ES2029776T1 - Procedimiento para la preparacion de composiciones farmaceuticas que contienen bromocriptina con una alta estabilidad. - Google Patents
Procedimiento para la preparacion de composiciones farmaceuticas que contienen bromocriptina con una alta estabilidad.Info
- Publication number
- ES2029776T1 ES2029776T1 ES199090106403T ES90106403T ES2029776T1 ES 2029776 T1 ES2029776 T1 ES 2029776T1 ES 199090106403 T ES199090106403 T ES 199090106403T ES 90106403 T ES90106403 T ES 90106403T ES 2029776 T1 ES2029776 T1 ES 2029776T1
- Authority
- ES
- Spain
- Prior art keywords
- preparation
- procedure
- pharmaceutical compositions
- compositions containing
- high stability
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- OZVBMTJYIDMWIL-AYFBDAFISA-N bromocriptine Chemical compound C1=CC(C=2[C@H](N(C)C[C@@H](C=2)C(=O)N[C@]2(C(=O)N3[C@H](C(N4CCC[C@H]4[C@]3(O)O2)=O)CC(C)C)C(C)C)C2)=C3C2=C(Br)NC3=C1 OZVBMTJYIDMWIL-AYFBDAFISA-N 0.000 title abstract 2
- 229960002802 bromocriptine Drugs 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 239000004480 active ingredient Substances 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 239000000546 pharmaceutical excipient Substances 0.000 abstract 2
- 239000002775 capsule Substances 0.000 abstract 1
- 239000008187 granular material Substances 0.000 abstract 1
- 238000005469 granulation Methods 0.000 abstract 1
- 230000003179 granulation Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/48—Ergoline derivatives, e.g. lysergic acid, ergotamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
PROCESOS PARA LA PREPARACION DE TABLETAS O CAPSULAS DE BROMOCRIPTINA, EN DONDE EL INGREDIENTE ACTIVO ESTA PROTEGIDO POR INCLUSION EN UN EXCIPIENTE O POR GRANULACION SEPARADA DE LOS EXCIPIENTES Y MEZCLADO DEL GRANULADO CON UNA MEZCLA DEL INGREDIENTE ACTIVO Y UN EXCIPIENTE QUE TIENE BAJO CONTENIDO DE HUMEDAD.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT8920063A IT1235053B (it) | 1989-04-07 | 1989-04-07 | Metodi per la preparazione di composizioni farmaceutiche a base di bromocriptina dotate di elevata stabilita' e prodotti derivanti. |
Publications (2)
Publication Number | Publication Date |
---|---|
ES2029776T1 true ES2029776T1 (es) | 1992-10-01 |
ES2029776T3 ES2029776T3 (es) | 1995-02-01 |
Family
ID=11163518
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES90106403T Expired - Lifetime ES2029776T3 (es) | 1989-04-07 | 1990-04-04 | Procedimiento para la preparacion de composiciones farmaceuticas que contienen bromocriptina con gran estabilidad y productos relacionados. |
Country Status (9)
Country | Link |
---|---|
US (1) | US5066495A (es) |
EP (1) | EP0391374B1 (es) |
AT (1) | ATE114968T1 (es) |
DD (1) | DD293961B5 (es) |
DE (2) | DE391374T1 (es) |
DK (1) | DK0391374T3 (es) |
ES (1) | ES2029776T3 (es) |
GR (1) | GR900300172T1 (es) |
IT (1) | IT1235053B (es) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2030174C (en) * | 1990-01-10 | 1996-12-24 | Anthony H. Cincotta | Process for the long term reduction of body fat stores, insulin resistance, hyperinsulinemia and hypoglycemia in vertebrates |
US5292520A (en) * | 1990-09-13 | 1994-03-08 | Akzo N.V. | Stabilized solid pharmaceutical composition containing acid addition salts of a basic drug and an alkaline stabilizer |
US5225204A (en) * | 1991-11-05 | 1993-07-06 | Chen Jivn Ren | Stable dosage of levothyroxine sodium and process of production |
IL112106A0 (en) * | 1993-12-22 | 1995-03-15 | Ergo Science Inc | Accelerated release composition containing bromocriptine |
SI9700186B (sl) | 1997-07-14 | 2006-10-31 | Lek, Tovarna Farmacevtskih In Kemicnih Izdelkov, D.D. | Nova farmacevtska oblika z nadzorovanim sproscanjem zdravilnih ucinkovin |
US6129931A (en) * | 1998-09-03 | 2000-10-10 | Isp Investments Inc. | Controlled-release, drug-delivery tableted composition including a complex between poly(maleic diacid-alkyl vinyl ether) and polyvinylpyrrolidone |
US8226972B2 (en) * | 2001-12-20 | 2012-07-24 | Femmepharma Holding Company, Inc. | Vaginal delivery of drugs |
US8821915B2 (en) | 2002-08-09 | 2014-09-02 | Veroscience, Llc | Therapeutic process for the treatment of the metabolic syndrome and associated metabolic disorders |
US9173836B2 (en) | 2003-01-02 | 2015-11-03 | FemmeParma Holding Company, Inc. | Pharmaceutical preparations for treatments of diseases and disorders of the breast |
AU2004203700B2 (en) * | 2003-01-02 | 2007-06-21 | Femmepharma Holding Company, Inc. | Pharmaceutical preparations for treatments of diseases and disorders of the breast |
AU2007216882B2 (en) * | 2003-01-02 | 2010-03-11 | Femmepharma Holding Company, Inc. | Pharmaceutical preparations for treatment of diseases and disorders of the breast |
WO2008083158A2 (en) * | 2006-12-26 | 2008-07-10 | Femmepharma Holding Company, Inc. | Topical administration of danazol |
GB0715628D0 (en) * | 2007-08-10 | 2007-09-19 | Generics Uk Ltd | Solid valsartan composition |
US9352025B2 (en) | 2009-06-05 | 2016-05-31 | Veroscience Llc | Combination of dopamine agonists plus first phase insulin secretagogues for the treatment of metabolic disorders |
US20110003000A1 (en) * | 2009-07-06 | 2011-01-06 | Femmepharma Holding Company, Inc. | Transvaginal Delivery of Drugs |
US8431155B1 (en) | 2012-04-30 | 2013-04-30 | Veroscience Llc | Bromocriptine formulations |
CN105640901A (zh) * | 2014-11-10 | 2016-06-08 | 匈牙利吉瑞大药厂 | 一种利用新型生产工艺制备甲磺酸溴隐亭片的方法及其应用 |
WO2017184875A1 (en) | 2016-04-20 | 2017-10-26 | Veroscience Llc | Composition and method for treating metabolic disorders |
CA3079522A1 (en) | 2017-10-18 | 2019-04-25 | Veroscience Llc | Improved bromocriptine formulations |
CN117323305B (zh) * | 2023-11-07 | 2024-06-07 | 杭州沐源生物医药科技有限公司 | 溴隐亭片剂及其制备方法 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE627516A (es) * | 1962-01-25 | |||
US3836618A (en) * | 1971-12-23 | 1974-09-17 | American Home Prod | Process for the uniform distribution of a drug on a granulated base |
NL7314066A (es) * | 1972-10-18 | 1974-04-22 | ||
DE3045135A1 (de) * | 1980-11-29 | 1982-06-09 | Sandoz-Patent-GmbH, 7850 Lörrach | Pharmazeutische kompositionen enthaltende bioabbaubare polymere |
US4479911A (en) * | 1982-01-28 | 1984-10-30 | Sandoz, Inc. | Process for preparation of microspheres and modification of release rate of core material |
GR79340B (es) * | 1982-07-06 | 1984-10-22 | Sterwin Ag | |
US4742054A (en) * | 1982-11-23 | 1988-05-03 | Naftchi Nosrat E | Treatment of mammals suffering from damage to the central nervous system |
GB2154874B (en) * | 1984-02-29 | 1987-11-04 | Sandoz Ltd | Bromoscriptine compositions |
-
1989
- 1989-04-07 IT IT8920063A patent/IT1235053B/it active
-
1990
- 1990-03-30 US US07/502,520 patent/US5066495A/en not_active Expired - Lifetime
- 1990-04-04 ES ES90106403T patent/ES2029776T3/es not_active Expired - Lifetime
- 1990-04-04 DE DE199090106403T patent/DE391374T1/de active Pending
- 1990-04-04 EP EP90106403A patent/EP0391374B1/en not_active Expired - Lifetime
- 1990-04-04 DK DK90106403.0T patent/DK0391374T3/da active
- 1990-04-04 DE DE69014691T patent/DE69014691T2/de not_active Expired - Lifetime
- 1990-04-04 AT AT90106403T patent/ATE114968T1/de not_active IP Right Cessation
- 1990-04-05 DD DD33947390A patent/DD293961B5/de not_active IP Right Cessation
-
1991
- 1991-09-27 GR GR90300172T patent/GR900300172T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
US5066495A (en) | 1991-11-19 |
ES2029776T3 (es) | 1995-02-01 |
DE391374T1 (de) | 1991-02-28 |
DK0391374T3 (da) | 1995-04-24 |
ATE114968T1 (de) | 1994-12-15 |
EP0391374B1 (en) | 1994-12-07 |
EP0391374A2 (en) | 1990-10-10 |
IT8920063A0 (it) | 1989-04-07 |
DE69014691D1 (de) | 1995-01-19 |
IT1235053B (it) | 1992-06-17 |
DE69014691T2 (de) | 1995-04-20 |
EP0391374A3 (en) | 1992-07-01 |
GR900300172T1 (en) | 1991-09-27 |
DD293961B5 (de) | 1994-11-10 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG2A | Definitive protection |
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