydroxy aliphatic derivatives of guanine,some new such derivatives and process for their preparation
DE3582399D1 (de) * 1984-09-20 1991-05-08 Beecham Group Plc Purin-derivate und ihre pharmazeutische verwendung.
SE8406538D0 (sv) * 1984-12-21 1984-12-21 Astra Laekemedel Ab Novel derivatives of purine
DE3671227D1 (de) * 1985-07-27 1990-06-21 Beecham Group Plc 9-substituierte guaninmonohydrate.
NZ225447A (en) * 1987-07-20 1991-12-23 Merck & Co Inc Piperazinyl derivatives of purine and purine isosteres and pharmaceutical compositions
GB8724765D0 (en) * 1987-10-22 1987-11-25 Beecham Group Plc Process
GB8817607D0 (en) * 1988-07-23 1988-09-01 Beecham Group Plc Novel process
US4988703A (en) * 1989-05-22 1991-01-29 Abbott Laboratories Carbocyclic nucleoside analogs with antiviral activity

Also Published As

Publication number Publication date
EP0420559A2 (en) 1991-04-03
IE903465A1 (en) 1991-04-10
HU207319B (en) 1993-03-29
KR910006288A (ko) 1991-04-29
GB8922076D0 (en) 1989-11-15
HUT55018A (en) 1991-04-29
NO904191D0 (no) 1990-09-26
MA21960A1 (fr) 1991-04-01
EP0420559B1 (en) 1996-05-22
KR0158208B1 (ko) 1998-12-01
AU6325890A (en) 1991-04-11
EP0420559A3 (en) 1992-04-15
DE69027084D1 (de) 1996-06-27
JP2877931B2 (ja) 1999-04-05
NO904191L (no) 1991-04-02
DE69027084T2 (de) 1996-10-24
CA2026238A1 (en) 1991-03-29
FI904774A0 (fi) 1990-09-27
NZ235465A (en) 1993-01-27
PT95427A (pt) 1991-05-22
US5220024A (en) 1993-06-15
AU627939B2 (en) 1992-09-03
GR3020455T3 (en) 1996-10-31
HU906228D0 (en) 1991-03-28
ATE138379T1 (de) 1996-06-15
ZA907682B (en) 1992-08-26
PT95427B (pt) 1996-08-30
JPH03120279A (ja) 1991-05-22

Similar Documents

Publication Publication Date Title
PT89134A (pt) Processo para a preparacao de compostos de acido propano-fosfinico substituido
MX9604942A (es) Preparacion de purina.
PT594291E (pt) Novos processos para a producao de derivados 13-eter de milbemicinas e de novos intermediarios para esse fim
ES2087130T3 (es) Procedimiento para la preparacion de compuestos de purina.
ES8801377A1 (es) Procedimiento para la produccion de d-l-amino acidos
AU2827792A (en) Process for the preparation of phenylaldehydes
KR880005129A (ko) 신규 화합물
PT991651E (pt) Intermediarios de carbapenem estabilizados e uso sintetico
ATE97903T1 (de) Titan- und zirkonium-pyrophosphate, ihre herstellung und verwendung.
PT89098A (pt) Processo para a preparacao de derivados de guanina
PT98700A (pt) Processo para a preparacao de acidos aminometanofosfonico e de acidos aminometil-fosfinicos
PT94244A (pt) Processo para a preparacao de compostos de acido propano-fosfinico p-substituido
ES2058192T3 (es) Diesteres de acido fosforico y sus sales.
BR8206330A (pt) Processo para a producao de acido aminometilfosfonico
HU9600300D0 (en) Thiocarbamoyl derivatives using as antimicrobial agents and process for producing of these
ES2028790T3 (es) Procedimiento para la preparacion de compuestos de beta-lactama.
CO4370020A1 (es) Proceso para la preparacion de agentes antivirales derivados de purina
ES2091010T3 (es) Procedimiento para la obtencion de acido 3-hidroxifenilacetico.
ES2194871T3 (es) Deshidrogenasa del acido clavulanico, preparacion y uso para la produccion de acido clavulanico.

Legal Events

Date Code Title Description
FG2A Definitive protection

Ref document number: 0420559

Country of ref document: ES