EA201592020A1 - Новая композиция для неалкогольной жировой болезни печени (нажбп) - Google Patents

Новая композиция для неалкогольной жировой болезни печени (нажбп)

Info

Publication number
EA201592020A1
EA201592020A1 EA201592020A EA201592020A EA201592020A1 EA 201592020 A1 EA201592020 A1 EA 201592020A1 EA 201592020 A EA201592020 A EA 201592020A EA 201592020 A EA201592020 A EA 201592020A EA 201592020 A1 EA201592020 A1 EA 201592020A1
Authority
EA
Eurasian Patent Office
Prior art keywords
nafld
liver disease
fatial
nonalcoholic
new composition
Prior art date
Application number
EA201592020A
Other languages
English (en)
Inventor
Панкадж Пател
Раджендракумар Харипрасад Джани
Original Assignee
Кадила Хелзкэр Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Кадила Хелзкэр Лимитед filed Critical Кадила Хелзкэр Лимитед
Publication of EA201592020A1 publication Critical patent/EA201592020A1/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)

Abstract

Настоящее изобретение относится к соединению формулы (I) или его фармацевтической приемлемой форме, в котором R имеет значения, указанные в настоящем документе. Кроме того, настоящее изобретение относится к композиции, включающей эффективное терапевтическое количество соединения формулы (I), и способу применения соединений для лечения или профилактики расстройства, такого как неалкогольная жировая болезнь печени (НАЖБП), включающая ожирение печени (стеатоз), неалкогольный стеатогепатит (НАСГ) и цирроз печени (прогрессирующее рубцевание печени).
EA201592020A 2013-04-22 2013-06-25 Новая композиция для неалкогольной жировой болезни печени (нажбп) EA201592020A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/IN2013/000391 WO2014174524A1 (en) 2013-04-22 2013-06-25 A novel composition for nonalcoholic fatty liver disease (nafld)
IN1468MU2013 IN2013MU01468A (ru) 2013-04-22 2013-06-25

Publications (1)

Publication Number Publication Date
EA201592020A1 true EA201592020A1 (ru) 2016-05-31

Family

ID=49253372

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201592020A EA201592020A1 (ru) 2013-04-22 2013-06-25 Новая композиция для неалкогольной жировой болезни печени (нажбп)

Country Status (21)

Country Link
US (3) US20160166539A1 (ru)
EP (1) EP2988736A1 (ru)
JP (1) JP6246895B2 (ru)
KR (1) KR101617812B1 (ru)
CN (1) CN105377246B (ru)
AP (1) AP2015008674A0 (ru)
AU (1) AU2013387996B2 (ru)
BR (1) BR112015020600A2 (ru)
CA (1) CA2900435C (ru)
EA (1) EA201592020A1 (ru)
GE (1) GEP201706663B (ru)
HK (1) HK1214968A1 (ru)
IL (2) IL240183A (ru)
IN (1) IN2013MU01468A (ru)
MA (1) MA38385A1 (ru)
MX (1) MX346943B (ru)
MY (1) MY180160A (ru)
PH (1) PH12015501795A1 (ru)
SG (1) SG11201506218UA (ru)
UA (1) UA114360C2 (ru)
WO (1) WO2014174524A1 (ru)

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Also Published As

Publication number Publication date
KR101617812B1 (ko) 2016-05-03
US20160166539A1 (en) 2016-06-16
BR112015020600A2 (pt) 2017-07-18
US9814697B2 (en) 2017-11-14
IL240183A (en) 2016-08-31
US20170087127A1 (en) 2017-03-30
SG11201506218UA (en) 2015-09-29
WO2014174524A8 (en) 2015-10-01
UA114360C2 (uk) 2017-05-25
GEP201706663B (en) 2017-05-10
CN105377246A (zh) 2016-03-02
US20180185330A1 (en) 2018-07-05
KR20150118990A (ko) 2015-10-23
AP2015008674A0 (en) 2015-08-31
AU2013387996B2 (en) 2015-12-10
IN2013MU01468A (ru) 2015-04-17
PH12015501795A1 (en) 2015-11-09
MY180160A (en) 2020-11-23
HK1214968A1 (zh) 2016-08-12
CA2900435A1 (en) 2014-10-30
CA2900435C (en) 2017-02-14
JP6246895B2 (ja) 2017-12-13
IL247231A (en) 2017-03-30
IL240183A0 (en) 2015-09-24
EP2988736A1 (en) 2016-03-02
MX2015010769A (es) 2015-11-26
JP2016515608A (ja) 2016-05-30
MA38385A1 (fr) 2017-09-29
CN105377246B (zh) 2018-03-20
WO2014174524A1 (en) 2014-10-30
MX346943B (es) 2017-04-06
AU2013387996A1 (en) 2015-09-24

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