EA201591230A1 - Композиция диклофенака - Google Patents
Композиция диклофенакаInfo
- Publication number
- EA201591230A1 EA201591230A1 EA201591230A EA201591230A EA201591230A1 EA 201591230 A1 EA201591230 A1 EA 201591230A1 EA 201591230 A EA201591230 A EA 201591230A EA 201591230 A EA201591230 A EA 201591230A EA 201591230 A1 EA201591230 A1 EA 201591230A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- composition
- diclofenac
- present
- relates
- administration
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
- A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
Abstract
Настоящее изобретение относится к композиции, содержащей диклофенак и его соли, где диклофенак или его соли присутствуют в количестве 25-200 мг. Композиция является применимой для парентерального введения посредством внутримышечного, внутривенного пути введения; а также для перорального, кожного, подкожного, назального введения в виде глазных капель, в виде ректальных суппозиториев, вагинальных суппозиториев, для внутрисуставной и ушной доставки. Настоящее изобретение относится также к композициям, содержащим комбинацию диклофенака и других лекарственных средств. Изобретение далее относится к способу получения указанной композиции.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN3704MU2012 | 2012-12-28 | ||
PCT/IN2013/000805 WO2014102824A1 (en) | 2012-12-28 | 2013-12-27 | Diclofenac composition |
Publications (2)
Publication Number | Publication Date |
---|---|
EA201591230A1 true EA201591230A1 (ru) | 2015-11-30 |
EA035079B1 EA035079B1 (ru) | 2020-04-24 |
Family
ID=54198802
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201591230A EA035079B1 (ru) | 2012-12-28 | 2013-12-27 | Композиция диклофенака |
Country Status (25)
Country | Link |
---|---|
US (1) | US20140187635A1 (ru) |
EP (1) | EP2938325B8 (ru) |
JP (1) | JP6117939B2 (ru) |
KR (1) | KR101730284B1 (ru) |
CN (1) | CN104968331A (ru) |
AP (1) | AP2015008534A0 (ru) |
AU (1) | AU2013368849B2 (ru) |
BR (1) | BR112015015699B1 (ru) |
CL (1) | CL2015001869A1 (ru) |
EA (1) | EA035079B1 (ru) |
ES (1) | ES2721400T3 (ru) |
HK (1) | HK1211858A1 (ru) |
HU (1) | HUE045030T2 (ru) |
IL (1) | IL239395A0 (ru) |
MA (1) | MA38292A1 (ru) |
MX (1) | MX365375B (ru) |
MY (1) | MY184886A (ru) |
PE (1) | PE20151208A1 (ru) |
PH (1) | PH12015501479B1 (ru) |
SG (1) | SG11201504577UA (ru) |
SI (1) | SI2938325T1 (ru) |
TR (1) | TR201905806T4 (ru) |
UA (1) | UA114123C2 (ru) |
WO (1) | WO2014102824A1 (ru) |
ZA (1) | ZA201504258B (ru) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR101524473B1 (ko) * | 2014-12-22 | 2015-06-02 | 주식회사 한국팜비오 | 주사제 조성물 |
WO2016170401A1 (en) * | 2015-04-20 | 2016-10-27 | Umedica Laboratories Pvt. Ltd | Novel injectable composition of diclofenac sodium |
US11110073B2 (en) | 2017-03-24 | 2021-09-07 | Cadila Healthcare Limited | Storage stable aqueous injectable solution comprising diclofenac |
GB201720992D0 (en) * | 2017-12-15 | 2018-01-31 | Hooper Mark | A medical use |
GR1009729B (el) * | 2018-08-02 | 2020-05-15 | Win Medica Φαρμακευτικη Ανωνυμη Εταιρεια | Σταθερος ενεσιμος συνδυασμος |
ES2964698T3 (es) * | 2018-11-16 | 2024-04-09 | Seikagaku Kogyo Co Ltd | Composición farmacéutica |
US20220280463A1 (en) | 2019-09-09 | 2022-09-08 | Ftf Pharma Private Limited | Pharmaceutical formulations comprising diclofenac |
US11707443B2 (en) | 2019-09-26 | 2023-07-25 | Rk Pharma Inc. | Storage stable aqueous parenteral solutions comprising diclofenac |
WO2021144476A1 (en) * | 2020-02-18 | 2021-07-22 | Novo Nordisk A/S | Pharmaceutical formulations |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3324193A1 (de) | 1983-07-05 | 1985-01-17 | Troponwerke Gmbh & Co Kg | Depot-antiphlogistika |
DE3446873A1 (de) | 1984-12-21 | 1986-07-10 | Merckle Gmbh | Fluessige diclofenac-zubereitungen |
US5283067A (en) * | 1987-01-30 | 1994-02-01 | Ciba-Geigy Corporation | Parenteral suspensions |
WO1993000895A1 (en) * | 1991-07-04 | 1993-01-21 | Taisho Pharmaceutical Co., Ltd. | Analgesic |
US5389681A (en) | 1992-10-22 | 1995-02-14 | Ciba-Geigy Corporation | Parenteral solutions for diclofenac salts |
ZA949182B (en) | 1993-12-02 | 1995-07-26 | South African Druggists Ltd | Pharmaceutical composition |
JP4542743B2 (ja) * | 2002-12-26 | 2010-09-15 | Kdl株式会社 | ピリドン誘導体の溶液状医薬組成物 |
EP1605900A4 (en) * | 2003-03-26 | 2007-10-17 | Becton Dickinson Co | USE OF BENZYL ALCOHOL AND OTHER PHENOLIC PRESERVATIVE SUBSTANCES TO REDUCE PAIN IN INTRADERMAL INJECTION |
US20050137164A1 (en) * | 2003-09-22 | 2005-06-23 | Moshe Arkin | Diclofenac compositions for the treatment of skin disorders |
ES2287658T3 (es) | 2004-03-10 | 2007-12-16 | Shimoda Biotech (Pty) Ltd | Composiciones inyectables estables de diclofenac. |
US20050214230A1 (en) * | 2004-03-23 | 2005-09-29 | J. B. Chemicals & Pharmaceuticals Ltd. | Novel stomatological gel |
WO2006095363A2 (en) * | 2005-02-01 | 2006-09-14 | Troikaa Pharmaceuticals Ltd | Injectable preparations of diclofenic and its pharmaceutically acceptable salts |
CN101217939A (zh) * | 2005-05-27 | 2008-07-09 | 灵药生物技术有限公司 | 可注射组合物及制备这类组合物的方法 |
CN102227211A (zh) | 2008-11-28 | 2011-10-26 | 先进控股有限公司 | 包含双氯芬酸和羟基脂肪酸聚氧化烯烃酯的药物配制剂 |
-
2013
- 2013-12-24 US US14/140,109 patent/US20140187635A1/en not_active Abandoned
- 2013-12-27 PE PE2015001194A patent/PE20151208A1/es not_active Application Discontinuation
- 2013-12-27 CN CN201380068194.2A patent/CN104968331A/zh active Pending
- 2013-12-27 AU AU2013368849A patent/AU2013368849B2/en active Active
- 2013-12-27 SI SI201331424T patent/SI2938325T1/sl unknown
- 2013-12-27 TR TR2019/05806T patent/TR201905806T4/tr unknown
- 2013-12-27 KR KR1020157017781A patent/KR101730284B1/ko active IP Right Grant
- 2013-12-27 WO PCT/IN2013/000805 patent/WO2014102824A1/en active Application Filing
- 2013-12-27 HU HUE13830158A patent/HUE045030T2/hu unknown
- 2013-12-27 MA MA38292A patent/MA38292A1/fr unknown
- 2013-12-27 UA UAA201506371A patent/UA114123C2/uk unknown
- 2013-12-27 MY MYPI2015001527A patent/MY184886A/en unknown
- 2013-12-27 MX MX2015008369A patent/MX365375B/es active IP Right Grant
- 2013-12-27 BR BR112015015699-1A patent/BR112015015699B1/pt active IP Right Grant
- 2013-12-27 EA EA201591230A patent/EA035079B1/ru not_active IP Right Cessation
- 2013-12-27 SG SG11201504577UA patent/SG11201504577UA/en unknown
- 2013-12-27 AP AP2015008534A patent/AP2015008534A0/xx unknown
- 2013-12-27 ES ES13830158T patent/ES2721400T3/es active Active
- 2013-12-27 JP JP2015550212A patent/JP6117939B2/ja active Active
- 2013-12-27 EP EP13830158.5A patent/EP2938325B8/en active Active
-
2015
- 2015-06-11 ZA ZA2015/04258A patent/ZA201504258B/en unknown
- 2015-06-14 IL IL239395A patent/IL239395A0/en unknown
- 2015-06-26 PH PH12015501479A patent/PH12015501479B1/en unknown
- 2015-06-26 CL CL2015001869A patent/CL2015001869A1/es unknown
- 2015-12-30 HK HK15112837.5A patent/HK1211858A1/xx unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG TJ TM |