EA201391440A1 - Производные пиразолопиримидина - Google Patents

Производные пиразолопиримидина

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Publication number
EA201391440A1
EA201391440A1 EA201391440A EA201391440A EA201391440A1 EA 201391440 A1 EA201391440 A1 EA 201391440A1 EA 201391440 A EA201391440 A EA 201391440A EA 201391440 A EA201391440 A EA 201391440A EA 201391440 A1 EA201391440 A1 EA 201391440A1
Authority
EA
Eurasian Patent Office
Prior art keywords
pyrazolopyrimidine
derivatives
diseases
pyrazolopyrimidines
angiogenesis
Prior art date
Application number
EA201391440A
Other languages
English (en)
Inventor
Чжэнмин Ду
Раджендер Редди Лелети
Юйган Лю
Вольфганг Мильтц
Берндт Оберхаузер
Андреа Фаупель
Юрай Велцицки
Клаус Вайганд
Original Assignee
Новартис Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Новартис Аг filed Critical Новартис Аг
Publication of EA201391440A1 publication Critical patent/EA201391440A1/ru

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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  • Veterinary Medicine (AREA)
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Abstract

Настоящее изобретение относится к производным пиразолопиримидина, к способам их получения, к комбинациям и фармацевтическим композициям, включающим пиразолопиримидины, и к их применению в лечении заболеваний и расстройств, которые могут включать, например, аутоиммунные заболевания, ангиогенез, боль и/или воспалительные заболевания.
EA201391440A 2011-04-01 2012-03-30 Производные пиразолопиримидина EA201391440A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161470630P 2011-04-01 2011-04-01
PCT/IB2012/051554 WO2012131633A1 (en) 2011-04-01 2012-03-30 Pyrazolo pyrimidine derivatives

Publications (1)

Publication Number Publication Date
EA201391440A1 true EA201391440A1 (ru) 2014-03-31

Family

ID=45976462

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201391440A EA201391440A1 (ru) 2011-04-01 2012-03-30 Производные пиразолопиримидина

Country Status (17)

Country Link
US (1) US8748435B2 (ru)
EP (1) EP2694513B1 (ru)
JP (1) JP5963843B2 (ru)
KR (1) KR20140023331A (ru)
CN (1) CN103502248B (ru)
AR (1) AR085750A1 (ru)
AU (1) AU2012235665A1 (ru)
BR (1) BR112013025001A2 (ru)
CA (1) CA2831929A1 (ru)
EA (1) EA201391440A1 (ru)
ES (1) ES2534444T3 (ru)
MX (1) MX2013011421A (ru)
PL (1) PL2694513T3 (ru)
PT (1) PT2694513E (ru)
TW (1) TW201245203A (ru)
UY (1) UY33976A (ru)
WO (1) WO2012131633A1 (ru)

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