ECSP12011651A - Derivados de 5-fluoro-2-oxopirimidina-1(2h)-carboxilato - Google Patents

Derivados de 5-fluoro-2-oxopirimidina-1(2h)-carboxilato

Info

Publication number
ECSP12011651A
ECSP12011651A ECSP12011651A ECSP12011651A EC SP12011651 A ECSP12011651 A EC SP12011651A EC SP12011651 A ECSP12011651 A EC SP12011651A EC SP12011651 A ECSP12011651 A EC SP12011651A
Authority
EC
Ecuador
Prior art keywords
fluoro
derivatives
oxopirimidina
carboxylate
oxopyrimidine
Prior art date
Application number
Other languages
English (en)
Spanish (es)
Inventor
Timothy Martin
Mark Andrew Pobanz
Timothy Boebel
Kristy Bryan
Beth Lorsbach
W Owen
Jeffery Webster
Chenglin Yao
Scott Thornburgh
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535293&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP12011651(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of ECSP12011651A publication Critical patent/ECSP12011651A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/16Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/20Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D239/22Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
ECSP12011651 2009-08-07 2012-02-07 Derivados de 5-fluoro-2-oxopirimidina-1(2h)-carboxilato ECSP12011651A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23223209P 2009-08-07 2009-08-07

Publications (1)

Publication Number Publication Date
ECSP12011651A true ECSP12011651A (es) 2012-03-30

Family

ID=43535293

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP12011651 ECSP12011651A (es) 2009-08-07 2012-02-07 Derivados de 5-fluoro-2-oxopirimidina-1(2h)-carboxilato

Country Status (28)

Country Link
US (1) US8318758B2 (forum.php)
EP (1) EP2462133B1 (forum.php)
JP (1) JP5818791B2 (forum.php)
KR (1) KR101792286B1 (forum.php)
CN (1) CN102548979B (forum.php)
AU (1) AU2010279408B2 (forum.php)
BR (1) BR112012002807B1 (forum.php)
CA (1) CA2769251C (forum.php)
CL (1) CL2012000314A1 (forum.php)
CO (1) CO6491089A2 (forum.php)
CR (1) CR20120033A (forum.php)
DK (1) DK2462133T3 (forum.php)
EA (1) EA022930B1 (forum.php)
EC (1) ECSP12011651A (forum.php)
ES (1) ES2506169T3 (forum.php)
HN (1) HN2012000261A (forum.php)
IL (1) IL217954A (forum.php)
IN (1) IN2012DN00695A (forum.php)
MX (1) MX2012001623A (forum.php)
NI (1) NI201200019A (forum.php)
NZ (1) NZ597638A (forum.php)
PE (1) PE20120689A1 (forum.php)
PL (1) PL2462133T3 (forum.php)
PT (1) PT2462133E (forum.php)
RS (1) RS53658B1 (forum.php)
UA (1) UA106086C2 (forum.php)
WO (1) WO2011017544A1 (forum.php)
ZA (1) ZA201305992B (forum.php)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5784603B2 (ja) * 2009-08-07 2015-09-24 ダウ アグロサイエンシィズ エルエルシー N1−スルホニル−5−フルオロピリミジノン誘導体
CN104884062B (zh) 2012-12-28 2018-11-06 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-甲酰胺衍生物
EP3689142A1 (en) * 2012-12-28 2020-08-05 Adama Makhteshim Ltd. 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
AU2013370493B2 (en) * 2012-12-28 2017-08-17 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxylate derivatives
NZ749557A (en) 2012-12-31 2020-01-31 Adama Makhteshim Ltd 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
CN111362881A (zh) 2013-12-31 2020-07-03 阿达玛马克西姆股份有限公司 一种化合物及其制备方法
PT3096619T (pt) 2013-12-31 2025-09-11 Adama Makhteshim Ltd Misturas fungicidas sinérgicas para controlo de fungos em cereais
WO2016040193A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
KR20180080262A (ko) 2015-11-06 2018-07-11 사뮤메드, 엘엘씨 골관절염의 치료
JP7010851B2 (ja) 2016-06-01 2022-02-10 バイオスプライス セラピューティクス インコーポレイテッド N-(5-(3-(7-(3-フルオロフェニル)-3H-イミダゾ[4,5-c]ピリジン-2-イル)-1H-インダゾール-5-イル)ピリジン-3-イル)-3-メチルブタンアミドを調製するための方法
IL271950B2 (en) 2017-07-17 2024-06-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one
BR112021008755A2 (pt) 2018-11-05 2021-08-10 Adama Makhteshim Ltd. misturas e composições contendo 5-fluoro-4-imino-3- metil-1-tosil-3,4-dihidropirimidina-2-ona, e métodos de uso.
AR120035A1 (es) 2019-09-23 2022-01-26 Adama Makhteshim Ltd Proceso para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
JP2000506171A (ja) * 1996-03-11 2000-05-23 ノバルティス アクチェンゲゼルシャフト 農薬としてのピリミジン−4−オン誘導体
WO2004037159A2 (en) * 2002-10-23 2004-05-06 Obetherapy Biotechnology Compounds, compositions and methods for modulating fat metabolism
AU2008249329C1 (en) * 2007-04-27 2013-07-04 Daiichi Sankyo Company Limited Nitrogenated aromatic 6-membered ring derivative, and pharmaceutical agent comprising the same
EP2647287A1 (en) 2008-08-01 2013-10-09 Dow AgroSciences LLC Use of 5-fluorocytosine and its derivatives as fungicides

Also Published As

Publication number Publication date
IL217954A0 (en) 2012-03-29
JP5818791B2 (ja) 2015-11-18
PL2462133T3 (pl) 2015-03-31
DK2462133T3 (en) 2015-01-05
CR20120033A (es) 2012-03-22
CO6491089A2 (es) 2012-07-31
EP2462133A1 (en) 2012-06-13
KR20120043069A (ko) 2012-05-03
US8318758B2 (en) 2012-11-27
BR112012002807B1 (pt) 2018-07-10
IN2012DN00695A (forum.php) 2015-06-19
CA2769251C (en) 2018-05-15
EA022930B1 (ru) 2016-03-31
WO2011017544A1 (en) 2011-02-10
NI201200019A (es) 2012-05-22
CN102548979A (zh) 2012-07-04
UA106086C2 (uk) 2014-07-25
RS53658B1 (sr) 2015-04-30
EA201270255A1 (ru) 2012-07-30
KR101792286B1 (ko) 2017-10-31
HK1172892A1 (en) 2013-05-03
PT2462133E (pt) 2014-12-26
BR112012002807A2 (pt) 2015-10-13
CA2769251A1 (en) 2011-02-10
US20110034491A1 (en) 2011-02-10
ES2506169T3 (es) 2014-10-13
CL2012000314A1 (es) 2012-10-05
ZA201305992B (en) 2014-10-29
HN2012000261A (es) 2015-01-05
AU2010279408A1 (en) 2012-02-09
BR112012002807A8 (pt) 2017-07-11
EP2462133B1 (en) 2014-09-24
JP2013501726A (ja) 2013-01-17
NZ597638A (en) 2014-06-27
PE20120689A1 (es) 2012-06-06
EP2462133A4 (en) 2013-01-16
CN102548979B (zh) 2015-05-13
IL217954A (en) 2016-02-29
MX2012001623A (es) 2012-04-11
AU2010279408B2 (en) 2015-09-10

Similar Documents

Publication Publication Date Title
ECSP12011651A (es) Derivados de 5-fluoro-2-oxopirimidina-1(2h)-carboxilato
ECSP12011654A (es) Derivados de 5-fluoropirimidinona
NI201200020A (es) Derivados de n1 - sulfonil - 5 - fluoropirimidinona
CO6592042A2 (es) Derivados de n3-sustituido -n1-sulfonil-5-fluorpirimidinona
ECSP12011653A (es) Derivados de n1-acil-5-fluoropirimidinona
CR11569A (es) Derivados de pirimidina 5-fluoro como fungicidas
ECSP12011652A (es) Derivados de 5-fluoro-2-oxopirimidinona-1 (2h)-carboxamida substituida-n1
ECSP14013251A (es) Derivados de 5-flúor-4-imino-3-(sustituido)-3,4-dihidropirimidin-2(1h)ona
CR20110044A (es) Uso de 5-fluorocitosina como un fungicida
CR20120158A (es) Compuestos de diòxido de iminotiadiazina como inhibidores de bace, composiciones y su uso.
MX386852B (es) Ciertas triazolopiridinas y triazolopirazinas, composiciones de estas y sus metodos de uso.
UY32292A (es) Agonistas de s1p1 y métodos de preparación y uso
UY32553A (es) Nuevos derivados de la pirrolidinadiona espiroheterocíclicos 3-sustituidos
SV2009003429A (es) Derivados de 7-alquinil-1,8-naftiridonas, su preparacion y su aplicacion en terapeutica
UY32667A (es) Nuevos derivados de furano espiroheterocíclico y tiofuranodiona
ECSP12012047A (es) Derivados de 2-aldoximino-5-fluoropirimidina
DOP2012000146A (es) Nuevos derivados (heterociclo-tetrahidro-piridin)-(piperazinil)-1-alcanona y (heterociclo-dihidro-pirrolidin)-(piperazinil)-1-alcanona y su utilizacion como inhibidores de p75
UY32772A (es) Etilamidas de benzotienilo novedosas y sus usos como microbicidas
GT201400024A (es) Derivados de n-(5-fluoro-2-((4-metilbencil)oxi)pirimidin-4-il) benzamida