EA201300420A1 - Комбинации, которые содержат замещенный n-(2-ариламино) арилсульфонамид - Google Patents

Комбинации, которые содержат замещенный n-(2-ариламино) арилсульфонамид

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Publication number
EA201300420A1
EA201300420A1 EA201300420A EA201300420A EA201300420A1 EA 201300420 A1 EA201300420 A1 EA 201300420A1 EA 201300420 A EA201300420 A EA 201300420A EA 201300420 A EA201300420 A EA 201300420A EA 201300420 A1 EA201300420 A1 EA 201300420A1
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EA
Eurasian Patent Office
Prior art keywords
combination
component
arylamino
stereoisomer
solvate
Prior art date
Application number
EA201300420A
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English (en)
Inventor
Флориан Пюлер
Мэрион Хичкок
Original Assignee
Байер Интеллектчуал Проперти Гмбх
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44719990&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201300420(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Байер Интеллектчуал Проперти Гмбх filed Critical Байер Интеллектчуал Проперти Гмбх
Publication of EA201300420A1 publication Critical patent/EA201300420A1/ru

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    • A61K31/17—Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
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    • A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
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    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/4035—Isoindoles, e.g. phthalimide
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    • C07C275/40—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by nitrogen atoms not being part of nitro or nitroso groups
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  • Medicinal Preparation (AREA)

Abstract

Изобретение относится к комбинации, которая состоит из компонента А: одно или более омега-карбоксиарилзамещенное соединение дифенилмочевины общей формулы (I) или его физиологически приемлемая соль, сольват, гидрат или стереоизомер; компонента В: одно или более соединение N-(2-ариламино) арилсульфонамида общей формулы (II) или его физиологически приемлемая соль, сольват, гидрат или стереоизомер; и, необязательно, компонента С: одно или более дополнительное фармацевтическое средство; в которой необязательно некоторые или все компоненты находятся в виде фармацевтической лекарственной формы, которая готова к применению для введения совместно, одновременно, отдельно или последовательно; зависимо друг от друга, перорально, внутривенно, местно, с помощью локальных установок, внутрибрюшинно или через нос; применению такой комбинации для изготовления лекарственного препарата для лечения или профилактики рака, а также набору, который включает такую комбинацию.
EA201300420A 2010-10-01 2011-09-29 Комбинации, которые содержат замещенный n-(2-ариламино) арилсульфонамид EA201300420A1 (ru)

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PCT/EP2011/067041 WO2012041987A1 (en) 2010-10-01 2011-09-29 Substituted n-(2-arylamino)aryl sulfonamide-containing combinations

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GT201300085A (es) 2015-02-16
WO2012041987A1 (en) 2012-04-05
AU2011310532B2 (en) 2016-01-14
MX2013003695A (es) 2013-05-20
CA2813069A1 (en) 2012-04-05
AU2011310532A1 (en) 2013-04-18
EP2621486A1 (en) 2013-08-07
CR20130147A (es) 2013-05-29
CN103228274A (zh) 2013-07-31
AU2011310532A8 (en) 2014-02-20
KR20130099117A (ko) 2013-09-05
US9381177B2 (en) 2016-07-05
ECSP13012538A (es) 2013-06-28
NZ608584A (en) 2015-07-31
PE20140165A1 (es) 2014-02-26
DOP2013000070A (es) 2014-07-15
CL2013000881A1 (es) 2013-09-13
CO6690783A2 (es) 2013-06-17
AP2013006834A0 (en) 2013-04-30
US20130261120A1 (en) 2013-10-03
SG189038A1 (en) 2013-05-31
BR112013007835A2 (pt) 2016-06-28
MA34553B1 (fr) 2013-09-02
CU20130050A7 (es) 2013-07-31
UA112163C2 (uk) 2016-08-10
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