EG15987A - Process and intermediates for preparation of 1,1-dioxopenicillan-oyloxymethyl 6-beta-aminopenicillanate - Google Patents

Process and intermediates for preparation of 1,1-dioxopenicillan-oyloxymethyl 6-beta-aminopenicillanate

Info

Publication number
EG15987A
EG15987A EG681/83A EG68183A EG15987A EG 15987 A EG15987 A EG 15987A EG 681/83 A EG681/83 A EG 681/83A EG 68183 A EG68183 A EG 68183A EG 15987 A EG15987 A EG 15987A
Authority
EG
Egypt
Prior art keywords
aminopenicillanate
beta
preparation
dioxopenicillan
oyloxymethyl
Prior art date
Application number
EG681/83A
Other languages
English (en)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of EG15987A publication Critical patent/EG15987A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Cultivation Of Plants (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cephalosporin Compounds (AREA)
EG681/83A 1982-11-01 1983-11-01 Process and intermediates for preparation of 1,1-dioxopenicillan-oyloxymethyl 6-beta-aminopenicillanate EG15987A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/438,228 US4530792A (en) 1982-11-01 1982-11-01 Process and intermediates for preparation of 1,1-dioxopenicillanoyloxymethyl 6-beta-aminopenicillanate

Publications (1)

Publication Number Publication Date
EG15987A true EG15987A (en) 1989-03-30

Family

ID=23739781

Family Applications (1)

Application Number Title Priority Date Filing Date
EG681/83A EG15987A (en) 1982-11-01 1983-11-01 Process and intermediates for preparation of 1,1-dioxopenicillan-oyloxymethyl 6-beta-aminopenicillanate

Country Status (25)

Country Link
US (1) US4530792A (fi)
EP (1) EP0108545B1 (fi)
JP (1) JPS5998090A (fi)
KR (1) KR860001494B1 (fi)
AT (1) ATE24322T1 (fi)
AU (1) AU541962B2 (fi)
CA (1) CA1204736A (fi)
CS (1) CS235986B2 (fi)
DD (1) DD213926A5 (fi)
DE (1) DE3368417D1 (fi)
DK (1) DK163515C (fi)
EG (1) EG15987A (fi)
ES (1) ES8602014A1 (fi)
FI (1) FI76576C (fi)
GR (1) GR78943B (fi)
GT (1) GT198303898A (fi)
HU (1) HU189769B (fi)
IE (1) IE56179B1 (fi)
IL (1) IL70095A (fi)
NZ (1) NZ206108A (fi)
PH (1) PH19573A (fi)
PL (1) PL142735B1 (fi)
PT (1) PT77580B (fi)
YU (1) YU43989B (fi)
ZA (1) ZA838091B (fi)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH01139584A (ja) * 1987-11-25 1989-06-01 Yoshitomi Pharmaceut Ind Ltd ペニシラン酸化合物の製造法
GB2231049A (en) * 1989-04-14 1990-11-07 Yoshitomi Pharmaceutical Method for producing diester compounds
ATE108797T1 (de) * 1990-04-13 1994-08-15 Pfizer Verfahren für sultamicillinzwischenprodukt.

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3896110A (en) * 1971-10-04 1975-07-22 American Home Prod Process for preparation of 6-aminopenicillanic acid
US3929767A (en) * 1971-11-16 1975-12-30 Yamanouchi Pharma Co Ltd Process of producing semi-synthetic penicillin
FR2275460A1 (fr) * 1974-06-20 1976-01-16 Schmoller & Bompard Procede pour la preparation de l'acide 6-aminopenicillanique
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
US4364957A (en) * 1979-09-26 1982-12-21 Pfizer Inc. Bis-esters of alkanediols as antibacterial agents
US4376076A (en) * 1981-03-23 1983-03-08 Pfizer Inc. Bis-esters of 1,1-alkanediols with 6-beta-hydroxymethylpenicillanic acid 1,1-dioxide
US4359472A (en) * 1981-12-22 1982-11-16 Pfizer Inc. Bis-hydroxymethyl carbonate bridged antibacterial agents
US4375434A (en) * 1982-06-21 1983-03-01 Pfizer Inc. Process for 6'-amino-penicillanoyloxymethyl penicillanate 1,1-dioxide

Also Published As

Publication number Publication date
DK163515B (da) 1992-03-09
YU43989B (en) 1990-02-28
AU541962B2 (en) 1985-01-31
IE832539L (en) 1984-05-01
ZA838091B (en) 1985-06-26
EP0108545A1 (en) 1984-05-16
JPH0329796B2 (fi) 1991-04-25
PH19573A (en) 1986-05-21
ES526942A0 (es) 1985-11-01
ATE24322T1 (de) 1987-01-15
FI76576B (fi) 1988-07-29
PL142735B1 (en) 1987-11-30
CA1204736A (en) 1986-05-20
GR78943B (fi) 1984-10-02
FI833961A (fi) 1984-05-02
HU189769B (en) 1986-07-28
AU2082183A (en) 1984-05-10
JPS5998090A (ja) 1984-06-06
IE56179B1 (en) 1991-05-08
IL70095A0 (en) 1984-01-31
DK497483A (da) 1984-05-02
IL70095A (en) 1988-03-31
DK163515C (da) 1992-08-24
FI833961A0 (fi) 1983-10-28
FI76576C (fi) 1988-11-10
KR860001494B1 (ko) 1986-09-27
DD213926A5 (de) 1984-09-26
CS235986B2 (en) 1985-05-15
US4530792A (en) 1985-07-23
PT77580B (en) 1986-05-27
EP0108545B1 (en) 1986-12-17
YU216283A (en) 1986-02-28
ES8602014A1 (es) 1985-11-01
PT77580A (en) 1983-11-01
GT198303898A (es) 1985-04-20
KR840007009A (ko) 1984-12-04
PL244352A1 (en) 1985-02-27
NZ206108A (en) 1986-06-11
DK497483D0 (da) 1983-10-31
DE3368417D1 (en) 1987-01-29

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