EA201591127A1 - Бициклические пиридинилпиразолы - Google Patents

Бициклические пиридинилпиразолы

Info

Publication number
EA201591127A1
EA201591127A1 EA201591127A EA201591127A EA201591127A1 EA 201591127 A1 EA201591127 A1 EA 201591127A1 EA 201591127 A EA201591127 A EA 201591127A EA 201591127 A EA201591127 A EA 201591127A EA 201591127 A1 EA201591127 A1 EA 201591127A1
Authority
EA
Eurasian Patent Office
Prior art keywords
piridinylpirazoly
bicyclic
formula
well
protection
Prior art date
Application number
EA201591127A
Other languages
English (en)
Inventor
Амос Маттес
Хендрик Хельмке
Штефан Хиллебранд
Горка Перис
Александер Зудау
Ларс Родефельд
Штефан Гаугер
Юрген Бентинг
Петер Дамен
Рут Майсснер
Ульрике Вахендорфф-Нойманн
Хироюки Хадано
Original Assignee
Байер Интеллектуэль Проперти Гмбх
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Байер Интеллектуэль Проперти Гмбх filed Critical Байер Интеллектуэль Проперти Гмбх
Publication of EA201591127A1 publication Critical patent/EA201591127A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Abstract

В изобретении описаны бициклические пиридинилпиразолы формулы (I)в которой символы имеют значения, приведенные в описании, а также их агрохимически действующие соли и их применение для борьбы с нежелательными микроорганизмами при защите растений и защите материалов и для уменьшения содержания микотоксинов в растениях и частях растений, а также способ получения соединений формулы (I).
EA201591127A 2010-04-07 2011-04-04 Бициклические пиридинилпиразолы EA201591127A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32170410P 2010-04-07 2010-04-07
EP10159210 2010-04-07

Publications (1)

Publication Number Publication Date
EA201591127A1 true EA201591127A1 (ru) 2015-09-30

Family

ID=42667988

Family Applications (2)

Application Number Title Priority Date Filing Date
EA201291007A EA023272B1 (ru) 2010-04-07 2011-04-04 Бициклические пиридинилпиразолы
EA201591127A EA201591127A1 (ru) 2010-04-07 2011-04-04 Бициклические пиридинилпиразолы

Family Applications Before (1)

Application Number Title Priority Date Filing Date
EA201291007A EA023272B1 (ru) 2010-04-07 2011-04-04 Бициклические пиридинилпиразолы

Country Status (11)

Country Link
US (1) US8507472B2 (ru)
EP (1) EP2556073B1 (ru)
JP (1) JP5738978B2 (ru)
KR (1) KR101797066B1 (ru)
AR (1) AR081810A1 (ru)
BR (1) BR112012025718A2 (ru)
CA (1) CA2795523C (ru)
CO (1) CO6630131A2 (ru)
EA (2) EA023272B1 (ru)
MX (1) MX2012011637A (ru)
WO (1) WO2011124539A1 (ru)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA114410C2 (uk) * 2011-10-06 2017-06-12 Байєр Інтеллектуал Проперті Гмбх Гетероциклілпіри(mi)динілпіразол
RS58712B1 (sr) * 2015-06-29 2019-06-28 Astrazeneca Ab Derivati policikličnih amida kao cdk9 inhibitori
WO2018017633A1 (en) 2016-07-21 2018-01-25 Bristol-Myers Squibb Company TGF Beta RECEPTOR ANTAGONISTS
KR20230069963A (ko) * 2020-09-17 2023-05-19 얀센 파마슈티카 엔.브이. 카제인 키나아제 1 델타 조절제

Family Cites Families (45)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1037399B (de) 1955-03-23 1958-08-28 Erich Sulzmann Waschanlage zum Waschen und Spuelen von textilen Flaechengebilden
US4272417A (en) 1979-05-22 1981-06-09 Cargill, Incorporated Stable protective seed coating
US4245432A (en) 1979-07-25 1981-01-20 Eastman Kodak Company Seed coatings
US4808430A (en) 1987-02-27 1989-02-28 Yazaki Corporation Method of applying gel coating to plant seeds
GB8810120D0 (en) 1988-04-28 1988-06-02 Plant Genetic Systems Nv Transgenic nuclear male sterile plants
US5559137A (en) 1994-05-16 1996-09-24 Smithkline Beecham Corp. Compounds
PL186091B1 (pl) 1995-04-20 2003-10-31 American Cyanamid Co Wyizolowany DNA, wektor, komórka, warianty białkaAHAS, sposób nadawania oporności na herbicydy komórce, sposób wytwarzania opornego na herbicydy białka oraz sposoby zwalczania chwastów
US5876739A (en) 1996-06-13 1999-03-02 Novartis Ag Insecticidal seed coating
HUP0001880A3 (en) 1997-05-22 2002-03-28 G D Searle & Co Chicago Substituted pyrazoles as p38 kinase inhibitors
BR9809451A (pt) 1997-05-22 2000-06-20 Searle & Co Pirazóis substituìdos com 3(5)-heteroarila como inibidores de quinase p38.
US6087496A (en) 1998-05-22 2000-07-11 G. D. Searle & Co. Substituted pyrazoles suitable as p38 kinase inhibitors
US6979686B1 (en) 2001-12-07 2005-12-27 Pharmacia Corporation Substituted pyrazoles as p38 kinase inhibitors
US6514977B1 (en) 1997-05-22 2003-02-04 G.D. Searle & Company Substituted pyrazoles as p38 kinase inhibitors
US6503904B2 (en) 1998-11-16 2003-01-07 Syngenta Crop Protection, Inc. Pesticidal composition for seed treatment
CN1326848C (zh) 1998-12-25 2007-07-18 帝国脏器制药株式会社 氨基吡唑衍生物
JP4627944B2 (ja) 1999-06-03 2011-02-09 あすか製薬株式会社 置換ピラゾール化合物
US6978019B1 (en) 1999-06-30 2005-12-20 Silverbrook Research Pty Ltd Method and system for user registration on terminal
WO2001030154A2 (de) * 1999-10-25 2001-05-03 Basf Aktiengesellschaft Pyrazole enthaltende agrochemische zusammensetzungen und ihre verwendung als fungizide flanzenschutzmittel
US6660690B2 (en) 2000-10-06 2003-12-09 Monsanto Technology, L.L.C. Seed treatment with combinations of insecticides
DE60223339T2 (de) 2001-01-22 2008-08-28 Sankyo Co., Ltd. Durch bicyclische aminogruppen substituierte verbindungen
US20020134012A1 (en) 2001-03-21 2002-09-26 Monsanto Technology, L.L.C. Method of controlling the release of agricultural active ingredients from treated plant seeds
WO2002078701A1 (en) * 2001-03-30 2002-10-10 Smithkline Beecham Corporation Use of pyrazolopyridines as therapeutic compounds
WO2002088124A2 (en) 2001-04-27 2002-11-07 Smithkline Beecham Corporation Pyrazolo'1,5-a!pyridine derivatives
PT1397364E (pt) * 2001-05-24 2007-10-22 Lilly Co Eli Novos derivados de pirrole como agentes farmacêuticos
GB0129476D0 (en) 2001-12-10 2002-01-30 Syngenta Participations Ag Organic compounds
AU2003217712A1 (en) 2002-03-07 2003-09-22 Smithkline Beecham Corporation Pyrazolopyrimidine and pyrazolotriazine derivatives and pharmaceutical compositions containing them
US7304068B2 (en) 2002-05-10 2007-12-04 Smithkline Beecham Corporation Substituted pyrazolo [1,5-A] pyrimidinyls and pharmaceutical uses therefore
JP2005539000A (ja) 2002-07-31 2005-12-22 スミスクライン・ビーチャム・コーポレイション Ａｌｋ５阻害剤としての２−フェニルピリジン−４−イル誘導体
GB0217786D0 (en) 2002-07-31 2002-09-11 Glaxo Group Ltd Compounds
WO2004029043A1 (ja) 2002-09-25 2004-04-08 Ube Industries, Ltd. ピラゾール化合物
WO2005044194A2 (en) 2003-10-28 2005-05-19 Pharmacia Corporation TREATMENT OR PREVENTION OF NEOPLASIA BY USE OF AN Hsp90 INHIBITOR
CA2543503A1 (en) 2003-10-28 2005-05-12 Pharmacia Corporation Combinations comprising an hsp90 inhibitor and a phophodiesterase inhibitor for treating or preventing neoplasia
PL1910370T3 (pl) 2005-07-22 2015-09-30 Lilly Co Eli Monohydrat pirolo [1,2-b] pirazolu podstawionego pirydynochinoliną jako inhibitor tgf-beta
BRPI0615150A2 (pt) 2005-08-10 2017-06-20 Takeda Pharmaceuticals Co agente para a profilaxia ou tratamento de diabete, sensibilizador de insulina, composto, pró-droga, agente farmacêutico, e, uso do composto ou um sal do mesmo ou uma pró-droga do mesmo
NZ568867A (en) 2005-08-24 2010-12-24 Pioneer Hi Bred Int Compositions providing tolerance to multiple herbicides and methods of use thereof
EA015908B1 (ru) 2005-08-31 2011-12-30 Монсанто Текнолоджи, Ллс Инсектицидный белок в.thuringiensis cry1a.105, кодирующий его полинуклеотид и их применение
NL2000397C2 (nl) 2006-01-05 2007-10-30 Pfizer Prod Inc Bicyclische heteroarylverbindingen als PDE10 inhibitoren.
JP2009525350A (ja) 2006-02-01 2009-07-09 スミスクライン ビーチャム コーポレーション Ｒａｆキナーゼ阻害薬として有用なピロロ［２，３，ｂ］ピリジン誘導体
JP2009530261A (ja) 2006-03-16 2009-08-27 ファイザー・プロダクツ・インク ピラゾール化合物
KR20090031721A (ko) 2006-06-28 2009-03-27 아스카 세이야쿠 가부시키가이샤 염증성 장 질환의 처치제
DE102006037399A1 (de) 2006-08-10 2008-02-14 Archimica Gmbh Verfahren zur Herstellung von Arylaminen
US20080119457A1 (en) * 2006-08-24 2008-05-22 Serenex, Inc. Benzene, Pyridine, and Pyridazine Derivatives
GB0708141D0 (en) 2007-04-26 2007-06-06 Syngenta Participations Ag Improvements in or relating to organic compounds
CN101889012A (zh) * 2007-12-12 2010-11-17 杜邦公司 杀真菌二环吡唑
CN102105459B (zh) 2008-07-24 2014-09-10 内尔维阿诺医学科学有限公司 作为蛋白激酶抑制剂的3,4-二芳基吡唑类

Also Published As

Publication number Publication date
KR20130040843A (ko) 2013-04-24
BR112012025718A2 (pt) 2023-12-05
US20110251178A1 (en) 2011-10-13
EA023272B1 (ru) 2016-05-31
CN102947303A (zh) 2013-02-27
AR081810A1 (es) 2012-10-24
CA2795523A1 (en) 2011-10-13
WO2011124539A1 (de) 2011-10-13
CA2795523C (en) 2018-06-19
EP2556073A1 (de) 2013-02-13
CO6630131A2 (es) 2013-03-01
MX2012011637A (es) 2012-11-23
EP2556073B1 (de) 2014-07-23
JP2013523794A (ja) 2013-06-17
KR101797066B1 (ko) 2017-11-13
US8507472B2 (en) 2013-08-13
JP5738978B2 (ja) 2015-06-24
EA201291007A1 (ru) 2013-05-30

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