EE04117B1 - Karboksüasendatud tsüklilised karboksamiidi derivaadid, nende valmistamise meetod ja kasutamine - Google Patents

Karboksüasendatud tsüklilised karboksamiidi derivaadid, nende valmistamise meetod ja kasutamine

Info

Publication number
EE04117B1
EE04117B1 EEP199900254A EE9900254A EE04117B1 EE 04117 B1 EE04117 B1 EE 04117B1 EE P199900254 A EEP199900254 A EE P199900254A EE 9900254 A EE9900254 A EE 9900254A EE 04117 B1 EE04117 B1 EE 04117B1
Authority
EE
Estonia
Prior art keywords
carboxy
preparation
substituted cyclic
carboxamide derivatives
cyclic carboxamide
Prior art date
Application number
EEP199900254A
Other languages
English (en)
Other versions
EE9900254A (et
Inventor
P. Burkholder Timothy
D. Maynard George
M. Kudlacz Elizabeth
Original Assignee
Hoechst Marion Roussel, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/971,891 external-priority patent/US5977139A/en
Application filed by Hoechst Marion Roussel, Inc. filed Critical Hoechst Marion Roussel, Inc.
Publication of EE9900254A publication Critical patent/EE9900254A/et
Publication of EE04117B1 publication Critical patent/EE04117B1/et

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/14—Antitussive agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pyrrole Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
EEP199900254A 1996-12-19 1997-11-21 Karboksüasendatud tsüklilised karboksamiidi derivaadid, nende valmistamise meetod ja kasutamine EE04117B1 (et)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US79415796A 1996-12-19 1996-12-19
US08/971,891 US5977139A (en) 1996-12-15 1997-11-17 Carboxysubstituted cyclic carboxamide derivatives
PCT/US1997/021586 WO1998027085A1 (en) 1996-12-19 1997-11-21 Novel carboxy substituted cyclic carboxamide derivatives

Publications (2)

Publication Number Publication Date
EE9900254A EE9900254A (et) 1999-12-15
EE04117B1 true EE04117B1 (et) 2003-08-15

Family

ID=27121482

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP199900254A EE04117B1 (et) 1996-12-19 1997-11-21 Karboksüasendatud tsüklilised karboksamiidi derivaadid, nende valmistamise meetod ja kasutamine

Country Status (27)

Country Link
EP (1) EP0946545B1 (et)
JP (1) JP4195513B2 (et)
KR (1) KR100468552B1 (et)
CN (1) CN1098259C (et)
AR (1) AR009666A1 (et)
AT (1) ATE205200T1 (et)
AU (1) AU718984B2 (et)
BR (1) BR9714156A (et)
CA (1) CA2275602C (et)
CL (1) CL2003002750A1 (et)
DE (1) DE69706564T2 (et)
DK (1) DK0946545T3 (et)
EE (1) EE04117B1 (et)
ES (1) ES2162686T3 (et)
HK (1) HK1020571A1 (et)
IL (1) IL130222A0 (et)
NO (1) NO318196B1 (et)
NZ (1) NZ335883A (et)
OA (1) OA11070A (et)
PL (1) PL189777B1 (et)
PT (1) PT946545E (et)
RU (1) RU2199535C2 (et)
SK (1) SK82799A3 (et)
TR (1) TR199901395T2 (et)
TW (1) TW544452B (et)
UA (1) UA58529C2 (et)
WO (1) WO1998027085A1 (et)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999003832A1 (en) * 1997-07-14 1999-01-28 Phytera Symbion Aps Piperidine oligomers and combinatorial libraries thereof
ID29137A (id) * 1998-07-27 2001-08-02 Schering Corp Ligan-ligan afinitas tinggi untuk reseptor nosiseptin orl-1
WO2001029027A1 (fr) * 1999-10-22 2001-04-26 Sankyo Company, Limited Dérivés de 2-alcoxybenzène
WO2002022582A2 (en) * 2000-09-14 2002-03-21 Ortho-Mcneil Pharmaceutical, Inc. Solid salt forms of n-[2-[4-[2-(1-methylethoxy)phenyl]-1-piperazinyl]ethyl]-2-oxo-1-piperidineacetamide
GB0217447D0 (en) * 2002-07-29 2002-09-04 Betts John A Personal deodorant
EP2385040A1 (en) 2003-03-14 2011-11-09 ONO Pharmaceutical Co., Ltd. Nitrogen-containing heterocyclic derivatives and drugs containing the same as the active ingredient
KR101231466B1 (ko) 2004-09-13 2013-02-07 오노 야꾸힝 고교 가부시키가이샤 질소 함유 복소환 유도체 및 이들을 유효 성분으로 하는약제
CN101443322A (zh) 2006-03-10 2009-05-27 小野药品工业株式会社 含氮杂环衍生物及含有该衍生物作为活性成分的药物

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0696280B1 (en) * 1993-05-06 1997-09-24 Merrell Pharmaceuticals Inc. Substituted pyrrolidin-3-yl-alkyl-piperidines useful as tachykinin antagonists

Also Published As

Publication number Publication date
CA2275602A1 (en) 1998-06-25
NO993012L (no) 1999-08-18
CN1098259C (zh) 2003-01-08
RU2199535C2 (ru) 2003-02-27
EP0946545A1 (en) 1999-10-06
KR100468552B1 (ko) 2005-01-29
HK1020571A1 (en) 2000-05-12
CN1240443A (zh) 2000-01-05
TW544452B (en) 2003-08-01
OA11070A (en) 2002-11-15
UA58529C2 (uk) 2003-08-15
DE69706564D1 (de) 2001-10-11
DE69706564T2 (de) 2002-07-11
AU718984B2 (en) 2000-05-04
EE9900254A (et) 1999-12-15
TR199901395T2 (xx) 1999-11-22
ATE205200T1 (de) 2001-09-15
CL2003002750A1 (es) 2005-04-22
EP0946545B1 (en) 2001-09-05
IL130222A0 (en) 2000-06-01
PL334077A1 (en) 2000-01-31
AR009666A1 (es) 2000-04-26
SK82799A3 (en) 2001-09-11
NZ335883A (en) 2001-07-27
NO993012D0 (no) 1999-06-18
WO1998027085A1 (en) 1998-06-25
NO318196B1 (no) 2005-02-14
DK0946545T3 (da) 2001-11-19
PT946545E (pt) 2002-02-28
PL189777B1 (pl) 2005-09-30
KR20000057667A (ko) 2000-09-25
JP4195513B2 (ja) 2008-12-10
AU5362798A (en) 1998-07-15
BR9714156A (pt) 2000-02-08
JP2002512596A (ja) 2002-04-23
ES2162686T3 (es) 2002-01-01
CA2275602C (en) 2003-07-22

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Legal Events

Date Code Title Description
KB4A Valid patent at the end of a year

Effective date: 20031231

HC1A Change of owner name
KB4A Valid patent at the end of a year

Effective date: 20041231

KB4A Valid patent at the end of a year

Effective date: 20051231

MM4A Lapsed by not paying the annual fees

Effective date: 20051121