EE9400296A - Piperidinüültioindooli derivaadid, ravimvormid, aktiivne valuvaigisti, nende valmistamise meetodid - Google Patents

Piperidinüültioindooli derivaadid, ravimvormid, aktiivne valuvaigisti, nende valmistamise meetodid

Info

Publication number
EE9400296A
EE9400296A EE9400296A EE9400296A EE9400296A EE 9400296 A EE9400296 A EE 9400296A EE 9400296 A EE9400296 A EE 9400296A EE 9400296 A EE9400296 A EE 9400296A EE 9400296 A EE9400296 A EE 9400296A
Authority
EE
Estonia
Prior art keywords
piperidinylthioindole
derivatives
preparation
methods
dosage forms
Prior art date
Application number
EE9400296A
Other languages
English (en)
Estonian (et)
Inventor
Bru-Magniez Nicole
Potin Dominique
Teulon Jean-Marie
Original Assignee
Laboratoires Upsa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Laboratoires Upsa filed Critical Laboratoires Upsa
Publication of EE9400296A publication Critical patent/EE9400296A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
EE9400296A 1993-05-18 1994-11-23 Piperidinüültioindooli derivaadid, ravimvormid, aktiivne valuvaigisti, nende valmistamise meetodid EE9400296A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9305966A FR2705346B1 (fr) 1993-05-18 1993-05-18 Nouveaux dérivés de pipéridinyl thio indole, leurs procédés de préparation, compositions pharmaceutiques les contenant, utiles notamment comme antalgiques .
PCT/FR1994/000410 WO1994026736A1 (fr) 1993-05-18 1994-04-13 Derives de piperidinyl thio indole comme antalgiques

Publications (1)

Publication Number Publication Date
EE9400296A true EE9400296A (et) 1996-04-15

Family

ID=9447241

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9400296A EE9400296A (et) 1993-05-18 1994-11-23 Piperidinüültioindooli derivaadid, ravimvormid, aktiivne valuvaigisti, nende valmistamise meetodid

Country Status (15)

Country Link
US (1) US5317025A (OSRAM)
EP (1) EP0699195A1 (OSRAM)
JP (1) JPH09500611A (OSRAM)
CN (1) CN1124026A (OSRAM)
AU (1) AU6571594A (OSRAM)
CA (1) CA2161021A1 (OSRAM)
CZ (1) CZ304195A3 (OSRAM)
EE (1) EE9400296A (OSRAM)
FI (1) FI954931A7 (OSRAM)
FR (1) FR2705346B1 (OSRAM)
HU (1) HUT74866A (OSRAM)
MD (1) MD522G2 (OSRAM)
NZ (1) NZ265304A (OSRAM)
TW (1) TW257756B (OSRAM)
WO (1) WO1994026736A1 (OSRAM)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK139593D0 (da) * 1993-12-16 1993-12-16 Lundbeck & Co As H Compounds
JPH10503501A (ja) * 1994-08-03 1998-03-31 アスタ メディカ アクチエンゲゼルシャフト 抗喘息、抗アレルギー、抗炎症及び免疫修飾作用を有するインドール、インダゾール、ピリドピロール及びピリドピラゾール誘導体
US5521196A (en) * 1994-10-05 1996-05-28 Eli Lilly And Company 5-HT1F agonists for the treatment of migraine
PL322843A1 (en) * 1995-03-20 1998-02-16 Lilly Co Eli 5-substituted 3-91,2,3,6-tetrahydropyridin-4-yl)- and 3-9piperydin-4-4-yl0-1h-indoles nevel 5-htif natagonists
TWI328009B (en) 2003-05-21 2010-08-01 Glaxo Group Ltd Quinoline derivatives as phosphodiesterase inhibitors
JP4980928B2 (ja) * 2004-12-24 2012-07-18 プロシディオン・リミテッド Gタンパク質共役受容体(gpr116)作動薬および肥満および糖尿病治療のためのその使用
AU2006264649A1 (en) * 2005-06-30 2007-01-11 Prosidion Limited GPCR agonists
PE20081659A1 (es) * 2007-01-04 2008-10-24 Prosidion Ltd Agonistas de gpcr
AR064736A1 (es) * 2007-01-04 2009-04-22 Prosidion Ltd Agonistas de gpcr
JP2013525490A (ja) * 2010-05-06 2013-06-20 メルク・シャープ・エンド・ドーム・コーポレイション Faahのモジュレータとして有用なアザインドール誘導体
MX384804B (es) 2015-07-02 2025-03-14 Horizon Orphan Llc Analogos de cisteamina resistentes a la ado y sus usos.
CN104945305A (zh) * 2015-07-03 2015-09-30 北京石油化工学院 一种实现吲哚类化合物选择性芳巯基化的方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB925429A (en) * 1960-04-01 1963-05-08 Irwin Neisler & Co Indole derivatives
US3264311A (en) * 1963-05-02 1966-08-02 Upjohn Co Esters of 3-(aminosulfinyl) indole-2-carboxylic acids

Also Published As

Publication number Publication date
JPH09500611A (ja) 1997-01-21
NZ265304A (en) 1997-02-24
CZ304195A3 (en) 1996-03-13
MD522G2 (ro) 1997-01-31
FI954931A0 (fi) 1995-10-17
CN1124026A (zh) 1996-06-05
FR2705346A1 (fr) 1994-11-25
FR2705346B1 (fr) 1995-08-11
MD522F1 (en) 1996-04-30
CA2161021A1 (en) 1994-11-24
FI954931L (fi) 1995-11-20
HUT74866A (en) 1997-02-28
FI954931A7 (fi) 1995-11-20
US5317025A (en) 1994-05-31
EP0699195A1 (fr) 1996-03-06
TW257756B (OSRAM) 1995-09-21
AU6571594A (en) 1994-12-12
HU9503281D0 (en) 1996-01-29
WO1994026736A1 (fr) 1994-11-24

Similar Documents

Publication Publication Date Title
NO20053106D0 (no) Oral, analgesisk doseringsform med forlenget frigivelse.
FI930657A7 (fi) Menetelmä pidennetyn aktiiviaineluovutuksen omaavien annosmuotojen valmistamiseksi
KR970006279A (ko) 약제학적 활성 성분으로서의 6-디메틸아미노메틸-1-페닐-사이클로헥산 화합물
EE9700241A (et) Farmatseutiline kompositsioon transdermaalseks manustamiseks
FI943687L (fi) Uudet 11-bentsaldoksiimiestradieenijohdannaiset, menetelmät niiden valmistamiseksi ja näitä yhdisteitä sisältävät lääkeaineet
DE19681389T1 (de) Dosierungsform, umfassend Oxybutynin
FI952230L (fi) Uusi aryylipropaanijohdannainen, menetelmä sen valmistamiseksi ja sen käyttö analgeettisena aineena
NO944700D0 (no) Nye tienotiazinderivater, fremgangsmåte for fremstilling derav samt farmasöytiske preparater inneholdende forbindelsene
NO922006L (no) Farmasoeytisk preparat
NO921958D0 (no) Farmasoeytisk preparat
NO308854B1 (no) Terapeutiske forbindelser, farmasøytisk akseptable salter og formuleringer inneholdende forbindelsene, samt anvendelser derav
DE69514087D1 (de) Pharmazeutisch aktive substituierte aromatische verbindungen
NO943888D0 (no) Farmasöytisk preparat
ITRM920412A0 (it) Eteroprostanoidi, procedimento per la loro preparazione e loro impiegoterapeutico.
IS3878A (is) Imidazodiazepines efnasambönd, framleiðsla þeirraog notkun sem lyfja
ITFI930030A0 (it) Composti pirrol-amidinici, e loro sali farmaceuticamente accettabili, processi di preparazione e composizione farmaceutiche che li contengo-no.
FI942499L (fi) Indolijohdannainen, menetelmä sen valmistamiseksi ja sen lääkekäyttö
EE9400296A (et) Piperidinüültioindooli derivaadid, ravimvormid, aktiivne valuvaigisti, nende valmistamise meetodid
NO942343L (no) Farmasöytisk preparat med analgetisk aktivitet
EE9800145A (et) Fenüülamidiini derivaadid, meetodid nende valmistamiseks ja nende kasutamine arstimitena
FI951631L (fi) Substituoituja kynureniinejä, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä
NO20002439L (no) Nye orale doseringsformer for carvediol
FI933544A7 (fi) Tiadiatsiinikarboksamidijohdannaiset, menetelmät niiden valmistamiseks i ja lääkkeet
NO973610D0 (no) Nytt farmasöytisk preparat
FI964277A7 (fi) O-asyyli-4-fenyyli-sykloalkanolit, niiden suolat, näitä yhdisteitä sisältävät lääkeaineet sekä niiden käyttö sekä menetelmä niiden valmistamiseksi