EA201990835A3 - Режимы дозирования антипрогестинов - Google Patents

Режимы дозирования антипрогестинов

Info

Publication number
EA201990835A3
EA201990835A3 EA201990835A EA201990835A EA201990835A3 EA 201990835 A3 EA201990835 A3 EA 201990835A3 EA 201990835 A EA201990835 A EA 201990835A EA 201990835 A EA201990835 A EA 201990835A EA 201990835 A3 EA201990835 A3 EA 201990835A3
Authority
EA
Eurasian Patent Office
Prior art keywords
estrogen
endometriosis
present
women
compositions
Prior art date
Application number
EA201990835A
Other languages
English (en)
Russian (ru)
Other versions
EA201990835A2 (ru
Inventor
Джозеф С. Подольски
Original Assignee
Репрос Терапьютикс Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Репрос Терапьютикс Инк. filed Critical Репрос Терапьютикс Инк.
Publication of EA201990835A2 publication Critical patent/EA201990835A2/ru
Publication of EA201990835A3 publication Critical patent/EA201990835A3/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/04—Drugs for genital or sexual disorders; Contraceptives for inducing labour or abortion; Uterotonics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32—Antioestrogens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/36—Antigestagens

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
EA201990835A 2008-04-28 2009-04-27 Режимы дозирования антипрогестинов EA201990835A3 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US4847208P 2008-04-28 2008-04-28

Publications (2)

Publication Number Publication Date
EA201990835A2 EA201990835A2 (ru) 2019-08-30
EA201990835A3 true EA201990835A3 (ru) 2019-12-30

Family

ID=40751037

Family Applications (3)

Application Number Title Priority Date Filing Date
EA201990835A EA201990835A3 (ru) 2008-04-28 2009-04-27 Режимы дозирования антипрогестинов
EA201071249A EA201071249A1 (ru) 2008-04-28 2009-04-27 Режимы дозирования антипрогестинов
EA201401347A EA032646B1 (ru) 2008-04-28 2009-04-27 Режимы дозирования антипрогестинов

Family Applications After (2)

Application Number Title Priority Date Filing Date
EA201071249A EA201071249A1 (ru) 2008-04-28 2009-04-27 Режимы дозирования антипрогестинов
EA201401347A EA032646B1 (ru) 2008-04-28 2009-04-27 Режимы дозирования антипрогестинов

Country Status (24)

Country Link
US (2) US8426394B2 (cg-RX-API-DMAC10.html)
EP (1) EP2293797B1 (cg-RX-API-DMAC10.html)
JP (1) JP5791499B2 (cg-RX-API-DMAC10.html)
KR (2) KR20130059442A (cg-RX-API-DMAC10.html)
CN (2) CN102014923A (cg-RX-API-DMAC10.html)
AR (1) AR071516A1 (cg-RX-API-DMAC10.html)
AU (1) AU2009241355B2 (cg-RX-API-DMAC10.html)
BR (1) BRPI0911563A2 (cg-RX-API-DMAC10.html)
CA (1) CA2722753C (cg-RX-API-DMAC10.html)
CL (1) CL2009001010A1 (cg-RX-API-DMAC10.html)
DK (1) DK2293797T3 (cg-RX-API-DMAC10.html)
EA (3) EA201990835A3 (cg-RX-API-DMAC10.html)
ES (1) ES2561810T3 (cg-RX-API-DMAC10.html)
IL (1) IL208844A0 (cg-RX-API-DMAC10.html)
ME (1) ME01123B (cg-RX-API-DMAC10.html)
MX (1) MX2010011272A (cg-RX-API-DMAC10.html)
MY (1) MY161059A (cg-RX-API-DMAC10.html)
NI (1) NI201000183A (cg-RX-API-DMAC10.html)
NZ (1) NZ589533A (cg-RX-API-DMAC10.html)
SG (1) SG10201408483QA (cg-RX-API-DMAC10.html)
TW (1) TWI477276B (cg-RX-API-DMAC10.html)
UA (1) UA102849C2 (cg-RX-API-DMAC10.html)
WO (1) WO2009134718A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA201007529B (cg-RX-API-DMAC10.html)

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US10806740B2 (en) 2012-06-18 2020-10-20 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
US10806697B2 (en) 2012-12-21 2020-10-20 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
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US11246875B2 (en) 2012-12-21 2022-02-15 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
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US10328087B2 (en) 2015-07-23 2019-06-25 Therapeuticsmd, Inc. Formulations for solubilizing hormones
KR20180126582A (ko) 2016-04-01 2018-11-27 쎄러퓨틱스엠디, 인코퍼레이티드 스테로이드 호르몬 약제학적 조성물
WO2017173044A1 (en) 2016-04-01 2017-10-05 Therapeuticsmd Inc. Steroid hormone compositions in medium chain oils
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Also Published As

Publication number Publication date
ES2561810T3 (es) 2016-03-01
ZA201007529B (en) 2011-07-27
UA102849C2 (ru) 2013-08-27
TW200950786A (en) 2009-12-16
US8735381B2 (en) 2014-05-27
US20130289008A1 (en) 2013-10-31
IL208844A0 (en) 2011-01-31
CN102014923A (zh) 2011-04-13
WO2009134718A8 (en) 2010-09-23
CA2722753C (en) 2018-07-03
AR071516A1 (es) 2010-06-23
JP5791499B2 (ja) 2015-10-07
EP2293797A1 (en) 2011-03-16
KR20130059442A (ko) 2013-06-05
EA032646B1 (ru) 2019-06-28
EA201071249A1 (ru) 2011-08-30
TWI477276B (zh) 2015-03-21
NI201000183A (es) 2012-06-06
MX2010011272A (es) 2010-12-21
MY161059A (en) 2017-04-14
SG10201408483QA (en) 2015-02-27
US20110046098A1 (en) 2011-02-24
DK2293797T3 (en) 2016-01-11
EA201990835A2 (ru) 2019-08-30
CL2009001010A1 (es) 2009-06-19
CN105616427A (zh) 2016-06-01
CA2722753A1 (en) 2009-11-05
ME01123B (me) 2013-03-20
JP2011518845A (ja) 2011-06-30
NZ589533A (en) 2012-06-29
BRPI0911563A2 (pt) 2016-07-12
EP2293797B1 (en) 2015-11-11
EA201401347A1 (ru) 2015-07-30
KR20110014162A (ko) 2011-02-10
AU2009241355A1 (en) 2009-11-05
US8426394B2 (en) 2013-04-23
WO2009134718A1 (en) 2009-11-05
AU2009241355B2 (en) 2013-11-14

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